Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
11/2000
11/07/2000US6143747 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
11/02/2000WO2000064970A1 Antistatic agents and resin compositions incorporated therein
11/02/2000WO2000064864A1 N-protected amines and their use as prodrugs
11/02/2000EP1048694A1 Azo compounds and process for producing the same
11/02/2000EP1048656A2 Process for the preparation of hydantoins or cyclic anhydrides of an aminoacid
11/02/2000EP1048641A1 Apoptosis inducer
11/02/2000DE19919494A1 Ionische Flüssigkeiten, ihre Herstellung und ihre Verwendung Ionic liquids, their preparation and their use
11/02/2000CA2370317A1 Antistatic agents and resin compositions incorporated therein
11/02/2000CA2368205A1 N-protected amines and their use as prodrugs
11/01/2000CN1271728A Process for synthesizing allantoin
11/01/2000CN1058004C Heterocyclo-benzoylguanidin
11/01/2000CN1058003C Process for synthesis of 4-methyl iminazole
11/01/2000CN1057999C 4-Aminobenzoylguanidine derivatives
10/2000
10/31/2000US6140508 Useful in the preparation of farnesyl-protein transferase inhibitors.
10/31/2000US6140354 N-substituted aminotetralins as ligands for the neuropeptide Y Y5 receptor useful in the treatment of obesity and other disorders
10/31/2000US6140353 Used as medicaments for the treatment and/or prevention of thromboses, apoplexy, cardiac infarction, inflammation and arteriosclerosis or as antitumor agents
10/31/2000US6140331 For treating anxiety disorders, depression, psychosis, impulse control disorders, alcohol abuse, ischaemic diseases, cardiovascular disorders, side effects induced by conventional antipsychotic agents and senile dementia
10/31/2000US6139603 Process for recovering oxygen
10/26/2000WO2000063157A1 Disubstituted benzene derivatives
10/26/2000WO2000062778A1 Cyclic protein tyrosine kinase inhibitors
10/24/2000US6137007 Enantiomer compositions of (1R,4S)-1-butyrylamino-4-(hydroxymethyl)-2-cyclopentene
10/24/2000US6136983 Pesticidal sulfur compounds
10/24/2000US6136837 α-substituted benzyl heterocyclic derivatives, intermediates for producing the same and agrochemical composition containing the same as active ingredient
10/24/2000US6136829 Nitric oxide synthetase inhibitors
10/24/2000US6136378 Coating a water-based paints including a novel polyfunctional glyoxylated compounds curing agent; imparting wet adhesion properties, resist to corrosion, scavenging formaldehyde and as additives to primer formulations
10/19/2000WO2000061549A2 Pharmaceutical compounds
10/19/2000WO2000061541A2 Pharmaceutical compounds
10/19/2000WO2000061537A2 Pharmaceutical compounds
10/19/2000WO2000061134A1 Antimicrobial agents
10/19/2000CA2370425A1 Pharmaceutical compounds
10/19/2000CA2370406A1 Pharmaceutical compounds
10/18/2000EP1044962A1 Novel method of catalytic removal of protective group with allyl group
10/18/2000CN1270582A Imidazoline compounds
10/18/2000CN1270166A Derivatives of tricyclo-substituted isohydroxyloxime acid
10/18/2000CN1270062A Glycobiazole metal salt as synergist for radiotherapy or chemicotherapy and its preparing process and application
10/17/2000US6133303 Various indene derivatives, with the exception of 5-(2-imidazole-1-yl-ethoxy)indan-1-one; treating cancer and treating or preventing restenosis or atherosclerosis
10/17/2000US6133295 Pharmaceutical composition
10/17/2000US6133293 Insulin sensitivity enhancer in combination with other antidiabetics differing from the enhancer in the mechanism of action; potent depressive effect on diabetic hyperglycemia; 2,4-thiazolidinediones and oxazolidinediones
10/17/2000US6133291 3-(piperidin-1-ylalkylene)imidazole derivatives; glaucoma, antiallergens; antiinflammation and hypotensive agents, sleeping disorders; hypermotility of the gastrointestinal tract, alzheimer's disease, schizophrenia and
10/17/2000CA2074533C 2-nitroimidazole derivative, production thereof, and radiosensitizer containing the same as active ingredient
10/12/2000WO2000059906A1 Aminoheterocycle-substituted glycerols
10/12/2000WO2000059883A2 Method for producing n-aryl-aza-heterocycles in the presence of cesium carbonate
10/12/2000WO2000059880A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000WO2000059878A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
10/12/2000WO2000059867A1 Hydroxyphenyl derivatives with hiv integrase inhibitory properties
10/12/2000WO2000059855A1 Ether compounds, compositions, and uses thereof
10/12/2000WO2000059506A1 HETEROCYCLIC CONTAINING BIPHENYL aP2 INHIBITORS AND METHOD
10/12/2000WO2000059304A1 Compositions and methods for preventing and treating sexual dysfunctions
10/12/2000WO2000009106A3 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
10/12/2000CA2369238A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000CA2369005A1 Inhibitors of lfa-1 binding to icams and uses thereof
10/12/2000CA2360923A1 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
10/11/2000EP1043316A2 Nitroimidazole derivatives as sensitivity enhancers for chemotherapy and radiotherapy
10/11/2000EP1042313A1 Benzopyran and benzothiopyran derivatives having retinoid antagonist like activity
10/11/2000EP1042305A1 INHIBITION OF p38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS
10/11/2000EP1042301A1 Novel acylguanidine derivatives as inhibitors of bone resorption and as vitronectin receptor antagonists
10/11/2000EP1042279A1 Substituted beta-alanines
10/11/2000EP1042276A1 Thiourea and benzamide compounds, compositions and methods of treating or preventing inflammatory diseases and atherosclerosis
10/11/2000EP1042272A1 Derivatives of 2,2-dimethyl 3-(2-fluoro vinyl) cyclopropane carboxylic acid, their preparation process and their use as pesticides
10/11/2000EP1041980A1 Acyl guanidine sodium/proton exchange inhibitors and method
10/10/2000US6130226 Immunotherapeutic agents
10/05/2000WO2000058306A1 Substituted benzoylpyrazoles as herbicides
10/05/2000WO2000058293A2 Glucokinase activators
10/05/2000WO2000058286A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
10/05/2000WO2000057877A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
10/05/2000CA2368631A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
10/05/2000CA2368459A1 Substituted benzoylpyrazoles as herbicides
10/05/2000CA2361019A1 Process for the preparation of heterocyclic carbamates from aza-heterocycles and carbon dioxide
10/04/2000EP1041067A2 Use of 2-mercapto-imidazole derivatives substituted in position 4 ( or 5 ) as antioxidants
10/04/2000EP1041064A2 N-substituted alpha aminoacid amides as calcium channel modulators
10/04/2000EP1040112A1 Imidazonaphthyridines and their use in inducing cytokine biosynthesis
10/04/2000EP1040094A1 Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors
10/04/2000EP0766672B1 Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors
10/04/2000EP0569384B2 Fungicides
10/04/2000CN1268938A Aminocycloalkane compounds
10/04/2000CN1268510A 4-methylimidazole refining process
10/03/2000US6127568 Phenylacetic acid derivatives, preparation thereof and intermediates thereof, and compositions containing them
10/03/2000US6127548 Preparing optionally substitued 3h-imidazole-4-carbaldehyde by protecting the 3-amino group, then formylating in presence of an organometallic compound and electrophile with formyl leaving group, deprotecting with acid or strong base
10/03/2000US6127546 Process for the preparation of oxazoline compound
10/03/2000US6127396 Imidazoline compounds
10/03/2000US6127372 Sulfonamide inhibitors of aspartyl protease
10/03/2000US6127366 Inhibitors of farnesyl-protein transferase
09/2000
09/28/2000WO2000056718A1 Imidazole compounds
09/28/2000WO2000056685A1 Methods for the preparation of biphenyl isoxazole sulfonamides
09/28/2000WO2000056681A1 Thiourea and urea liquid-phase combinatorial libraries: synthesis and apoptosis induction
09/28/2000WO2000042971A3 Novel cationic 2-sulphonylaminophenols, their use as couplers for oxidation dyeing, compositions containing them and dyeing methods
09/28/2000DE19914140A1 Substituierte Benzoylpyrazole Substituted benzoylpyrazoles
09/28/2000DE19913483A1 Verfahren zur Herstellung von Heterocyclischen Carbamaten aus Aza-Heterocyclen und Kohlendioxid Process for the preparation of heterocyclic carbamates from carbon dioxide and aza heterocycles
09/28/2000CA2367916A1 Methods for the preparation of biphenyl isoxazole sulfonamides
09/28/2000CA2367857A1 Thiourea and urea liquid-phase combinatorial libraries: synthesis and apoptosis induction
09/27/2000EP1038864A1 Novel metalloproteinase inhibitors
09/27/2000EP1037905A1 Antipicornaviral compounds and methods for their use and preparation
09/27/2000EP1037883A1 NOVEL HETEROCYCLICALLY SUBSTITUTED $g(a)-HYDROXYCARBOXLIC ACID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
09/27/2000EP1037880A1 Retinoic acid mimetic anilides
09/27/2000EP1037868A2 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS
09/27/2000EP1037631A1 Heterocyclic cationic lipids
09/27/2000EP0885188B1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
09/27/2000EP0848703B1 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclo-oxygenase ii
09/27/2000CN1268120A Novel dihydronaphthalene compound and process and producing the same
09/27/2000CN1268116A 3-amidinoaniline derivatives activated blood coagulation factor X inhibitors, and intermediates for producing both