Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
01/2002
01/31/2002DE10035011A1 Pure N,N'-carbonyl-diazole preparation in high yield, by reacting azolide salt with phosgene in aromatic or ether solvent
01/31/2002DE10034802A1 Stabile Salze von O-Acetylsalicylsäure mit basischen Aminosäuren Stable salts of O-acetylsalicylic acid with basic amino acids
01/31/2002CA2417426A1 Efficient ligand-mediated ullmann coupling of anilines and azoles
01/31/2002CA2417127A1 Compounds and inhibitors of phospholipases
01/31/2002CA2416870A1 Potassium channel inhibitors
01/31/2002CA2416865A1 Potassium channel inhibitors
01/31/2002CA2415362A1 Method for treating fibrotic diseases or other indications
01/31/2002CA2415054A1 Cyanomethyl substituted thiazoliums and imidazoliums and treatments of disorders associated with protein aging
01/31/2002CA2410766A1 Novel imidazolidinones as ns3-serine protease inhibitors of hepatitis c virus
01/31/2002CA2410562A1 Colchinol derivatives as angiogenesis inhibitors
01/30/2002EP1176141A1 HETEROCYCLIC COMPOUNDS HAVING EFFECT OF ACTIVATING NICOTINIC ACETYLCHOLINE $g(a)4$g(b)2 RECEPTOR
01/30/2002EP1175406A1 Imidazoline derivatives as alpha-1a adrenoceptor ligands
01/30/2002EP1175383A1 Glucocorticoid receptor modulators
01/30/2002EP1175214A2 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
01/30/2002EP1175213A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
01/30/2002CN1333782A New derivatives of erythromycin, process for making them and use as medicaments
01/30/2002CN1333769A Thiourea inhibitors of herps viruses
01/29/2002US6342765 Imidazole derivatives and their use as farnesyl protein transferase inhibitors
01/29/2002US6342516 Phenylazole compounds, process for producing the same and drugs for hyperlipemia
01/29/2002US6342508 N-hydroxy-2-(Alkyl,Aryl or Heteroaryl sulfanyl, sulfinyl or sulfonyl) 3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
01/29/2002CA2094390C N-substituted imidazol-2-one compounds for treatment of circulatory disorders
01/24/2002WO2002006349A1 Gel compositions containing metronidazole
01/24/2002WO2002006215A1 3-arylsulfonyl-2-hydroxy-2-methylpropanoic acid derivates
01/24/2002WO2002005782A2 Stable salts of o-acetylsalicyclic with basic amino acids
01/24/2002WO2001058869A3 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
01/24/2002WO2001027107A3 Heterocyclic sodium/proton exchange inhibitors and method
01/24/2002US20020010338 Phenyl-keto-imidazolidine thioamide derivatives
01/24/2002US20020010173 Reacting an amide derivative with a piperidine containing guanidine group to produce the product
01/24/2002US20020009650 High electroconductivity
01/24/2002DE10130740A1 Malonic acid monoester and beta-keto-ester preparation from epoxide in high yield, for use as intermediates, by hydroesterification over cobalt compound catalyst followed by catalytic oxygenation
01/23/2002EP1174135A2 Pharmaceutical composition for use in treatment of diabetes
01/23/2002EP1173414A1 N-protected amines and their use as prodrugs
01/23/2002EP1173169A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof
01/23/2002CN1332723A Arylalkanoyl derivatives, processes for their preparation, their use and pharmaceutical compositions containing them
01/23/2002CN1332722A 2-substituted Retoamides
01/23/2002CN1332167A Eprosartan dihydrate and its prep.
01/22/2002US6340371 Cationic ortho-phenylenediamines, their use for the oxidation dyeing of keratin fibers, dye compositions and dyeing processes
01/22/2002CA2064872C Aryloxymethylcarbonochloridate ester intermediates, their production and use in synthesizing prodrugs and their use therefor
01/22/2002CA2049882C Process for iodinating or brominating the alpha-methylenic carbon of a secondary amide
01/22/2002CA2038848C Hydantoin derivatives
01/22/2002CA2027876C Use of substituted imidazoles
01/17/2002WO2002003912A2 Novel c-4 substituted retinoids
01/17/2002US20020007074 Imidazole derivatives having affinity for alpha2 receptors
01/17/2002US20020007062 Enyme inhibitors for treating neurodegenerative diseases; inhibition of lipidic peroxidation and nitrogen oxide synthase in warm-blooded animal; for treatment of cardiovascular/brain disorders
01/17/2002US20020007045 For inhibiting the aggregation of blood platelets; 3-(4-Aminomethyl-phenyl)-1-(2-(3,4-dichloro-phenyl)-2-hydroxy-ethyl)-1 -isopropyl-urea for example
01/17/2002US20020006951 Solid-state form of celecoxib having enhanced bioavailability
01/17/2002US20020006936 Anticancer agents; restenosis
01/17/2002US20020006929 Antiarrhythmia agent, antiproliferative agent
01/17/2002US20020006922 Metalloprotease inhibitors
01/17/2002DE10033337A1 Biphenylcarbonsäureamide, ihre Herstellung und ihre Verwendung als Arzneimittel Biphenylcarbonsäureamide, their preparation and their use as medicaments
01/17/2002DE10010984A1 Preparation of 2-phenyl-4,5-dihydro-oxazole-5-carboxylic acid derivatives, used as intermediates, by catalytic cyclization of N-benzoyl-aminoalkene compound
01/16/2002EP1019095B1 Method for the preparation of facial metal tricarbonyl compounds and their use in the labelling of biologically active substrates
01/16/2002EP0638075B1 Thiazole or imidazole derivatives as maillard reaction inhibitors
01/16/2002CN1331681A Synthesis of histamine dihydrochloride
01/16/2002CN1331680A N-aryl (thio) anthranilic acid amide derivatives, their prepn. and their use as VEGF receptor tyrosine kinase inhibitors
01/16/2002CN1077886C Amidino derivatives useful as nitric oxide synthase inhibitors
01/16/2002CN1077878C Prepn. of bicyclohexane derivative
01/15/2002US6339099 Guanidine mimics as factor Xa inhibitors
01/15/2002US6339082 Tricyclic compounds, preparation method and said method intermediates, application as medicines and pharmaceutical compositions containing same
01/15/2002US6339081 Composition and use
01/15/2002US6338960 Histamine measuring apparatus and a histamine measuring method
01/10/2002WO2002002567A1 Thienopyrrolidinones
01/10/2002WO2002002512A2 Compounds to treat alzheimer's disease
01/10/2002WO2002002218A1 Catalysis in an ionic fluid, supercritical fluid two phase system
01/10/2002US20020004512 Sexual disorders
01/10/2002US20020004503 Viricides
01/10/2002CA2414705A1 Thienopyrrolidinones
01/10/2002CA2410651A1 Compounds to treat alzheimer's disease
01/09/2002EP1170289A2 Retroviral protease inhibiting compounds
01/09/2002EP1170288A2 Diphenylureum derivatives and their use as alpha2/5-HT2c antagonists
01/09/2002EP1169312A2 Glucokinase activators
01/09/2002EP1169301A1 A topical antiandrogen for hair loss and other hyperandrogenic conditions
01/09/2002EP1169298A2 Pharmaceutical compounds
01/09/2002EP1169294A2 Pharmaceutical compounds
01/09/2002EP1169038A1 Cyclic protein tyrosine kinase inhibitors
01/09/2002EP1169031A1 Antimicrobial agents
01/09/2002CN1330640A Cyclic hydrazine derivatives as TNF-alpha inhibitors
01/09/2002CN1330064A Method for producing malonate derivative or beta-ket-acid ester by epoxide derivative
01/09/2002CN1077570C Sulfamate compounds containing N-substituted carbanoyl and process for preparing the same
01/08/2002US6337340 Carboxylic acids and isosteres of heterocyclic ring compounds having multiple heteroatoms for vision and memory disorders
01/08/2002US6337178 Quantitative analysis; measuring electrode potential
01/03/2002WO2002000659A2 Methods of synthesis for 9-substituted hypoxanthine derivatives
01/03/2002WO2002000647A1 Heteroaryl-phenyl substituted factor xa inhibitors
01/03/2002WO2001070693A3 Difluorobutyric acid derivatives and their use as metalloprotease inhibitors
01/03/2002WO2000061549A3 Pharmaceutical compounds
01/03/2002US20020002307 Process for the selective N-formylation of N-hydroxylamines
01/03/2002US20020002195 Pesticidal 1-polyarylpyrazoles
01/03/2002US20020002186 Pharmaceutical composition
01/03/2002DE10030893A1 New N-(2'-hydroxy-5'-aminobenzyl)-2-oxo- and -2-imino-thiazol(id)ine and -imidazol(id)ine compounds are used as developer component in oxidation colorant for keratin fibers, especially hair
01/03/2002DE10030685A1 Production of aliphatic sulfonic acid chlorides, useful for the production of agrochemicals, comprises reacting with phosgene in the presence of dimehtylformamide and a base or a sulfonic acid salt of a base
01/03/2002CA2409762A1 Heteroaryl-phenyl substituted factor xa inhibitors
01/02/2002EP1167356A2 Wet adhesion monomer and derived copolymers for latex paints
01/02/2002EP1166768A1 Use of ergothioneine and its derivatives as a glycation inhibitor
01/02/2002EP1165547A1 Substituted benzoylpyrazoles as herbicides
01/02/2002EP1165530A2 Dihetero-substituted metalloprotease inhibitors
01/02/2002EP1165512A2 Method for arylating aza-heterocycles with activated aromatic compounds in the presence of cesium carbonate
01/02/2002EP1165511A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
01/02/2002EP1165505A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
01/02/2002EP1165504A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
01/02/2002EP1165492A1 Hydroxyphenyl derivatives with hiv integrase inhibitory properties