Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
09/2002
09/12/2002WO2002070511A1 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
09/12/2002WO2002070493A1 Bisaryl derivatives having fsh receptor modulatory activity
09/12/2002WO2002070490A1 Agonists of beta-adrenoceptors
09/12/2002WO2002070473A2 Carboxamide derivatives as therapeutic agents
09/12/2002WO2002070469A2 Selective pde3b inhibitors and use of the same in therapy
09/12/2002WO2002070467A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments
09/12/2002WO2002069937A1 Compounds and compositions for delivering active agents
09/12/2002WO2002069901A2 Cathepsin cysteine protease inhibitors
09/12/2002WO2002069740A1 Compositions containing creatine and creatinine
09/12/2002WO2001096334A3 Heteroarylalkanoic acids as integrin receptor antagonists
09/12/2002US20020128315 Amidinophenol derivatives as leukotriene B4 (LTB4)antagonists, phospholipase A2 inhibitors, and trypsin inhibitors.
09/12/2002US20020128308 Useful as medicines having an osteogenesis promoting effect and chondrogensis promoting effect.
09/12/2002US20020128289 Insulin sensitivity enhancer in combination with other antidiabetics differing from the enhancer in the mechanism of action
09/12/2002US20020128263 Treatment or prevention of mGluR5 receptor mediated disorders.
09/12/2002US20020128255 Substituted hydroxyl amine derivatives; inhibitors of beta-secretase, inhibit beta-secretase-mediated cleavage, inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques
09/12/2002US20020127726 Karl fischer reagent
09/12/2002DE10111877A1 Neue Imidazolidinderivate, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate New imidazolidine derivatives, their preparation, their use and pharmaceutical compositions containing them
09/12/2002CA2439827A1 Peptide deformylase inhibitors
09/12/2002CA2438849A1 Compounds and compositions for delivering active agents
09/12/2002CA2437594A1 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
09/12/2002CA2434184A1 Bisaryl derivatives having fsh receptor modulatory activity
09/11/2002EP1237876A1 N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
09/11/2002EP1237875A1 Substituted imidazole neuropeptide y y5 receptor antagonists
09/11/2002EP1237874A2 Selective neurokinin antagonists
09/11/2002EP1237852A1 N-phenylcarbamates having a microbicide, insecticide and acaricide effect
09/11/2002EP1177199B1 Ionic liquids and production and use thereof
09/11/2002EP0813529B1 Arginine analogues having nitric oxide synthase inhibitor activity
09/11/2002CN1368962A Fluorene derivatives
09/11/2002CN1368958A Arylsulfonamido-substituted hydroxamic acid derivatives
09/10/2002US6448410 Production of compacted biocidal agent from particulate biocidal agent without using a binder
09/10/2002US6448373 Inhibitors of enzymes such as phospholipase a2; treatment of inflammatory diseases including atopic dermatitis and inflammatory bowel disease
09/10/2002US6448286 Imino pyrrolidine derivatives useful as nitric oxide synthase inhibitors
09/10/2002US6448282 1H-4(5)-substituted imidazole derivatives
09/10/2002US6448277 VEGF receptor tyrosine kinase inhibitors
09/06/2002WO2002068440A1 Glycopyranosyloxypyrazole derivatives and medicinal use thereof
09/06/2002WO2002068439A1 Glycopyranosyloxypyrazole derivatives and medicinal use thereof
09/06/2002WO2002068395A1 Hiv inhibiting n-aminoimidazole derivatives
09/06/2002WO2002068380A1 Synthetic excitatory amino acids
09/06/2002WO2002068377A1 Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells
09/06/2002WO2002068367A1 A method to inhibit ethylene responses in plants
09/06/2002WO2002067865A2 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof
09/06/2002WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors
09/06/2002CA2439053A1 Hiv inhibiting n-aminoimidazole derivatives
09/05/2002US20020123631 Reacting an aromatic or heteroaromatic carbamate with a heteroarylamine compound to form an intermediate, coupling the intermediate with an electrophile in suitable base and a catalyst
09/05/2002US20020123512 Pharmaceutical composition
09/05/2002US20020123491 Selective neurokinin antagonists
09/04/2002EP1236712A1 Amidinophenylpyruvic acid derivative
09/04/2002EP1235786A2 Method for the preparation of enantiomerically enriched compounds
09/04/2002EP1235776A1 Triphenylalkene derivatives and their use as selective estrogen receptor modulators
09/04/2002EP0920418B1 Substituted imidazolium salts and their use for the inhibition of protein ageing
09/04/2002EP0882043B1 Halogen pyrimidines and its use thereof as parasite abatement means
09/04/2002EP0644880B1 1,2,3-triazole and imidazole compounds and their antitumor use
09/04/2002CN1367785A Heterocyclic carboxamide-containing thiourea inhibitors of herpes viruses containing substituted phenylenediamine group
09/04/2002CN1367775A Cubane derivatives as metabotropic glutamate receptor antagonists and process for their preparation
09/04/2002CN1090178C Tricyclic compounds having activity specific for integrins, particularly alpha V beta 3 integrins, method for preparing same
09/04/2002CN1090177C Preparation of aromatic nitriles
09/03/2002US6444815 Method for producing heteroaromatic aldehydes
09/03/2002US6444704 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
09/03/2002US6444687 Eating disorders and diabetes
09/03/2002US6444615 Compounds effective as preemergent and postemergent herbicides
09/01/2002CA2356201A1 Compounds and compositions for delivering active agents
08/2002
08/29/2002WO2002067053A2 High speed photothermographic materials containing tellurium compounds and methods of using same
08/29/2002WO2002066672A2 Treatment of cns disorders using d-amino acid oxidase and d-aspartate oxidase antagonists
08/29/2002WO2002066442A1 Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
08/29/2002WO2002066431A1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
08/29/2002WO2002066425A2 Compositions and methods for hydration of terminal alkynes
08/29/2002WO2002066418A2 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor
08/29/2002WO2002039991A3 Prevention of development of dyskinesias
08/29/2002WO2001091807A3 Ethylenedicysteine (ec)-drug conjugates
08/29/2002WO2000067746A9 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
08/29/2002WO2000066104A9 Ace-2 inhibiting compounds and methods of use thereof
08/29/2002US20020120148 Benzocycloheptenylamino derivatives; treatment of pollakiuria or urinary incontinence
08/29/2002US20020120140 Phosgene-free process for preparing carbamates
08/29/2002US20020120007 Benzamide inhibitors of factor Xa
08/29/2002US20020119999 Imidazole dione or one, thione derivatives as antitumor and antiinflammatory agents, also treats cardiovascular disease, nephropathies and retinopathies
08/29/2002US20020119988 Modulators of TNF-alpha signaling
08/29/2002US20020119972 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases
08/29/2002US20020119963 Fertility; antidiabetic agents
08/29/2002CA2435446A1 Process for synthesis of heteroaryl-substituted urea compounds useful as antiinflammatory agents
08/29/2002CA2433866A1 Treatment of cns disorders using d-amino acid oxidase and d-aspartate oxidase antagonists
08/29/2002CA2432208A1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
08/28/2002EP1233936A1 Process for preparing ambient temperature ionic liquids
08/28/2002EP0885189B1 Method for the synthesis of poly-pyrrole and poly-imidazole carboxamides on a solid support
08/28/2002EP0861094B1 Gas/vapor delivery from solid materials
08/28/2002CN1366521A Substituted 1-aza-2-imino heterocycles and their use as nicotinic acetylcholine receptors activators
08/28/2002CN1365973A New cycloheplene compound, its preparation method and medicine composition containing same
08/27/2002US6441237 Drugs; antiarrhthymia agents, antiischemic agents
08/27/2002US6441189 Process for the preparation of matrix metalloproteinase inhibitors
08/27/2002US6441183 Useful as an intermediate in the preparation of certain small molecules that are useful in therapy or prophylaxis of inflammatory and immune cell-mediated diseases
08/27/2002US6441177 (4-bromo-phenyl)-(4-(6-(cyclopropyl-methyl-amino)-hexyloxy)-2-fluoro -phenyl)-methanone; antimycotic and cholesterol lowering activity
08/27/2002US6441172 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
08/27/2002US6441064 Imidazole-phosphoric acid salts as accelerators for dicyandiamide in one-component epoxy compositions
08/27/2002US6441023 For therapy of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone disease, diabetes (insulin resistance) and hiv infection
08/27/2002US6440965 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
08/27/2002US6440957 Cephalosporines having cyclic aminoguanidine substituents as antibiotics
08/22/2002WO2002064577A2 Method for preparing compounds derived from thiazolidinedione, oxazolidinedione
08/22/2002WO2002064570A1 Novel alkyl phenylimino-imidazolidine derivatives for treating urinary incontinence
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002WO2002064136A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
08/22/2002WO2002063957A2 Selective substituted aryl ketone and safener based herbicides