Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
04/2003
04/22/2003US6552030 Inhibit human factor Xa; treating thrombotic activity; 3-((3,5-difluoro-6-(3-(1-methylimidazolin-2-yl)phenoxy)-4-((2-(1,2 -dihydoxyethyl)-4-hydroxy-5-ethoxytetrahydrofuran-3-yl)oxy)-pyridin-2 -yl)oxy)4-hydroxybenzamidine
04/22/2003US6552022 Atherosclerosis in a mammal, pancreatitis, non-insulin dependent diabetes mellitus, coronary heart disease in a lowering serum lipid levels
04/22/2003US6551816 Enzymatic method for preparing synthesis intermediates
04/17/2003WO2003031437A1 Propylcarbamate derivatives as inhibitors of serine and cysteine proteases
04/17/2003WO2003031419A1 Substituted diphenyloxazoles, the synthesis thereof, and the use thereof as fluorescence probes
04/17/2003WO2003031414A1 Novel heterocyclic compound and anti-inflammatory agent
04/17/2003WO2003030889A1 Para-amino benzoic acids as integrin antagonists
04/17/2003WO2003030612A2 Methods for modulating activity of the fxr nuclear receptor
04/17/2003WO2003013484A3 N-monoacylated derivatives of o-phenylenediamines, their six membered heterocyclic analogues and their use as pharmaceutical agents
04/17/2003WO2003007887A3 Substituted imidazoles as cannabinoid receptor modulators
04/17/2003WO2000037430A3 Use of androgen receptor suppressors
04/17/2003WO1999064401A3 Imidazolyl derivatives and their use as somatostatin receptor ligands
04/17/2003US20030073862 Antidiabetic agents, anticancer agents, anticholesterol agents
04/17/2003US20030073853 Cationic aminoanthraquinones, their use for dyeing keratinous fibers, dyeing compositions containing them and methods of dyeing
04/17/2003US20030073850 Incontinence; nasal congestion
04/17/2003US20030073848 Accelerated process for preparing O-methyl phenols, N-methyl heteroaromatic compounds, and methylated aminophenols
04/17/2003US20030073847 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production
04/17/2003US20030073839 Compounds useful for preparation of Beta-3 adrenoreceptor agonist
04/17/2003US20030073836 Heteroarylcarboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions
04/17/2003US20030073835 Imidazolidinone derivatives
04/17/2003US20030073832 Novel aminophenyl ketone derivatives
04/17/2003US20030073723 Antiinflammatory agents; rheumatic diseases; antiallergens
04/17/2003US20030073712 Antiinflamamtory agents; antiischemic agents
04/17/2003US20030073669 N-heterocyclic derivatives as NOS inhibitors
04/17/2003US20030073641 Novel N-(arylsulphonyl) amino acid derivatives, process for their preparation and pharmaceutical compositions containing them
04/17/2003US20030070240 N-heteroarylmethyl-p-phnylendiamine derivatives and compounds containing oxidationcoloring agents
04/17/2003CA2462301A1 Para-amino benzoic acids as integrin antagonists
04/17/2003CA2462185A1 Methods for modulating activity of the fxr nuclear receptor
04/17/2003CA2462000A1 Substituted diphenyloxazoles, the synthesis thereof, and the use thereof as fluorescence probes
04/16/2003EP1302468A1 Processes and intermediates for manufacturing retroviral protease inhibiting compounds
04/16/2003EP1302461A1 Tnf-alpha production inhibitors
04/16/2003EP1301829A1 Radiation sensitive compositions containing image quality and profile enhancement additives
04/16/2003EP1301517A1 Thienopyrrolidinones
04/16/2003EP1301506A1 Cyclic amino acid derivatives
04/16/2003EP1301498A1 Colchinol derivatives as angiogenesis inhibitors
04/16/2003EP1301486A2 Imidazolidinones as ns3-serine protease inhibitors of hepatitis c virus
04/16/2003EP1301464A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
04/16/2003EP1255737A4 Process for preparing a 1-substituted 5-hydroxymethyl imidazole
04/16/2003EP1094812A4 Angiogenesis inhibitors
04/16/2003EP0998451B1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
04/16/2003EP0972769B1 Novel amide derivatives and medicinal compositions thereof
04/16/2003CN1411493A Method of colouring hair using cationic dyes
04/16/2003CN1411449A N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
04/16/2003CN1411447A Polymorphic crystalline forms of celecoxib
04/16/2003CN1411444A Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same
04/16/2003CN1411435A Novel use of phenyl hetero alkylamine derivatives
04/15/2003US6548671 Quinoxalinyl amide derivatives
04/15/2003US6548529 Heterocyclic containing biphenyl aP2 inhibitors and method
04/15/2003US6548512 Nitrogen containing heteroaromatics as factor Xa inhibitors
04/15/2003CA2290843C Cationic aminoanthraquinones, their use in the dyeing of keratin fibres, dyeing compositions containing them and dyeing processes
04/15/2003CA2103665C Oligopeptide antiretroviral agents
04/15/2003CA2097715C Indan derivatives
04/15/2003CA2051504C 1-phenyl-3-aryl-2-propyne-1-ones as calcium uptake inhibitors
04/10/2003WO2003029245A1 Spiro-hydantoin compounds useful as anti-inflammatory agents
04/10/2003WO2003029218A1 Novel nitrogenous compound and use thereof
04/10/2003WO2003029211A1 Difluoroalkene derivative, pest control agent containing the same, and intermediate therefor
04/10/2003WO2003029199A1 Benzene derivatives, process for preparing the same and use thereof
04/10/2003WO2003028728A1 4-(4-substituted piperazinyl-1yl)-butylcarboxamides as d3 dopamine subtype selective ligands
04/10/2003WO2003028721A2 Substituted benzimidazole compounds and their use for the treatment of cancer
04/10/2003WO2002078596A3 Novel dyeing composition for dyeing keratinous fibres comprising a particular dicationic diazo dye
04/10/2003WO2002042414A3 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
04/10/2003US20030069392 Cationic lipids
04/10/2003US20030069292 Central nervous system disorders; anticonvulsants
04/10/2003US20030069287 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
04/10/2003US20030069258 Novel guanidine mimics factor Xa inhibitors
04/10/2003US20030069257 Benzimidazole and pyridylimidazole derivatives
04/10/2003US20030069250 Anticoagulants
04/10/2003US20030069210 Especially imidazolyl- or 1,2,4-triazolyl- pyrimidine derivatives
04/10/2003US20030066988 Electroconductivity coloring
04/10/2003US20030066143 Cationic hair dye
04/10/2003CA2462112A1 Spiro-hydantoin compounds useful as anti-inflammatory agents
04/09/2003EP1300397A1 Compound for protective and anchor groups and its use
04/09/2003EP1300392A1 Process for producing optically active alpha-amino acid and optically active alpha-amino acid amide
04/09/2003EP1017681B1 Hydrazono-benzazulene derivatives, pharmaceutical compositions and intermediates
04/09/2003EP0934280B1 Pde iv inhibiting 2-cyanoiminoimidazole derivatives
04/09/2003EP0918746B1 Immunotherapeutic agents and their use in the reduction of cytokine levels
04/09/2003EP0901472B1 Mercapto-imidazolyl derivatives and their use as microbicides
04/09/2003EP0873123B1 Inhibitors of protein isoprenyl transferases
04/09/2003EP0771197B1 Use of heterocyclic compounds as dopamines-d 3- ligands
04/09/2003EP0724439B1 Use of 2-(2alkylphenylamino)oxazolines and -thiazolines for the manufacture of a medicament with alpha 2 adrenergic effect
04/09/2003CN1105114C Sulfonyl divalent aryl alpha-hydroxy-iso-hydroximic acid compounds
04/09/2003CN1105106C Naphthol derivatives and rpocess for preparation thereof
04/09/2003CN1104898C Ocular tension depressant
04/08/2003US6545163 Process to prepare 1-aryl-2-(1-imidazolyl) alkyl ethers and thioethers
04/08/2003US6545162 Solid phase biosynthesis of viricide antibiotic
04/08/2003US6545054 Alkenyl and alkynyl compounds as inhibitors of factor Xa
04/08/2003US6545018 Oxamic acids and derivatives as thyroid receptor ligands
04/08/2003US6545015 Useful in therapy of bacterial infections, fungal infections
04/08/2003US6545009 Retinoid-related receptor function regulating agent
04/08/2003US6544995 Use of cysteine derivatives for preparing a medicine for treating pathologies resulting from the formation of heterotrimeric G protein
04/08/2003US6544499 Polysiloxane or silicone resin, a linker, and a molecular hook for treating amino acid based substrates; hair care
04/08/2003US6544298 Dyeing human hair using coupler
04/08/2003CA2109830C Lhrh antagonists and intermediate products
04/08/2003CA2097824C Functionalized vinyl azoles and their use
04/08/2003CA2062271C Derivatives of substituted imidazol-2-one and process for their preparation
04/03/2003WO2003027130A2 Transition metal complexes for preparing olefin oligomers
04/03/2003WO2003027079A1 Ruthenium complexes, process for preparation thereof, and processes for producing open-ring polymers of cycloolefins and hydrogenation products thereof by using the complexes as catalyst
04/03/2003WO2003027076A2 1h-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1- antagonistic activity
04/03/2003WO2003027068A2 Substituted amines for the treatment of neurological disorders
04/03/2003WO2002101182A3 Solvent extraction mixture comprising substituted imidazole or benzimidazole for the separation of groups of base metals