Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
01/2015
01/14/2015EP2822925A1 Cf3o-containing enaminoketones and their utilization for the preparation of cf3o-containing pyrazoles
01/14/2015CN104277002A 甘氨酰胺衍生物、中间体、制备方法、药物组合物及应用 Glycinamide derivatives, intermediates, preparation methods, pharmaceutical compositions and applications
01/14/2015CN104277001A 1-烷基-3-卤代烷基吡唑-4-羧酸衍生物的区域选择性制备方法 1- alkyl-3-haloalkyl-pyrazole-4 regioselective preparation of carboxylic acid derivatives
01/14/2015CN104276960A 盐酸他喷他多和塞来昔布共晶及其组合物和制备方法 Tapentadol hydrochloride and celecoxib its eutectic composition and preparation methods
01/14/2015CN102844306B 吡唑羧酸酰胺的制备方法 Prepared pyrazole carboxylic acid amide
01/14/2015CN102193315B 着色感光性树脂组合物 The colored photosensitive resin composition
01/13/2015USRE45337 Ethers, secondary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
01/13/2015USRE45336 Primary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
01/13/2015US8933246 Process for preparing 1-phenylpyrazoles
01/13/2015US8933113 Mineralocorticoid receptor antagonists
01/13/2015US8933095 KAT II inhibitors
01/08/2015WO2015002119A1 Pyrazole-alcohol compound and pharmaceutical application therefor
01/08/2015WO2015002118A1 Fluorene-amide compound and pharmaceutical application therefor
01/08/2015WO2014153226A9 Arginine methyltransferase inhibitors and uses thereof
01/08/2015US20150011779 Method for producing 3,5-bis(fluoroalkyl)-pyrazol-4-carboxylic acid derivatives and 3,5-bis(fluoroalkyl)-pyrazoles
01/08/2015US20150011592 Substituted Phenylureas and Phenylamides as Vanilloid Receptor Ligands
01/08/2015US20150011565 Heterocyclic Compounds and Methods For Their Use
01/08/2015US20150011527 Novel glp-1 receptor modulators
01/07/2015EP2820006A1 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists
01/07/2015EP2819998A1 Crystalline forms of 1- (3 -tert-butyl- 1 - p-tolyl- 1h- pyrazol- 5 -yl) -3- (5-fluoro-2- (1- ( 2 - hydroxyethyl) - indazol- 5 -yloxy) benzyl) urea hydrochloride
01/07/2015EP2819997A1 Process for the preparation of phenyl substituted 3 - difluoromethyl - 1 -methyl - 1h - pyrazole - 4 - carboxylic n-methoxy- [1 -methyl- 2 - phenylethyl]amides
01/07/2015CN104262365A 含铜螺旋配位聚合物及其制备方法 Spiral copper coordination polymer and preparation method
01/07/2015CN104262294A 六氟异丙醇衍生物 Hexafluoroisopropanol derivatives
01/07/2015CN104262257A 一种吡唑衍生物的制备方法 A method for preparing pyrazole derivatives
01/07/2015CN104262256A 利用α,β-不饱和羰基化合物制备多取代吡唑类化合物的方法 The use of α, β- unsaturated carbonyl compound prepared poly-substituted pyrazole group compound
01/07/2015CN104262255A 一种不对称催化合成γ-硝基吡唑酰胺化合物的方法 One kind of amide compounds nitropyrazole way catalytic asymmetric synthesis of γ-
01/07/2015CN104262254A 一种具有双核铜簇的配位聚合物及其制备方法 A dual-core copper cluster coordination polymer and preparation method
01/07/2015CN104262253A 一种甲酰化方法 One kind formylation method
01/07/2015CN104262175A 调控相行为的离子液体及其制备方法和应用 Ionic liquid and its preparation method and application phase behavior regulation
01/07/2015CN102827082B 具有pde7抑制活性的噻吩并吡唑衍生物 Inhibitory activity having pde7 thieno-pyrazole derivative
01/07/2015CN102812008B 蓄尿障碍的治疗剂或预防剂 Urinary storage disorder therapeutic or prophylactic agent
01/07/2015CN102574778B 新的联苯基和苯基-吡啶酰胺类化合物 New biphenyl and phenyl - pyridine amides
01/07/2015CN102190622B 依达拉奉的水溶性衍生物及其制备方法和应用 Edaravone soluble derivatives, preparation method and application
01/07/2015CN102174035B 芳香双酰肼类plk1抑制剂及其用途 Aromatic double hydrazide plk1 inhibitors and their use
01/07/2015CN101875961B 用于预防和治疗相关病症而作为5-ht2a血清素受体调节剂的二芳基和芳基杂芳基脲衍生物 Diaryl and aryl-heteroaryl urea derivatives useful in the prevention and treatment of related disorders and as 5-ht2a serotonin receptor modulators
01/01/2015US20150005503 Method for preparing 2-aminobenzamide derivatives
01/01/2015US20150005500 Novel ruthenium catalysts and their use for asymmetric reduction of ketones
01/01/2015US20150005357 Substituted 4,5-Dihydro-2H-Benzo[e]Indazole-9-Carboxylates For The Treatment Of Diabetes And Related Disorders
01/01/2015US20150005345 Benzhydrol-pyrazole derivatives having kinase inhibitory activity and uses thereof
01/01/2015US20150005320 Compounds for inflammation and immune-related uses
01/01/2015US20150005293 5-Membered Heterocyclic Amides And Related Compounds
01/01/2015US20150005279 Primary carboxamides as btk inhibitors
01/01/2015US20150005232 Indazole derivatives
12/2014
12/31/2014CN104254523A 制备1-烷基-3-氟烷基-1h-吡唑-4-羧酸氯的方法 Preparation of 1-alkyl-3-fluoroalkyl -1h- pyrazole-4-carboxylic acid chloride method
12/31/2014CN102584706B 安乃近成品离心母液的回收工艺 Dipyrone finished centrifugal mother liquor recovery process
12/31/2014CN102399189B 一种3,4-二甲基吡唑磷酸盐的合成方法 A method of synthesis of 3,4-dimethyl-pyrazol-phosphate
12/30/2014US8921575 O-cyclopropylcyclohexyl-carboxanilides and their use as fungicides
12/30/2014US8921574 Method for producing pyrazolinone salt
12/30/2014US8921545 Synthesis of chiral 2-(1H-indazol-6-yl)-spiro[cyclopropane-1,3′-indolin]-2′-ones
12/30/2014US8921407 Pyrazole compounds that modulate HSP90 activity
12/30/2014US8921406 5-ring heteroaromatic compounds and their use as binding partners for 5-HT5 receptors
12/30/2014US8921402 Substituted pyrazoles as estrogen receptor ligands
12/30/2014US8921401 Pyrazole compounds, compositions and methods for treatment of degenerative diseases and disorders
12/30/2014US8921400 Arthropodicidal anthranilamides
12/30/2014US8921378 Androgen receptor modulating carboxamides
12/30/2014US8921364 Modulators of calcium release-activated calcium channel
12/30/2014US8921360 Heterobicycle-substituted azolyl benzene fungicides
12/25/2014US20140378474 5-membered heteroarylcarboxamide derivatives as plasma kallikrein inhibitors
12/25/2014US20140378466 Derivatives of n-(arylamino) sulfonamides as inhibitors of mek
12/25/2014US20140378461 Novel compounds
12/24/2014CN104245688A 活化ampk的吲哚和吲唑类化合物 Activation of indole and indazole compounds ampk of
12/24/2014CN104245677A 1-(3-叔丁基-1-对甲苯基-1h-吡唑-5-基)-3-(5-氟-2-(1-(2-羟乙基)-1h-吲唑-5-基氧基)苯甲基)脲盐酸盐的晶形 1- (3-tert-butyl-1-p-tolyl -1h- pyrazol-5-yl) -3- (5-fluoro-2- (1- (2-hydroxyethyl) -1h- indazole - 5- yloxy) benzyl) urea hydrochloride crystalline form
12/24/2014CN104245676A 用于制备3,5-双(氟烷基)吡唑-4-甲酸衍生物和3,5-双(氟烷基)吡唑类化合物的方法 Methods for the preparation of 3,5-bis (fluoroalkyl) pyrazole-4-carboxylic acid derivatives and 3,5-bis (fluoroalkyl) pyrazole compounds
12/24/2014CN104244713A 除草的亚磺酰亚氨酰基苯甲酰基衍生物和磺酰亚氨酰基苯甲酰基衍生物 Herbicidal sulfinyl imino group benzoyl derivative imide group and benzoyl derivative
12/24/2014CN104230904A 一类含萘环骨架的二氢吡唑磺胺衍生物的合成及在抗癌药物中的应用 Dihydropyrazolo synthesis of a class of sulfonamide derivatives of naphthalene skeleton and application of anti-cancer drugs
12/24/2014CN104230811A 一种吡唑吡啶化合物及其制备方法 Pyrazole pyridine compounds and methods
12/24/2014CN104230810A 大孔强酸性聚苯乙烯催化制备乙虫腈的方法 Preparation of strongly acidic macroporous polystyrene catalytic method ethiprole
12/24/2014CN104230809A 一种合成吡螨胺的工业化新工艺 Industrialization new process of synthesis tebufenpyrad
12/24/2014CN103025716B 二环化合物衍生物及其作为acc抑制剂的用途 Bicyclic compound derivative and its use as an inhibitor acc
12/24/2014CN102753527B 用作crf受体拮抗剂的环己基酰胺衍生物 Receptor antagonists used as crf cyclohexyl amide derivative
12/24/2014CN102690234B 具有取代基的苯基链烷烃酸的结晶和制造方法 And a method for producing a crystalline substituted phenyl paraffins acid
12/24/2014CN102464612B 含哌嗪氨基甲酸酯的二卤丙烯醚类化合物与应用 Piperazine-containing urethane dihalopropene ether compound and Applications
12/24/2014CN102382054B 异噁唑衍生物及其应用 Isoxazole derivative and Applications
12/23/2014US8916601 Aza-aryl 1H-pyrazol-1-YL benzene sulfonamides
12/23/2014US8916600 Phenyl and benzodioxinyl substituted indazoles derivatives
12/23/2014US8916598 Compounds, compositions, and methods for the treatment of β-amyloid diseases and synucleinopathies
12/23/2014US8916555 3,5-diaminopyrazole kinase inhibitors
12/23/2014US8916545 Pharmaceutical compositions comprising POH derivatives
12/18/2014US20140371467 Glucagon receptor modulators
12/18/2014US20140371261 Indomethacin analogs for the treatment of castrate-resistant prostate cancer
12/18/2014US20140371213 3,4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
12/18/2014US20140371202 Indazole compounds as kinase inhibitors and method of treating cancer with same
12/17/2014CN104220429A 非全身性tgr5激动剂 Non-systemic tgr5 agonist
12/17/2014CN104220426A 雌激素受体调节剂及其用途 Estrogen receptor modulators and their use
12/17/2014CN104220425A N-环烧基-n-[(环稀基苯基)亚甲基]-(硫代)羧酰胺衍生物 N- ring burn yl -n - [(cyclic dilute yl) methylene] - (thio) carboxamide derivatives
12/17/2014CN104220419A 含cf3o的烯胺酮和它们用于制备含CF30的吡唑类的用途 Enaminone and their containing cf3o for preparing pyrazoles containing CF30 use
12/17/2014CN104211705A 一种西地那非的制备方法 Method for preparing sildenafil
12/17/2014CN104211642A 一类含四氢化萘或色满骨架的二氢吡唑磺胺衍生物的合成及在抗癌药物中的应用 Dihydropyrazolo synthesis of a class of sulfonamide derivatives of tetralin or color full skeleton and application of anti-cancer drugs
12/17/2014CN104211641A 一种吡唑醚菌酯的合成工艺 A synthesis of pyrazole Kresoxim
12/17/2014CN102762540B 吡唑杀微生物剂 Pyrazole microbicides
12/17/2014CN101945855B I-苄基-3-羟基甲基吲唑衍生物及其在治疗基于MCP-1、CX3CR1和p40表达的疾病中的用途 I- benzyl-3-hydroxymethyl-indazole derivatives and their use in the treatment based on MCP-1, CX3CR1 and p40 expression in the diseases in
12/16/2014US8912342 Pyrazole synthesis by coupling of carboxylic acid derivatives and enamines
12/16/2014US8912202 N-(benzimimdazol-2-yl)-cyclopropane carboxamides as lysophosphatidic acid antagonists
12/11/2014US20140364623 Process for preparing acetanilides
12/11/2014US20140364622 Process for the stereoselective preparation of a pyrazole carboxamide
12/11/2014US20140364621 Electrically Conducting Oligo(pyrazoles)
12/11/2014US20140364603 Neprilysin inhibitors
12/11/2014US20140364398 C-Linked Hydroxamic Acid Derivatives Useful As Antibacterial Agents
12/10/2014CN104203921A 杀真菌剂n-环烷基-n-双环亚甲基-羧酰胺衍生物 Fungicides n- cycloalkyl -n- bicyclic methylene - carboxamide derivatives
12/10/2014CN104193693A 新除草剂 New Herbicide
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