Patents
Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931)
03/1994
03/08/1994CA1327524C Prostaglandins for use in medicine
03/03/1994WO1994004495A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
03/01/1994US5290936 Nitro substituted chemiluminescent labels and their conjugates, and assays therefrom
02/1994
02/23/1994CN1082536A Condensed bis-(3,4-dihydro-1-pyridinyl) methane and application of same in preparation of pharmaceutical
02/22/1994US5288726 Tetrahydrothienopyridine derivatives, furo and pyrrolo analogs thereof and their preparation and uses for inhibiting blood platelet aggregation
02/17/1994WO1994003437A1 Benzodiazepine derivatives
02/17/1994WO1994003426A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
02/17/1994CA2141791A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
02/17/1994CA2140009A1 Benzodiazepine derivatives
02/16/1994EP0582829A1 9-(substituted glycyl) amido - 6-demethyl-6-deoxytetracyclines as antibiotic agents
02/16/1994EP0582810A1 Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxyetracyclines as antibiotic agents
02/15/1994US5286894 Phenyl acrylic acid derivatives
02/15/1994US5286723 Bactericides
02/08/1994US5284952 Sulfonyl substituted chemiluminescent labels and their conjugates, and assays therefrom
02/08/1994US5284951 Hydrolytically stable chemiluminescent labels and their conjugates, and assays therefrom
02/03/1994WO1994002466A1 Unsymmetrical mono-3-nitro bis-naphthalimides as anticancer agents
02/01/1994US5283334 Side-chain functional chemiluminescent labels and their conjugates, and assays therefrom
01/1994
01/25/1994US5281712 Chemiluminescent aryl ester or thiolester of a carboxylic acid substituted heterocyclic ring
01/17/1994CA2074014A1 Chemiluminescent compounds
01/12/1994EP0577847A1 Morphinan derivative and medicinal use
01/12/1994EP0577753A1 Bis-naphthalimides containing amino-acid derived linkers as anticancer agents
01/12/1994CN1080639A Inhibitors of 5-alpha-testosterone reductase
01/06/1994WO1994000458A1 N-substituted 3-azabicyclo[3.2.0]heptane derivates useful as neuroleptic agents, etc.
01/06/1994WO1994000122A1 Use of condensed bis-(3,4-dihydro-pyridinyl)methane for treating crohn's disease, colitis ulcerosa, chronic inflamatory processes and as an antiproliferative
01/06/1994CA2138167A1 Use of condensed bis-(3,4-dihydro-1-pyridinyl)methanes for treating crohn's disease, ulcerative colitis, chronic inflammatory processes and as antiproliferative agents
01/04/1994US5276053 Dibenzothiopyranylamines
12/1993
12/29/1993EP0575526A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES
12/23/1993WO1993025527A1 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
12/23/1993DE4243287A1 N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung N-substituted Azabicycloheptan derivatives, their preparation and use
12/22/1993EP0287603B1 Sunscreen compositions and compounds for use therein
12/15/1993EP0574195A1 Antitumoral aza- and diazaanthracenes
12/09/1993WO1993024462A1 Substituted-hexahydrobenzo[a]phenanthridines
12/08/1993EP0572952A1 4-Benzylpiperidine derivatives, a process for preparing them and pharmaceutical compositions containing them
12/08/1993EP0572537A1 Cytokine inhibitors
12/07/1993US5268386 Certain 3,4-dihydro 4-oxospiro [2H-1 benzopyrans] useful for treating hyperuricemia
12/06/1993CA2097731A1 Antitumoral compounds
12/02/1993DE4217395A1 Prepn. of 2-acyl-1-aza:cyclo:alkene(s) useful as flavourings for bakery prods. - by intramolecular Aza-Wittig reaction using omega-azido:alkyl:di:ketone(s)
12/01/1993EP0572165A1 New 7B-substituted-4-aza-5a-cholestan-ones as 5a-reductase inhibitors
11/1993
11/30/1993US5266571 Treatment of hemorrhoids with 5-HT2 antagonists
11/25/1993WO1993023419A1 NEW 7β-SUBSTITUTED-4-AZA-5α-CHOLESTAN-ONES AS 5α-REDUCTASE INHIBITORS
11/25/1993WO1993023380A1 Bridged aza-bicyclic derivatives as substance p antagonists
11/23/1993US5264454 Certain 2-oxo-tetrahydro-cycloalkyl-benzopyran-3yl ureas having acyl-CoA-cholesterol acyl transferase inhibitory activity
11/21/1993CA2096576A1 7beta-substituted-4-aza-5alpha-cholestan-ones as 5alpha-reductase inhibitors
11/16/1993US5262425 α-mannosidase inhibitors
11/11/1993WO1993022286A1 Novel tetracyclic compound
11/02/1993US5258520 Process for preparing substituted 2-cyanopyridines
11/02/1993US5258386 Side effect reduction; nonhabit-forming
11/02/1993US5258384 S-11-hydroxy-10-methylaporphine and its biologically active salt forms as 5HT1A inhibitors
10/1993
10/28/1993WO1993021179A1 Novel amidoalkyl- and imidoalkyl-piperazines
10/28/1993WO1993021172A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
10/28/1993CA2109816A1 Novel amidoalkyl- and imidoalkyl-piperazines
10/27/1993EP0566567A1 Antihypertensive benzopyran derivatives
10/19/1993US5254564 Substituted isoquinoline compounds, pharmaceutical composition and method of use in treating pain in mammals
10/19/1993US5254561 Tricyclic antipsychotic agents
10/19/1993US5254478 Use in magnetometry by electronic paramagnetic resonance (EPR) of tetracyanoquinodimethane derivatives
10/13/1993EP0564648A1 Novel aconitine compound and analgesic/antiinflammatory agent
10/12/1993US5252699 Process for preparing 1-cyano-3H-dibenz[f,ij] isoquinoline-2,7-diones and their use as toners for polyesters
10/06/1993EP0564193A1 Heteroannulation process
10/05/1993US5250539 5-alpha reductase inhibitors; administer as therapy for benign prostatic hyperplasia, hirsutism and acne
10/04/1993CA2092782A1 Heteroannulation process
09/1993
09/30/1993WO1993019045A1 Arthropodicidal amides
09/30/1993WO1993018789A1 Non-azo naphthalimide dyes and uses for same
09/28/1993US5248677 Biogentic amine uptake inhibitors
09/28/1993CA1322522C Traumatic and ischemic brain injury treatment with opiate-receptor antagonists
09/14/1993US5245028 Process for preparing tetracyclic amines useful as cerebrovascular agents
09/14/1993US5244888 5-HT selective agents
09/02/1993WO1993014760A3 Methods
09/01/1993EP0558156A2 Intermediates for 3-aminopiperidine derivates
08/1993
08/31/1993US5240940 Quinoline and cinnoline fungicide compositions
08/31/1993US5240934 Quinoline derivatives
08/31/1993US5240464 Organic materials having sulfonamido linked poly(oxyalkylene) moieties and their preparation
08/24/1993US5239075 Process for the preparation of benzo (f) quinolinones
08/24/1993CA1321589C2 Intermediates for preparing benzo ¬5,6| cycloheptapyridines
08/10/1993US5235045 Viricides
08/10/1993US5234930 Pyrazolopyridine compounds which have useful pharmaceutical utility
08/05/1993WO1993014760A2 Methods
08/05/1993CA2128535A1 A method for delaying hiv induced aids by administration of substituted azaperane compounds
08/03/1993US5232927 Useful for enhancing memory
07/1993
07/24/1993WO1993015081A1 Morphinan derivative and medicinal use
07/22/1993WO1993014086A1 Substituted 1-isoquinolone derivatives as angiotensin ii antagonists
07/22/1993WO1993014066A1 Amino acid derivatives with anticholecystokinin activity
07/21/1993EP0551831A1 Process for the preparation of substituted pyridines 2-cyanopyridines
07/21/1993CN1074446A Tetrahydrothienopyridine derivatives, furo and pyrrolo analogs thereof and their preparation and uses for inhibiting blood platelet aggregation
07/20/1993CA1320488C 4-halogen-n-phenyl-3-pyridine-carboxamide compounds
07/16/1993CA2087315A1 Process for preparing substituted 2-cyanopyridines
07/14/1993EP0550444A1 Substituted naphthoxazines useful as dopaminergics
07/13/1993US5227383 Sampangine analogs
07/08/1993WO1993013069A1 Heterocycle-substituted benzylamine derivatives as antiretroviral compounds
07/08/1993CA2125675A1 Heterocycle-substituted benzenemethanamine derivatives
07/07/1993EP0550025A1 Azaspiroheptanes and octanes and processes for their production
07/07/1993CN1073942A Heterocycle-substituted benzenemethanamine derivatives
06/1993
06/29/1993US5223510 Alkylaminoalkyl derivatives of benzofuran, benzothiophene, indole and indolizine, process for their preparation and compositions containing them
06/29/1993US5223506 Cyclic antitumor compounds
06/24/1993WO1993012092A1 Highly water soluble bis-naphthalimides useful as anticancer agents
06/24/1993WO1993011761A1 Aryl-triflates and related compounds
06/24/1993CA2126242A1 Aryl-triflates and related compounds
06/24/1993CA2125142A1 Highly water soluble bis-naphthalimides useful as anticancer agents
06/23/1993EP0547224A1 14-O-p-CHLOROBENZOYLACONINE AND ANALGESIC/ANTIINFLAMMATORY AGENT
06/16/1993EP0546563A2 Complex crystal
06/15/1993US5220027 Sulfone-containing azamethide compounds with a nitrogen-containing aromatic ring of nitrogen containing aliphatic