| Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931) |
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| 07/24/2008 | WO2008087936A1 Condensed tetrahydroquinoline derivative and use thereof for medical purposes |
| 07/24/2008 | WO2008086678A2 The medical use of levo-phencynonate as neuroprotective agent |
| 07/24/2008 | WO2008055068A8 Inhibitors of histone deacetylase |
| 07/24/2008 | WO2008024497A3 INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE TYPE 1 |
| 07/24/2008 | US20080176899 Such as 1-Benzo[1,3]dioxol-5-yl-cyclopropanecarboxylic acid [5-(2-methoxy-pyridin-3-ylmethyl)-thiazol-2-yl]-amide 5-(2-Methoxy-pyridin-3-ylmethyl)-thiazol-2-ylamine; cystic fibrosis transmembrane conductance regulator disorders |
| 07/24/2008 | US20080176891 N-(2-Aminoethyl)-4-(2-ethyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzene-sulfonamide; respiratory disorders; rheumatoid arthritis |
| 07/24/2008 | US20080176869 e.g. N-(4-fluorobenzyl)-3-hydroxy-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-2-carboxamide; viricide in combination with other HIV/AIDS antivirals, immunomodulators, antibiotics or vaccines; AIDS |
| 07/24/2008 | US20080176841 (amidomethyl-amido)-(carboxy/amido)epoxide derivatives; cathepsin inhibitor; antiinflammatory, anticarcinogenic, antidiabeticagent, antiallergen, autoimmune and neurodegenerative disorders |
| 07/24/2008 | US20080176833 Dihydropyridine derivatives as useful as protein kinase inhibitors |
| 07/24/2008 | US20080175914 Inflammatory and/or allergic diseases; cognitive impairment |
| 07/23/2008 | EP1945615A2 Preparation of dutasteride |
| 07/23/2008 | EP1565464B1 4-oxo-1-(3-substituted phenyl-1,4-dihydro-1,8-naphthyridine-3-carboxamide phosphodiesterase-4 inhibitors |
| 07/23/2008 | EP1080092B1 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation |
| 07/23/2008 | CN101228160A Azaindoles useful as inhibitors of protein kinases |
| 07/23/2008 | CN101227903A Novel 3-spirocyclic indolyl derivatives useful as ORL-1 receptor modulators |
| 07/23/2008 | CN101225072A Heterocycle-containing organometallic complex and organic light emitting device including the same |
| 07/23/2008 | CN100404510C Enantioselective alkylation of tricyclic compounds |
| 07/22/2008 | US7402696 exert an ACC activity-inhibiting effect that is effective in the treatment of obesity, hyperlipemia, fatty liver, hyperglycemia, impaired glucose tolerance, diabetes, diabetic complications (diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, and diabetic macroangiopathy, hyperten |
| 07/22/2008 | US7402671 UV excitable fluorescent energy transfer dyes |
| 07/22/2008 | US7402592 Pharmaceutical compositions and methods for relieving pain and treating central nervous system disorders |
| 07/22/2008 | CA2238171C Quinoline derivatives as nk3 antagonists |
| 07/17/2008 | WO2008084496A1 Novel substituted 1h-benz [de] isoquinoline-1, 3 -diones |
| 07/17/2008 | WO2008029349A3 Muscarinic receptor antagonists |
| 07/17/2008 | US20080171874 Method for the regioselective preparation of substituted benzo[g]quinoline-3-carbonitriles and benzo[g]quinazolines |
| 07/17/2008 | US20080171863 Reacting fluorine salt containing radioactive fluorine-18 with alkyl halide or alkyl sulfonate in presence of alcohol; decreased reaction time; high yield; reduces the formation of side products |
| 07/17/2008 | US20080171788 N-(diaminomethylene)-9H-fluorene-2-carboxamide derivatives; dual antagonist for 5-HT2B and 5-HT7 receptors having selective binding affinities for 5-HT2B and 5-HT7 receptors; side effect reduction, nontoxic |
| 07/17/2008 | US20080171775 Ramipril-amlodipine salt |
| 07/17/2008 | US20080171765 e.g. 1-[3-(acridin-9-ylamino)-5-hydroxymethylphenyl]-3-{4-[bis(2-chloroethyl)amino]phenyl}urea; anticarcinogenic agent; improved chemical stability and efficacy; brain tumor, breast cancer, colon cancer, leukemia, and neuroblastoma |
| 07/17/2008 | US20080171763 Compounds and methods for treatment and prevention of diseases |
| 07/17/2008 | US20080171732 e.g. ethyl6-{4-[(benzylsulfonyl)carbamoyl]piperidin-1-yl}-5-cyano-2-methoxynicotinate; reversible and selective purinergic receptor antagonist; anticoagulant; cardiovascular diseases; platelet aggregation, thrombotic occlusion, myocardial infarction and unstable angina |
| 07/16/2008 | EP1944292A1 8-substituted-2,6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents |
| 07/16/2008 | EP1943250A1 Fused and spirocycle compounds and the use thereof |
| 07/16/2008 | CN100402529C Hydroxy alkyl substituted 1,3,8-triazaspiro[4.5]decan-4-one derivatives useful for the treatment of orl-1receptor mediated disorders |
| 07/16/2008 | CN100402528C Urea substituted imidazopyridines |
| 07/15/2008 | US7399768 1-methyl-3 beta -hydroxymethyl-6-methoxy-1,2,3,4,4a alpha ,5,10, 10a beta -octahydrobenzo[q]quinoline; decrease on the intraocular pressure; glaucoma and myopia; excellent tolerability, and a long duration of action |
| 07/15/2008 | CA2330669C Improved method for preparing pharmaceutically valuable norbenzomorphane derivatives |
| 07/10/2008 | WO2008082715A2 Sox-based kinase sensor |
| 07/10/2008 | WO2008080290A1 Selective m4 receptor antagonist and its medical use |
| 07/10/2008 | US20080167468 Silacycle compounds and methods of use thereof |
| 07/10/2008 | US20080167467 photovoltaics; emitters in chemiluminescence applications; field-effect transistors and electrophotography; N,N'-Bis(2,6-diisopropylphenyl)-1,7- and -1,6-bis(2,6-diisopropylphenoxy)-perylene-3,4:9,10-tetracarboximide |
| 07/10/2008 | US20080167334 Modulators of estrogen receptor alpha/beta G protein-coupled receptor 30, e.g., 1-(4-(6-Bromo-benzo[1,3]dioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl)1-ethanone; treating diseases such as cancer, neurodegenerative disorders, obesity, osteoporosis, and symptoms of menopause |
| 07/10/2008 | US20080167316 6-Heteroaryl-1,2,3,4,4A, 10B-Hexahydrophenanthridines as Pde4-Inhibitors for the Treatment of Inflammatory Disorders |
| 07/10/2008 | US20080167307 Carboxylic Acid Derivative Containing Thiazole Ring and Pharmaceutical Use Thereof |
| 07/10/2008 | US20080167306 Novel Heteroaryl Derivative |
| 07/10/2008 | US20080167301 Novel Hydroxy-6-Heteroarylphenanthridines and Their Use as Pde4 Inhibitors |
| 07/10/2008 | US20080167288 Substituted cyclic hydroxamates as lnhibitors of matrix metalloproteinases |
| 07/09/2008 | EP1942110A1 Preparation of clopidogrel and its analogues methyl tetrahydrothienopyridine acetate compounds |
| 07/09/2008 | EP1940401A2 Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators |
| 07/09/2008 | EP1421068B1 A process of synthesis of a tricyclic ketone intermediate |
| 07/09/2008 | EP1332133B1 Metabotropic glutamate receptor antagonists |
| 07/09/2008 | EP0984969B1 Fused dihydropyrans |
| 07/09/2008 | CN100400601C Thermochromic rylene dyes |
| 07/09/2008 | CN100400515C Isoquinoline derivatives and methods of use thereof |
| 07/09/2008 | CN100400514C 9-cyano-substituted perylene-3,4-dicarboxylic acid monoimides |
| 07/08/2008 | US7396930 making spiro(benzo(c)thiophene-1 (3H),4'-piperidine) derivatives; involves reacting a mercapto compound with a 2-halophenylalkyl halide, reacting with an alkyllithium, then N-ethoxycarbonyl-4-piperidone, dehydration and cyclization; industrial scale; novel intermediates to neurokinin receptor antagonist |
| 07/08/2008 | US7396844 3-(4-amidinobenzoylamino)-4-[5-amidino-2-(2-carboxy-2-oxoethyl)phenoxy]butanoic acid; anticoagulant; blood coagulation factor X and thrombin inhibitor; cerebral infarction, thrombosis, embolism, transient ischemic attack (TIA) and subarachnoidal hemorrhage (vasospasm); ischemic heart diseases |
| 07/03/2008 | WO2008078824A1 Benzofluoranthene compound and organic light-emitting device using the compound |
| 07/03/2008 | WO2008056059A3 4-azasterol derivatives, methods for the synthesis thereof and use of same as drugs |
| 07/03/2008 | WO2007118151A3 Spirocyclic heterocyclic derivatives and methods of their use |
| 07/03/2008 | US20080161569 Dimerizing a naphthalene-1,8-dicarboximide, reoxidation of the resulting perylene-3,4:9,10-tetracarboxylic diimide, hydrolyzing the diimide to the tetraalkali metal salt of perylene-3,4:9,10-tetracarboxylic acid, convert it into perylene-3,4:9,10-tetracarboxylic dianhydride |
| 07/03/2008 | US20080161339 Novel Thio-Containing Hydroxy-6-Phenylphenanthridines and their Use as Pde4 Inhibitors |
| 07/03/2008 | US20080161303 Imidazo- and triazolo-pyridine compounds and methods of use thereof |
| 07/03/2008 | US20080161281 Amino-Substituted Tricyclic Derivatives and Methods of Use |
| 07/02/2008 | EP1939170A1 Process for the preparation of gabapentin hydrochloride |
| 07/02/2008 | EP1937268A2 Indenoisoquinolinone analogs and methods of use thereof |
| 07/02/2008 | EP1539166B1 Pharmaceutical compositions comprising dextromethorphan and quinidine for the treatment of neurological disorders |
| 07/02/2008 | CN101209994A Selectivity M4 acceptor antagonist and medical use thereof |
| 07/02/2008 | CN101209993A Medical use for levorotatory phencynonate as nerve protecting agent |
| 07/02/2008 | CN100398519C Tetracyclic benzamide derivatives and methods of use thereof |
| 07/01/2008 | US7393956 Dimerization of naphthalene-1,8-dicarboximide in aprotic solvent and alkali base |
| 07/01/2008 | US7393955 Synthesis and use of tetracyclic benzamide derivatives; antidiabetic agents; coupling isochromene anhydride with cyanobenzene compound and performing ring substitution reactions |
| 06/26/2008 | WO2008076427A2 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof |
| 06/26/2008 | US20080154040 Azafluorene derivative and organic light-emitting device using the derivative |
| 06/26/2008 | US20080153868 Substituted Tetrahydroisoquinolines as Beta-secretase Inhibitors |
| 06/26/2008 | US20080153863 Spiropiperidine derivatives |
| 06/26/2008 | US20080153862 Vasopressin receptor (V1a) antagonists, treatment of anxiety and depressive disorders and other diseases |
| 06/26/2008 | US20080153861 Vasopressin receptor (V1a) antagonists, treatment of anxiety and depressive disorders and other diseases |
| 06/26/2008 | US20080153860 3H-(4's)-1'-azaspiro[benzofuran-2,4']-tricyclo[3.3.1.13,7]decane; for therapy of memory disorder, cognitive disorder, neurodegeneration, and neurodevelopmental disorder; attention deficit disorder, attention deficit hyperactivity disorder (ADHD), Alzheimer's disease (AD), mild cognitive impairment |
| 06/26/2008 | US20080153809 Novel amides useful for treating pain |
| 06/25/2008 | EP1934184A1 3 -azabicyclooctane derivatives as muscarinic receptor antagonists |
| 06/25/2008 | CN101208341A Hexarylene and pentarylene tetracarboxylic acid diimides |
| 06/24/2008 | US7390901 Fluorinated dyes or colorants and their uses |
| 06/24/2008 | US7390818 3-(2,4-dimethoxyphenyl)-1,9-dimethyl-2-oxo-2,9-dihydro-1H-pyrido[2,3-b]indole-6-carboxylic acid; gamma-aminobutyric acid modulator; anticarcinogenic, antitumor, antiproliferative agent |
| 06/19/2008 | WO2008073613A2 Materials and methods for co-crystal controlled solid-state synthesis of imides and imines |
| 06/19/2008 | WO2008072850A1 Triazine derivatives having inhibitory activity against acetyl-coa carboxylase |
| 06/19/2008 | US20080146805 dissolving the morphinan in the biphasic mixture, extracting the organic layer including the morphinan with a water soluble amine base, isolating the morphinan, forming a salt of the morphinan, crystallizing |
| 06/19/2008 | US20080146606 Novel compounds |
| 06/19/2008 | US20080146605 Preparation and utility of ccr5 inhibitors |
| 06/19/2008 | US20080146588 Piperidinyl Piperidine Tachykinin Receptor Antagonists |
| 06/19/2008 | US20080146580 Anititumoral Ecteinascidin Derivatives |
| 06/19/2008 | US20080146564 the major cause of lower respiratory tract illness during infancy and childhood |
| 06/19/2008 | US20080146563 1,7-Naphthyridines as Pde4 Inhibitors |
| 06/19/2008 | US20080146546 Bicyclic and Tricyclic Heteroaromatic Compounds |
| 06/19/2008 | US20080146536 2-Aminoimidazopyridines for treating neurodegenerative diseases |
| 06/19/2008 | CA2668464A1 Materials and methods for co-crystal controlled solid-state synthesis of imides and imines |
| 06/18/2008 | EP1931638A1 Process for the synthesis of compounds for selectin inhibition |
| 06/18/2008 | EP1931637A2 Methods of modulating neurotrophin-mediated activity |
| 06/18/2008 | CN101203495A Benzocycloheptapyridines as inhibitors of the receptor tyrosine kinase met |
| 06/17/2008 | CA2383114C Substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines and their use as pharmaceutical compositions |
| 06/17/2008 | CA2302347C 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-oles, processes for their preparation and their use for medicaments |