Patents
Patents for C07D 221 - Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups (10,931)
07/1980
07/22/1980US4214085 Analgesics, narcotic antagonists
07/15/1980US4212973 From cyclopentanone-cyanoacetamide-cyanoacetate reaction product(s) with basic catalyst via b,b-tetramethylene-a,a'-dicyanoglutarimide intermediate
07/08/1980CA1081214A1 Process for preparing an intermediate for cns depressants
07/01/1980CA1080705A1 Azabicycloalkanes and precursors thereof
07/01/1980CA1080704A1 6,7-benzomorphan derivatives, methods for their preparation and novel intermediates
06/1980
06/25/1980EP0012170A1 7-Phenyl-quinolizidine derivatives (I), their preparation, pharmaceutical compositions containing them and (I) for use in treating diseases
06/17/1980US4208523 Narcotics, analgesics
06/17/1980CA1079734A1 1-(3,3,3,-triarylpropyl)-4-phenyl-4-piperidinemethanols
06/17/1980CA1079726A1 2'-hydroxy-2-(5-isoxazolylmethyl)-6,7-benzomorphanes, their acid addition salts and pharmaceutical comprising same
06/10/1980US4207107 Use in recording information
06/10/1980CA1079273A2 Preparation of 2;6-methano-benzazocines
06/03/1980US4206225 Analgesics
06/03/1980US4206117 Pyridinyl aminoalkyl ethers
05/1980
05/28/1980EP0011483A1 Azocine compounds suitable as analgesics, and process for their production
05/28/1980EP0011255A1 1,2,3,4-Tetrahydro-6-oxo-2,8a-methano-6H-dibenz(c,e)-azocines, medicaments containing them, and process for their preparation
05/27/1980US4205172 7,10-Dichloro-3-methyl-4-phenyl-1,2,3,4-tetrahydrobenz[H]isoquinoline hydrobromide
05/27/1980US4205171 Aminomethanobenzazocines and nitromethanobenzazocines
05/27/1980CA1078389A1 (2-azabicyclo (2.2.2) octan-2-yl) diphenylalkanones and related compounds
05/20/1980US4204063 N(Aminoalkyl)-naphthalimides and their derivatives
05/15/1980WO1980000963A1 Aromatic compounds and their manufacture
05/14/1980EP0010994A1 Process for producing substituted naphthalic acid compounds
05/13/1980US4202984 Analgesics
05/13/1980US4202983 11-(Lower-alkoxy- and lower-alkylthio-3-oxo-lower-alkyl)-hexahydro-2,6-m ethano-benzazocines
05/13/1980US4202982 Process for the preparation of 14-hydroxymorphinan derivatives
05/13/1980US4202980 Process for the preparation of 1-hydroxyaporphine-derivatives
05/06/1980US4201862 Neuroleptic agents
05/06/1980CA1077042A1 (?)-4-hydroxy-1,2,9,10-tetraalkoxy-aporphine derivatives
04/1980
04/29/1980US4200752 Fluorescent dyes
04/29/1980US4200636 Muscle relaxant
04/22/1980CA1076116A1 Homophthalimides carrying amino substituents in the 2-position
04/22/1980CA1076111A1 6-aryl-s-triazolo-(4,3-a)-pyrido-(2,3-f)-1,4-diazepines
04/15/1980US4198415 Dopamine agonists, treatment of parkinsonism
04/08/1980US4197241 Analgesics
04/08/1980US4197239 Hexahydroazepine, piperidine and pyrrolidine derivatives
04/08/1980US4197111 1,8-Naphthalimides and herbicide antidotes
04/03/1980WO1980000566A1 N-substituted-6-oxamorphinans
04/02/1980EP0009386A1 2,10-Disubstituted dibenzo(b,d)pyrans and benzo(c)quinolines and pharmaceutical compositions thereof
04/02/1980EP0009290A1 3-Azabicyclo(3.1.0)hexane derivatives and process for their preparation
04/02/1980EP0009227A1 Fluorination process and fluoro analogs of hydrocodone and oxycodone
04/02/1980EP0009140A1 Polyalkyl-dihydroxy piperidines and process for their preparation
04/01/1980CA1074793A1 8-alkyl-5-oxo-5,8-dihydro-pyrido(2,3-d) pyrimidine-6-carboxylic acids and their preparation
03/1980
03/25/1980CA1074320A2 1'-hydroxy-5-lower alkoxy-2-lower alkyl-7,8-cyclopentano (h)-1,2,3,4-tetrahydroisoquinoline
03/25/1980CA1074310A1 Benzomorphane derivatives
03/18/1980US4194044 Process for preparing 3-phenoxy morphinans
03/18/1980US4193998 1,2,3,4,6,7-Hexahydro-11BαH-benzo[a]quinolizine-derivatives
03/18/1980CA1073912A1 Derivatives of dibenzo (de,h) quinolein; their preparation and compositions thereof
03/04/1980US4191683 Derivatives of 4-aminopiperidine as stabilizers for polymers
02/1980
02/21/1980WO1980000215A1 Medicament against glaucoma
02/19/1980US4189583 Synthesis of 4A-aryl-decahydroisoquinolines
02/19/1980CA1072089A1 1,1,1 triaryl alkylamines
02/12/1980US4188392 Antimicrobial compositions
01/1980
01/29/1980CA1070686A1 2-substituted-9-phenyl-2,3,4,4a,9,9a-hexahydro-1h-indeno(2,1-c) pyridines and related compounds
01/22/1980US4185119 Antiallergic methods
01/22/1980CA1070311A1 N-(1-((1,3-dihydro-1,3-dioxo-2h-benz(de) isoquinolin-2-yl)-alkyl)-4-piperidinyl)-n-phenylalkylamides
01/09/1980EP0006449A1 2-(2-Alkoxyethyl)-2'-hydroxy-6.7-benzomorphane derivatives, their acid addition salts, medicaments containing them and process for their preparation
01/01/1980US4181659 Bis-penicillanoyloxy-alkanes
12/1979
12/25/1979US4180667 2-Azabicyclo[2.2.2]oct-5-enes
12/25/1979US4180666 3,9-Dihydro-3,9-dioxo-2H-indeno(2,1-c)-pyridine-4-(carbonitriles/carboxamides)
12/25/1979US4180579 2-Substituted-1H-benz[de]-isoquinoline-1,3(2H)-diones
12/25/1979CA1068705A 2-(substituted-piperidinyl or tetrahydro-pyridinyl)alkyl)-1h-benzs(de) isoquinoline-1,3(2h)-diones
12/25/1979CA1068703A 2-((substituted piperazinyl, piperidinyl or tetrahydropyridinyl)-alkyl)-2,3-dihydro-3-hydroxy-1h-benz (de) isoquinolin-1-ones
12/18/1979CA1068285A1 6-oxatetracycline and 6-thiatetracycline compounds and process for their preparation
12/18/1979CA1068279A1 2,4,5-trimethyl-thieno (3,2-f) morphan, and intermediates
12/18/1979CA1068267A1 Benzazocine derivative
12/04/1979US4177275 Antihistamine, antiserotonine
10/1979
10/31/1979EP0004960A1 9.9-Dimethyl-6.7-benzomorphan derivatives, processes for their preparation and pharmaceutical compositions comprising them
10/23/1979US4172202 Process for the preparation of 4-amino-1,8-naphthalimides
10/23/1979CA1064923A1 N-acyl-n-norsalutaridines and process for making them
10/16/1979CA1064486A1 Aminobenzazocines and preparation thereof
10/09/1979US4170651 Antiinflammatory agents
10/03/1979EP0004260A1 Substituted quinolizidine and indolizidine-methanol derivatives, method for their preparation and medicaments containing them
10/02/1979US4169893 4-hydroxy-naphthpyridine-2(1h)-one-3-carboxylic acids and esters
09/1979
09/25/1979US4169200 Substituted 3,6-dihydro-1(2H)-pyridinylpropanols
09/25/1979CA1063118A1 5 ou l'-hydroxy-2-alkyl-7,8-cyclopentano (h)-1,2,3,4-tetrahydroisoquinolines and esters
09/25/1979CA1063117A1 Cyclopentano (h) or (f) 1,2,3,4-tetrahydroisoquinolines
09/25/1979CA1063116A1 L'-substituted amino-2-alkyl-5-hydroxy-7,8-cyclopentano (h)-1,2,3,4-tetrahydroisoquinolines
09/25/1979CA1063105A1 Aminobenzazocines and preparation thereof
09/19/1979EP0004255A2 4-Hydroxy-naphthopyridin-2(1H)-3-one carboxylic acids, their esters, process for their preparation, and pharmaceutical compositions containing them
09/18/1979US4168379 Pyridin-3-ols
09/18/1979US4168311 Aphidicides
09/18/1979CA1062616A1 Analgetic composition containing an indole-3-acetic acid derivative
09/04/1979CA1061791A1 N-substituted-7,8-dihydroxycyclopentano(f)-1,2,3,4-tetrahydroisoquinolines and ethers and esters thereof
09/04/1979CA1061790A1 N-substituted-5,6-dihydroxycyclopentano(h)-1,2,3,4-tetrahydroisoquinolines and ethers and esters thereof
08/1979
08/28/1979US4166183 Tricyclic cyclitolamines
08/28/1979US4166174 Analgesics
08/08/1979EP0003278A1 Polysubstituted-2-(3-loweralkylamino-2-R0-propoxy)pyridines, process for preparing the same, and pharmaceutical compositions containing the same
08/08/1979EP0003258A1 Preparation of N-chloroimides and a novel N-chloroimide
08/08/1979EP0003253A1 Hexahydroazepine, piperidine and pyrrolidine derivatives and processes for making and using them
08/07/1979US4163853 1-(P-phenoxy)benzyl-1,2,3,4,5,6,7,8-octahydroisoquinolines
08/07/1979US4163841 Pyridylamides of nitriloprostacyclins
07/1979
07/24/1979US4162361 Morphine/apomorphine rearrangement process
07/24/1979CA1059126A1 Benzo/a/quinolisidine derivatives and a process for the preparation thereof
07/17/1979US4161598 Analgesics, narcotic antagonists
07/17/1979US4161597 Neutralization, decarboxylation, amidation, rearrangments
07/17/1979US4161584 Cycloamides of nitriloprostacyclins
07/11/1979EP0002937A1 Novel pyrindines and their preparation, formulations and use
07/10/1979US4160844 Composition for treating skin mast cells and/or delayed cellular hypersensitivity reactions
07/10/1979CA1058178A1 2-((substituted-piperazinyl)alkyl)-1h-benz(de)isoquinoline-1,3(2h)-diones
07/03/1979US4160094 Tetrahydroquinoline derivatives
07/03/1979CA1057755A1 Heterocyclic compounds, their preparation and compositions thereof_