Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
05/2008
05/21/2008EP1362027B1 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
05/20/2008US7375227 May be combined with ACE inhibitors, angiotensin or endothelin receptor antagonists, vasopressin antagonists, alpha- and beta-adrenergic antagonists, TNFalpha antagonists, and peroxisome proliferator activator receptor modulators; cardiovascular, renal, metabolic, pulmonary and psychological disorders
05/20/2008US7375218 highly convergent and this convergency manifests itself in a much shorter synthetic sequence
05/20/2008US7375134 N1-(1-cyanocyclopropyl)-4-fluoro-N2-{(1S)-2,2,2-trifluoro-1-[4'-(methylsulfonyl)-1,1'-biphenyl-4-yl]ethyl}-L-leucinamide; osteoporosis and other bone loss disorders
05/20/2008US7375099 Malonamide derivatives
05/20/2008CA2395717C Fused imidazolium derivatives
05/20/2008CA2322309C Quinolin-4-yl derivatives
05/15/2008WO2008058118A2 Preparation of montelukast and its salts
05/15/2008WO2008056148A1 Chemical compounds
05/15/2008WO2008023333A3 Process for the preparation of 4-(isobutylamino)-3-amino-quinoline
05/15/2008WO2007138112A3 Compounds that interact with ion channels, in particular with ion channels from the kv family
05/15/2008US20080113975 Thiourea compounds
05/15/2008CA2669034A1 Chemical compounds
05/14/2008EP1921062A2 Amino acid derivatives as HIV aspartyl protease inhibitors
05/14/2008EP1919879A1 9-aminocarbonylsubstituted derivatives of glycylcyclines
05/14/2008EP1919872A2 Chemical compounds
05/14/2008EP1919871A2 Method for the synthesis of quinoli e derivatives
05/14/2008EP1713776B1 Quinoline derivatives for use as mycobacterial inhibitors
05/14/2008EP1711468B1 Process for preparing purified ciprofloxacin
05/14/2008EP1485365B1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase
05/14/2008CN101180302A Process for preparing (alpha s, beta r)-6-bromo-alpha-[2-(dimethylamino)ethyl]-2-methoxy-alpha-1-naphthalenyl-beta-phenyl-3-quinolineethanol
05/14/2008CN101180273A Methods of synthesizing 6-alkylaminoquinoline derivatives
05/14/2008CN101180269A Method of preparing 3-cyano-quinolines and intermediates made thereby
05/14/2008CN101177412A Method for synthesizing acetyl substituted nitrogen heterocycle compounds
05/14/2008CN101177385A Aryl sulfonic acid amides and analogues as well as its purpose in curing neural degeneration disease
05/14/2008CN100387576C Substituted phenylalkanoic acid derivatives and use thereof
05/13/2008US7371868 Bactericides; 2-[(1R)-1-methyl-2-trityl-2,3-dihydro-1H-5-isoindolyl]-1,3,6,2-dioxazaborocane.
05/13/2008US7371865 Reacting an organophosphouus compound with metallized alkane; forming atorvastatin, lorastatin, pitavastatin, fluvastatin
05/13/2008US7371765 Quinoline derivatives having VEGF inhibiting activity
05/13/2008US7371764 agricultural and horticultural fungal infections of plants; novel N-alkynyl-2-quinolin-(isoquinolin- and quinazolin-)oxyalkylamides; 2-(6-quinolinyloxy)-N-(4-methylpent-2-yn-4-yl) butyramide
05/13/2008US7371752 such as 5-(4-Fluorophenyl)-7-[(2-pyridyl)-methyloxy]-thieno[3,2-b]pyridine, used as prodrugs or antagonists for GABA receptors, in diagnosis and treatment of anxiety, depression, Down Syndrome, sleep and epileptic disorders, as cognition activators and as antidotes to benzodiazepines
05/08/2008WO2008053913A1 Sulfonylurea derivative capable of selectively inhibiting mmp-13
05/08/2008WO2008053863A1 Novel compound having 1,4-benzothiazin-3-one skeleton or 3,4-dihydroquinolin-2-one skeleton
05/08/2008WO2008053158A1 Inhibitors of p38 mitogen-activated protein kinase
05/08/2008WO2007028022A3 Novel compounds as p2x7 modulators and uses thereof
05/08/2008US20080108656 3-Fluoro-2-(2-methylsulfanyl-phenyl)-quinolin-4-yl]-pyridin-4-yl-amine; modulating transforming growth factor (TGF) - beta; fibroproliferative diseases or diseases associated with fibrosis; cardiovascular, urogenital and gastrointestinal disorders; antihypotensive, -arthritic agents; angioplasty
05/08/2008US20080108651 5-[3-((R)(-)-5,7-Dibromo-1,2,3,4-tetrahydro-naphthalen-1-ylamino)-propylamino]-4H-thieno[3,2-b]pyridine-7-one; optically active; new target antibiotic, inhibitor of bacterial methionyl tRNA synthetase; antibiotic resistance; Clostridium difficile infection; mostly in immunodeficient, elderly
05/08/2008US20080108601 anticancer agents; catalytic hydrogenation
05/08/2008US20080108122 Microchemical nanofactories
05/07/2008EP1918272A1 Pharmaceutically active compounds and methods of use
05/07/2008EP1917245A1 Heterocyclic compounds and their use as binding partners for 5-ht5 receptors
05/07/2008EP1917244A2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-ht5-receptors
05/07/2008EP1603880B1 Quinolinone/benzoxazinone derivatives and uses thereof
05/07/2008EP1405848B1 Tetrahydroquinoline derivative compound and drug containing the compound as active ingredient
05/07/2008CN101173058A Method for producing molecular engram polyalcohol microsphere and method for separating enrofloxacin thereof
05/07/2008CN101172966A Method for producing aripiprazole crystallite
05/07/2008CN100386318C Tetrahydroquinoline derivatives and their use as FSH receptor modulators
05/06/2008US7368592 Process for the preparation of alkyl n-alkylanthranilate
05/06/2008US7368573 Triamide-substituted heterobicyclic compounds
05/06/2008US7368572 Anticancer agents
05/06/2008US7368479 Alpha-sulfonylamino-acetonitriles
05/02/2008WO2008049922A2 A new process for the preparation of montelukast
05/02/2008CA2666539A1 Substituted phenylmethyl bicyclocarboxyamide compounds
05/01/2008US20080103174 Ether derivatives
05/01/2008US20080103173 Compounds Having Activity At Nk3 Receptor And Uses Thereof In Medicine
05/01/2008US20080103135 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine
04/2008
04/30/2008EP1915382A2 Hepatitis c serine protease inhibitors and uses therefor
04/30/2008CN101171234A Dihydropyridine derivatives
04/30/2008CN100384833C Therapeutic chroman compounds
04/30/2008CN100384825C Benzheterocyclic derivatives
04/30/2008CN100384824C Acetyl 2-hydroxy-1, 3-diaminoalkanes
04/30/2008CN100384823C Bicyclic androgen and progesterone receptor modulator compounds and methods
04/29/2008USRE40278 Heterocyclic amines having central nervous system activity
04/29/2008US7365209 Nitrogen heterocycle biaryls for osteoporosis and other diseases
04/29/2008US7365203 Process for the synthesis of 6-amino-4-(3-chloro-4-fluoro-phenylamino)-7-ethoxy-quinoline-3-carbonitrile
04/29/2008US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives
04/29/2008US7365089 Triazolo-quinolin derivatives useful as adenosine receptor ligands
04/29/2008US7365081 Antitumor agents
04/29/2008US7365076 for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/29/2008US7365065 Antigonadotrophins; Breast and prostate cancer, endometriosis and benign prostate hyperplasia; regulation of fertility; in-vitro fertilisation; oral administration; inexpensive; 3-Amino-4-chloro-N-[4-chloro-5-(2,3-dihydro-benzo[1,4]oxazine-4-carbonyl)-thiophen-3-ylmethyl]-N-methyl-benzenesulfonamide
04/24/2008WO2008049047A2 Quinoline compounds
04/24/2008WO2008048698A2 Chemical switches for detecting reactive chemical agents
04/24/2008WO2008046598A1 DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE β2 ADRENERGIC RECEPTOR
04/24/2008US20080097119 preventing, treating or ameliorating retinoid poisoning, overdose by a retinoid; Z-4-[3-(3,3-Dimethyl-1-p-tolyl-3H-inden-5-yl)-3-hydroxyimino-propenyl]-3-fluoro-benzoic acid
04/24/2008US20080097104 Novel Compounds and Preparation for Montelukast Sodium
04/24/2008US20080097102 Aminotetralin-derived urea modulators of vanilloid vr1 receptor
04/24/2008US20080096936 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
04/24/2008US20080096917 for plants; 2-(dibenzofuranyl-2-oxy)-2-methylthio-N-(2-methylpent-3-yn-2-yl)acetamide; 2-(indanyl-5-oxy)-2-methylthio-N-(2-methylpent-3-yn-2-yl)acetamide; 2-(3-phenylquinolinyl-6-oxy)-2-methylthio-N-(2-methylpent-3-yn-2-yl)acetamide; phytopathogenic fungi
04/24/2008US20080096894 Anti-Bacterial Compounds
04/24/2008US20080096885 Methyl 1-(2-fluorophenyl)-2-[(3-methoxy-2-phenylquinolin-4-yl)carbonyl]hydrazinecarboxylate; schizophrenia
04/24/2008US20080096884 phosphodiesterase inhibitors; inflammatory and/or allergic diseases such as chronic obstructive pulmonary disease (COPD), asthma, rheumatoid arthritis or allergic rhinitis
04/24/2008US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia
04/24/2008US20080096875 Hepatitis C virus infection; thiourea-substituted dibenzofuran, fluorene, or carbazole compounds
04/24/2008US20080096873 New compounds
04/24/2008US20080096869 Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors
04/24/2008CA2672926A1 Bicyclic heteroaromatic compounds
04/24/2008CA2666508A1 Quinoline compounds
04/24/2008CA2665376A1 Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the .beta.2 adrenergic receptor
04/23/2008EP1914227A1 Polymorphic crystal form of a indan-2-ylamino-hydroxyethyl-quinolinone maleate derivative as beta-adrenoceptor agonist
04/23/2008EP1912970A2 Acyltryptophanols for fertility control
04/23/2008EP1912958A1 Substituted malononitrile compounds for combating animal pests
04/23/2008EP1912948A1 Antibacterial quinoline derivatives
04/23/2008EP1912648A2 Quinoline derivatives as antibacterial agents
04/23/2008EP1912647A2 Quinoline derivatives as antibacterical agents
04/23/2008EP1474145B1 Quinoline derivatives as npy antagonists
04/23/2008EP0998459B1 Pyridine derivatives
04/23/2008CN101166726A Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity
04/23/2008CN100383124C Quinoline derivatives as NPY antagonists
04/22/2008US7361756 by mixing 7-hydroxy-tetrahydroquinolinone, dibromobutane, and at least one base to form a reaction mixture; using phase transfer catalysts; or using a low boiling point solvent
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