Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676) |
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10/22/2009 | WO2009077956A3 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM |
10/22/2009 | WO2008110355A8 Quinoline derivatives as fungicides |
10/22/2009 | US20090264653 Useful indole compounds |
10/22/2009 | US20090264464 Antitumor agent for undifferentiated gastric cancer |
10/22/2009 | US20090264435 Novel Aryl- and Heteroarylpiperazines |
10/22/2009 | US20090264424 Vanilloid receptor ligands and their use in treatments |
10/22/2009 | US20090263488 Pressurised metered dose inhalers containing solutions of beta-2 agonists |
10/22/2009 | CA2721785A1 New arylsulphonylglycine derivatives, the preparation thereof and their use as medicaments |
10/22/2009 | CA2718538A1 Quinoline derivatives as axl kinase inhibitors |
10/21/2009 | EP2109603A1 Process for the preparation of 8-hydroxy-5-[(1r)-1-hydroxy-2[[(1r)-2-(4-methoxyphenyl)-1-methylethyl]amino]-ethyl]-2(1h)-quinolinone monohydrochloride |
10/21/2009 | EP1513531B1 Basic non-peptide bradykinin antagonists and pharmaceutical compositions therefrom |
10/21/2009 | EP1363980B1 Luminescent polymers |
10/21/2009 | EP1280776B1 Substituted benzoic acid amides and use thereof for the inhibition of angiogenesis |
10/21/2009 | CN101563347A Vasopressin V1a antagonists |
10/21/2009 | CN101563318A N- (5, 6, 7, 8-tetrahydronaphthalen-1-yl) urea derivatives and related compounds as trpv1 vanilloid receptor antagonists for the treatment of pain |
10/21/2009 | CN101562234A Organic electroluminescent display element |
10/21/2009 | CN101562232A Color-adjustable organic electroluminescent device and preparation method thereof |
10/21/2009 | CN101560184A N-chiral quaternary ammonium salt derived from amino acid and preparation method thereof |
10/21/2009 | CN101560158A Novel organic electroluminescent compounds and organic electroluminescent device using the same |
10/20/2009 | US7605267 Process for the preparation of 5-(halocetyl)-8-(substituted oxy)-(1h)-quinolin-2-ones |
10/15/2009 | WO2009125597A1 Acylthiourea compound or salt thereof, and use of the compound or the salt |
10/15/2009 | US20090259044 Compositions and methods for modulating sirtuin activity |
10/15/2009 | US20090258884 Substituted amides |
10/15/2009 | CA2720552A1 Acylthiourea compound or salt thereof, and use thereof |
10/14/2009 | EP1720829B1 Derivatives of heteroaryl-alkylcarbamates, preparation method thereof and use of same as faah enzyme inhibitors |
10/14/2009 | EP1687276B1 Novel method of preparing 3-fluorinated quinolines |
10/14/2009 | CN101558042A Method of preparing montelukast and intermediates used therein |
10/14/2009 | CN101555225A Method for preparing poly-substituted quinoline compound |
10/13/2009 | US7601842 Asymmetric hydrogenation of enaminoesters without protecting the secondary amino group with a protective group; good asymmetric, chemical yields and workability; methyl (2R,4S)-(2-ethyl-6-trifluoromethyl-1,2,3,4-tetrahydroquinolin-4-yl)carbamate |
10/13/2009 | US7601841 Quinolinyl and benzothiazolyl modulators |
10/13/2009 | US7601837 Quinoline derivatives and their use as 5-HT6 ligands |
10/13/2009 | US7601741 decyclization of {3-[(E)-2(7-chloro-2-quinolinyl)vinyl]phenyl}-4,5-dihydro-3H-benzo[c]thiepin-1-one by methylmagnesium halide with following conversion to montelukast |
10/13/2009 | US7601674 α-oxygenated or α-thiolated carboxylic acid phenethylamide derivatives |
10/13/2009 | CA2341678C Potassium channel inhibitors and method |
10/08/2009 | WO2009123241A1 Inhibitor of plasminogen activator inhibitor-1 |
10/08/2009 | WO2009123194A1 Heterocyclic compound |
10/08/2009 | WO2009122034A2 Novel hsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
10/08/2009 | US20090253908 Novel m3 muscarinic acetylchoine receptor antagonists |
10/08/2009 | US20090253740 Substituted n-bicyclicalkyl bicycliccarboxyamide compounds |
10/08/2009 | US20090253739 Amine Derivatives |
10/08/2009 | US20090253726 Tri-, tetra-substituted-3-aminopyrrolidine derivative |
10/08/2009 | US20090253656 Bcrp/abcg2 inhibitor |
10/08/2009 | US20090253655 Quinolinone farnesyl transferase inhibitors for the treatment of synucleinopathies and other indications |
10/08/2009 | CA2718488A1 Novel dhsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
10/07/2009 | EP2107052A1 Novel n-(2-aminophenyl)benzamide derivative having an urea structure |
10/07/2009 | EP1709027B1 Hydrazide type compounds and the use thereof in pharmaceutical compositions for the treatment of cardiovascular diseases |
10/07/2009 | CN101553472A Tetrahydronaphthaline derivatives, methods for the production and use thereof as anti-inflammatory agents |
10/07/2009 | CN101553471A 抗菌喹啉衍生物 Antibacterial quinoline derivatives |
10/07/2009 | CN101553470A Antibacterial quinoline derivatives |
10/07/2009 | CN101553469A Carboxylic acid derivative |
10/07/2009 | CN100546977C New compounds for the inhibition of rotamases and use thereof |
10/06/2009 | US7598412 Cystic fibrosis transmembrane conductance regulator; ABC transporter mediated diseases like cystic fibrosis; 5-methoxy-N-((1-(3,4-dimethoxyphenyl)-cyclohexyl)methyl)benzofuran-2-carboxamide; or sulfonamide analogs; chloride or bicarbonate channel modulators |
10/06/2009 | US7598390 1-Benzyl-4-methyl-2-(1-methylimidazoyl)-quinolinium acetate, for example; compounds are stains that become fluorescent upon illumination and interaction with double stranded DNA, but exhibit reduced or no fluorescence in the absence of double stranded DNA |
10/06/2009 | US7598385 Reacting unsubstituted or substituted 2-methylbenzothiazole, 2-methylbenzooxazole or 2,3,3-trimethyl-3H-indoline with substituted or unsubstituted benzylhalide, forming 4-methylquinoline quaternary ammonium salt intermediates, condensing with N,N'-diphenylformamidine; for staining nucleic acids |
10/06/2009 | US7598384 Specific binding is extremely high; low toxicity; high degree of activity; 2-(5-m-Tolyl-thiazol-2-yl )-7,8-dihydro-6H-quinolin-5-one, acute and/or chronic neurological disorders |
10/06/2009 | US7598383 mitogen activated protein kinase inhibitors; 4-(2-fluoro-4-methylphenylamino)-1,3-dimethyl-6,7-dihydro-1H-pyrrolo[3,4-b]pyridine-2,5-dione; used in the treatment of hyperproliferative diseases, such as cancer and inflammation in mammals |
10/06/2009 | US7598263 9-[(3-hydroxy-5-methoxyphenyl)amino]-1,2-dihydrothieno[3,2-f]quinoline-8-carbonitrile 3,3-dioxide; protein tyrosine kinases inhibitor, especially erythropoetin-producing hepatoma amplified sequence (Eph) receptors antagonist; antitumor, angiogenesis inhibitor, neurodegenerative diseases |
10/06/2009 | US7598258 Quinoline derivatives and quinazoline derivatives inhibiting autophosphorylation of macrophage colony stimulating factor receptor |
10/06/2009 | US7598242 Compounds for the treatment of inflammatory disorders |
10/06/2009 | US7598236 Diazabicyclic central nervous system active agents |
10/06/2009 | US7597926 Electroluminescent quinolates |
10/06/2009 | CA2301377C N-aroylphenylalanine derivatives |
10/06/2009 | CA2291048C Dehydration plant |
10/06/2009 | CA2258924C Cftr channel activator compounds and pharmaceutical compositions containing same |
10/01/2009 | WO2009120774A2 Method of preparing huperzine a and derivatives thereof |
10/01/2009 | WO2009119817A1 Stable vinamidinium salt and nitrogen-containing heterocyclic ring synthesis using the same |
10/01/2009 | WO2009117484A2 Small molecule e2f inhibitor |
10/01/2009 | WO2009087098A3 Quinoline derivatives and their use as fungicides |
10/01/2009 | WO2009060835A8 Novel ubiquilin-binding small molecule |
10/01/2009 | WO2009049716A3 Novel fungicides |
10/01/2009 | US20090247761 Preparation of 3,4-Dihydroisoquinolines in the Synthesis of Morphinans |
10/01/2009 | US20090247760 Preparation of Amides from an Acid and Amine for Intermediates in the Synthesis of Morphinans |
10/01/2009 | US20090247759 Purification process of Montelukast and its Amine Salts |
10/01/2009 | US20090247758 Novel Quinoline Compound, and Composition Containing Centipede Extract or Compounds Isolated Therefrom for Prevention and Treatment of Cardiovascular Disease |
10/01/2009 | US20090247754 Method of preparing huperzine a and derivatives thereof |
10/01/2009 | US20090247745 adenosine A3 receptor antagonists; improved bioavailability; treatment of diseases such as asthma, COPD and ARDS, glaucoma, tumor, allergic and inflammatory diseases, ischemia, hypoxia, arrythmia and renal diseases; e.g. 4-Methoxy-N-[6-(morpholin-4-yl)-4-benzylamino-3-cyanoquinolin-2-yl]-benzamide |
10/01/2009 | US20090247731 Boronic ester and acid compounds, synthesis and uses |
10/01/2009 | US20090247578 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
10/01/2009 | US20090247576 Anti-tumor agent for multiple myeloma |
10/01/2009 | US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders |
10/01/2009 | US20090247506 Antibacterial agents |
09/30/2009 | EP2105443A1 Oxime derivatives and their use in photopolymerizable compositions for colour filters |
09/30/2009 | EP1962849B1 Quinoline derivatives useful in the treatment of mglur5 receptor-mediated disorders |
09/30/2009 | EP1711181B1 Quinoline derivatives and use thereof as mycobacterial inhibitors |
09/30/2009 | CN101547907A 抗菌的喹啉衍生物 Antibacterial quinoline derivatives |
09/30/2009 | CN101547906A Antibacterial quinoline derivatives |
09/30/2009 | CN101547905A Antibacterial quinoline derivatives |
09/30/2009 | CN101547904A Fumarate salt of (alpha S, beta R)-6-bromo-alpha-[2-(dimethylamino)ethyl]-2-methoxy-alpha-1-naphthalenyl-beta-phenyl-3-quinolineethanol |
09/30/2009 | CN101544602A Fleroxacin lactate and preparation method thereof |
09/30/2009 | CN101544601A Method for synthesizing 5,6,7,8-tetrahydroquinoline |
09/29/2009 | US7595501 Electroluminescent iridium compounds with fluorinated phenylpryidines, phenylpyrimidines, and phenylquinolines and devices made with such compounds |
09/29/2009 | US7595402 Treating dry eye, use as male contraceptive, or against prostate cancer; ester, carbonate, glycoside prodrugs of SARMS such as N-(4-Cyano-3-trifluoromethylphenyl)-3-(p-fluorophenoxy)-2-hydroxy-2-methyl-propionamide; bioavailability |
09/29/2009 | US7595399 Tyrosine derivatives |
09/29/2009 | US7595343 Inhibitors of histone deacetylase |
09/29/2009 | CA2176796C Substituted benzyloxycarbonylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament containing them |
09/24/2009 | WO2009117381A2 Preparation of montelukast and its salts |
09/24/2009 | WO2009115257A1 Substituted sulfonamide derivatives |
09/24/2009 | WO2009024611A3 4-benzylaminoquinolines, pharmaceutical compositions containing them and their use |
09/24/2009 | US20090240053 2-(4-(1-methyl-4-piperidinoxy)benzylamino)-2-methyl-propanamide; nervous system disorders; analgesics; anticonvulsants; sodium channel moderators; antidepressants, antiarrhythmics and for the treatment or prevention of diabetic neuropathy |
09/24/2009 | US20090239906 Alkoxyalkyl-substituted cyclic ketoenols |