Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
11/1998
11/12/1998CA2289602A1 Protease inhibitors
11/12/1998CA2288149A1 N-methyl-d-aspartate (nmda) receptor blockers for the prevention of atherosclerosis
11/11/1998EP0877019A1 Substituted diaminocarboxylic acid
11/11/1998EP0876349A1 Quinoline derivatives as gnrh antagonists
11/11/1998EP0876348A1 Salts of quinoline derivatives as nk3 antagonists
11/11/1998EP0876347A1 Quinoline derivatives
11/11/1998EP0876346A1 Antimalarial quinolin derivatives
11/11/1998EP0876345A1 Heterocyclic compounds as h+-atpases
11/11/1998EP0876337A2 New lh-rh antagonists with improved effectiveness
11/11/1998EP0876330A1 Aryl or heteroaryl amides of tetrahydronaphthalene, chroman, thiochroman and 1,2,3,4-tetrahydroquinoline carboxylic acids having retinoid-like biological activity
11/11/1998EP0640074B1 Salts of a quinolone-carboxylic acid
11/11/1998CN1198816A Polyoxyhydrocarbyl related products and methods for fluorescence assays
11/10/1998US5834485 Quinoline sulfonamides and their therapeutic use
11/10/1998US5834467 HIV protease inhibitors
11/10/1998US5834447 Thiophene derivatives
11/10/1998US5834434 Inhibitors of farnesyltransferase
11/09/1998CA2237052A1 Substituted diaminocarboxylic acids
11/05/1998WO1998049155A1 Cell differentiation inducing amide derivatives, their production and use
11/05/1998WO1998049152A1 Protease inhibitors
11/05/1998WO1998048807A1 Hyaluronate synthesis inhibitors
11/05/1998WO1998013349A3 Heteroaryloxyethylamines as 5-ht1a ligands
11/05/1998CA2287567A1 Protease inhibitors
11/05/1998CA2285402A1 Amide derivatives, their production and use
11/04/1998EP0875506A1 Quinoline and quinazoline compounds useful in therapy
11/04/1998EP0874827A1 Quinoline derivatives as nk3 antagonists
11/04/1998EP0874826A1 Naphthalene quinolines having leukotriene-antagonistic action
11/04/1998EP0874625A1 Indane derivatives for antipsychotic compositions
11/03/1998US5831093 Preparation of n-aryl- and n-hetarylhydroxylamines
11/03/1998US5830890 Fungicidal acrylate derivatives
11/03/1998US5830834 Ammonium carboxylate type fluorine-containing compound, solid surface modifier containing the same and magnetic recording medium using the same
10/1998
10/29/1998WO1998047890A1 Substituted benzopyran derivatives for the treatment of inflammation
10/29/1998WO1998047885A1 A bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5ht1a, 5ht1b and 5ht1d receptor antagonistic activity
10/29/1998WO1998047874A1 Crf antagonistic quino- and quinazolines
10/29/1998WO1998047873A1 Process for producing quinolone derivatives
10/29/1998WO1998047869A1 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
10/29/1998WO1998047868A1 Heterocycle-containing urea derivatives as 5ht1a, 5ht1b and 5ht1d receptor antagonists
10/29/1998CA2288172A1 A bicyclic aryl or a bicyclic heterocyclic ring containing compounds having a combined 5ht1a, 5ht1b and 5ht1d receptor antagonistic activity
10/29/1998CA2287255A1 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
10/28/1998EP0656887B1 Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
10/28/1998CN1197450A Esters and amides as PLA2 inhibitors
10/28/1998CN1197083A Bulk dyeing using quinophthalone dyestuffs
10/28/1998CN1040440C Process for preparing dehydrocycloclausenamide derivatives
10/27/1998US5827891 For treatment of aids, blocking replication of hiv virus
10/27/1998US5827859 HIV protease inhibitors
10/27/1998US5827858 Administered to treat aids
10/22/1998WO1998046229A1 Il-8 and mcaf production inhibitors
10/21/1998EP0872478A2 Intermediates for the preparation of 1-substituted, 2-substituted 1H-imidazo[4,5-c]quinolin-4-amines
10/21/1998EP0871616A1 Process for the preparation of anti-malarial drugs
10/21/1998EP0871448A1 Aryl and heteroaryl quinazoline compounds which inhibit csf-1r receptor tyrosine kinase
10/21/1998EP0871439A1 Substituted (aryl, heteroaryl, arylmethyl or heteroarylmethyl) hydroxamic acid compounds
10/21/1998CN1196724A Piperazine devivatives and process for preparation thereof
10/20/1998US5824705 Carbamates and crop protection agents containing them
10/20/1998US5824689 Quinoline compound extracted from scolopendra subspinipes, and derivatives thereof
10/20/1998US5824688 HIV protease inhibitors
10/15/1998WO1998045277A1 Preparation of heterocycles using 1,3-dihalopropenes
10/15/1998WO1998045269A1 Quinoline derivatives, having in particular antiviral properties, preparation and biological applications thereof
10/14/1998EP0870752A1 Bulk dyeing using quinophthalone dyestuffs
10/14/1998EP0695293B1 10,11-methanodibenzosuberane derivatives used as chemosensitizing agents
10/14/1998EP0678090B1 Piperazine derivatives
10/14/1998CN1195987A Use of carbostyril derivative for inhibiting carcinogenesis
10/14/1998CN1040176C Drug prepared by quinolone derivative for preventing and treating disturbances of intestinal mucous membrance and its use
10/13/1998US5821264 Used in foodstuffs and dietary supplements to decrease lipoprotein concentration or increase feed conversion
10/13/1998US5821251 Nitrogen heterocycles
10/13/1998US5821244 Condensed nitrogen heterocycles and their use as pesticides, fungicides and antimycotics
10/08/1998WO1998043960A1 Substituted 3-cyano quinolines
10/08/1998WO1998043959A1 Hydroxamic acids substituted by heterocycles useful for inhibition of tumor necrosis factor
10/08/1998CA2285241A1 Substituted 3-cyano quinolines
10/07/1998EP0869122A1 Quinolinic sulfide derivatives acting as NMDA receptor antagonists and process for preparation thereof
10/07/1998CN1194978A Benzyloxy-substituted, fused N heterocycles, process for their preparation and their use as bradykinin receptor antagonists
10/07/1998CN1040106C Process for preparing piperazine derivatives
10/07/1998CN1040062C Process for preparing pharmacologically active catechol derivatives
10/06/1998US5817674 Antiotensin ii receptor antagonists
10/06/1998US5817496 Kynurenine aminotransferase
10/01/1998WO1998042673A1 Quinoline-2-carboxylic acid derivative and its use as excitatory amino acids antagonist
10/01/1998WO1998042672A1 Benzene derivatives
10/01/1998WO1998042341A1 Anti-fiv agent
10/01/1998CA2284710A1 Quinoline-2-carboxylic acid derivative and its use as excitatory amino acids antagonist
09/1998
09/30/1998EP0867432A2 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists
09/30/1998EP0866692A1 Use of bicyclic mono- or diketone derivatives, resulting compounds, and use thereof as a drug for treating inflammation, migraine and shock
09/30/1998CN1194637A Process for preparing quinoline bases
09/30/1998CN1039998C Substituted cycloalkylacetamides and its preparation, medicine and use
09/27/1998CA2232499A1 Benzyloxy-substituted, fused n heterocycles, process for their preparation, and their use as bradykinin reception antagonists
09/24/1998WO1998041506A1 Novel quinoline- and naphthalenecarboxamides, pharmaceutical compositions and methods of inhibiting calpain
09/24/1998CA2284035A1 Novel quinoline- and naphthalenecarboxamides, pharmaceutical compositions and methods of inhibiting calpain
09/23/1998EP0866063A1 10, 11-Methanodibenzosuberane derivatives used as chemosensitizing agents
09/23/1998EP0865440A1 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
09/23/1998EP0865424A1 Pesticides
09/23/1998EP0865421A1 Arylethanolamine derivatives and their use as agonists of atypical beta-adrenoceptors
09/23/1998EP0865279A1 Hemoregulatory compounds
09/22/1998US5811576 1-carboxy-2-loweralkyl-3,4,6-tri(halo)benzenes; grampositive and-negative bacteria; infections; sterilization of medical equipment
09/22/1998US5811553 Quinoline derivatives(2)
09/22/1998US5811455 Compounds useful for treating allergic or inflammatory diseases
09/22/1998US5811427 Heterocyclic N-acetonylbenzamides
09/22/1998US5811370 Used for thermal transfer
09/22/1998CA2056911C Hiv protease inhibitors
09/17/1998WO1998040790A1 Photosensitive quinolone compounds and a process of preparation
09/17/1998WO1998040383A1 Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with n- or c-linked imidazoles
09/17/1998WO1998039970A1 Quinoline leukotriene antagonists
09/16/1998EP0863883A1 Alpha-(1,3-dicarbonylenol ether) methyl ketones as cysteine protease inhibitors
09/16/1998EP0863876A1 Quinoline derivatives containing a diol as leukotriene antagonists