Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
12/2002
12/19/2002CA2449256A1 Modulators of peroxisome proliferator activated receptors
12/19/2002CA2445653A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/18/2002EP1267495A1 RF receiver having cascaded filters and an intermediate amplifier stage
12/18/2002EP1267170A1 Method for characterising polypeptides
12/18/2002EP1266888A1 Quinoline derivatives and medicinal use thereof
12/18/2002EP1265853A1 Carboxylic acid derivatives as ip antagonists
12/18/2002EP1265640A1 Fluorescent membrane intercalating probes and methods for their use
12/17/2002US6495693 N-(aryl/heteroaryl) amino acid derivatives, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
12/17/2002US6495581 Drug for treating diabetes mellitus, hyperlipemia, impaired glucose tolerance, arterial sclerosis and improving insulin resistance, inflammatory disease
12/17/2002US6495566 Potent antagonists at the strychnine insensitive glycine binding site associated with the n-methylaspartic acid receptor complex
12/17/2002US6495565 For therapy of acute infection, acute phase response, age related macular degeneration, alcoholism, anorexia, asthma, autoimmune disease, autoimmune hepatitis, bechet's disease, cachexia, calcium pyrophosphate dihydrtate deposition
12/17/2002US6495552 Treatment or prevention of the diseases and conditions which respond to treatment by retinoids and or which in healthy mammals, including humans, are controlled by natural retinoic acid.
12/17/2002CA2061675C Quinoline-containing ketoacids as leukotriene antagonists
12/12/2002WO2002099124A2 Characterising polypeptides
12/12/2002WO2002098859A1 Process for preparation of a quinolinecarbaldehyde
12/12/2002WO2002098856A2 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
12/12/2002WO2002098848A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents
12/12/2002WO2002098425A1 Substituted 4-aryl-3-(3-aryl-1-oxo-2-propenyl)-2(1h)-quinolinones and analogs as activators of caspases and inducers of apoptosis and the use thereof
12/12/2002WO2002098424A1 Novel anti-infectives
12/12/2002WO2002098406A1 Novel compounds and compositions as cathepsin inhibitors
12/12/2002WO2002098367A2 Hybrid 2-aminotetralin and aryl-substituted piperazine compounds and their use in altering cns activity
12/12/2002US20020188122 Such as pyridine-4-carboxaldehyde-(4-Morpholinylprop-3-yl) imine for use in therapy as cytokine inhibitors
12/12/2002US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV
12/12/2002US20020187983 Process for the synthesis of derivatives of 2, 3-dihydro-1, 4-dioxino- [2, 3-f] quinoline
12/12/2002CA2449942A1 Characterising polypeptides
12/12/2002CA2449770A1 Novel anti-infectives
12/12/2002CA2449021A1 Novel compounds and compositions as cathepsin inhibitors
12/12/2002CA2446719A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents
12/11/2002EP1264827A1 Process for the preparation of Tosylbenzylformamides
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263756A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
12/11/2002EP1263755A2 Cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
12/11/2002EP1263733A2 Derivatives of quinoline as alpha-2 antagonists
12/11/2002EP1263716A2 Amino acid derivatives as hiv aspartyl protease inhibitors
12/11/2002EP1263503A2 Use of cyanoquinolines for treating or inhibiting colonic polyps
12/11/2002EP1100805B1 Medicine nitrate salts
12/11/2002EP0966436B1 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
12/11/2002EP0805796B1 Cell adhesion inhibitors
12/11/2002EP0752813B1 Inhibitors of metazoan parasite proteases
12/11/2002EP0624155B2 Carbamates and plant-protecting agents containing them
12/11/2002CN1095834C Quinolinone derivatives and antianaphylactic agent containing said quinolinone derivative as biological active component
12/10/2002US6492517 The present invention relates to a method for preparing 5- and 6-halomethyl quinoxalines in presence of a radical initiator in a solvent selected from the group consisting of fluorobenzene, difluorobenzenes, trifluorobenzenes,
12/10/2002US6492412 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
12/10/2002US6492393 Compounds useful as anti-inflammatory agents
12/10/2002US6492390 Treating cyclooxygenase-2 mediated disorders.
12/10/2002US6492373 6-fluoro-1,4-dihydro-7-[4-(2-hydroxyiminoethyl)-1-piperazinyl]-4-oxoquinoline-3-carboxylic acid derivatives, their preparation and pharmaceutical compositions
12/10/2002US6492368 Benzamidine derivatives as factor XA inhibitors
12/10/2002US6492362 Compounds and compositions as cathepsin S inhibitors
12/09/2002WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
12/09/2002CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments
12/05/2002WO2002096903A2 Chemical derivatives and the use thereof as an anti-telomerase agent
12/05/2002WO2002096879A1 Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands
12/05/2002WO2002096869A2 Piperazine mono(dithio)carbamate ester compounds and analogs thereof
12/05/2002WO2002096858A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002WO2002096516A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/05/2002WO2002096424A1 Hetereocyclic beta-aminoacids and their use as anti-epileptogenic agents
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002US20020183321 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
12/05/2002CA2448894A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002CA2448160A1 Heterocyclic beta-amino acids and their use as anti-epileptogenic agents
12/05/2002CA2447657A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
12/04/2002EP1262477A1 Anti-acid-fast bacterial agents containing pyridonecarboxylic acids as the active ingredient
12/04/2002EP1262476A1 Processes for preparing quinoline derivatives and intermediates thereof
12/04/2002EP1261579A1 Dehydroamino acids
12/04/2002EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
12/04/2002EP1097139B1 Quinoline derivatives
12/04/2002EP0815124B1 Heterocyclecarbonyl amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors
12/04/2002CN1383424A Aryl and heteroacrylcyclopropyl oxime ethers and their use as fungicides
12/03/2002US6489479 Process for the preparation of mixed anhydrides
12/03/2002US6489478 4-amino substituted-2-substituted-1,2,3,4-tetrahydroquinolines
12/03/2002US6489475 Method of producing heterocyclic derivatives
12/03/2002US6489339 C3A receptor ligands
11/2002
11/28/2002WO2002094809A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/28/2002WO2002094799A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
11/28/2002WO2002094789A1 Quinoline derivatives as ligands for the neuropeptide y receptor
11/28/2002WO2002094788A1 2-substituted 1,2,3,4-tetrahydroquinolines and derivatives thereof, compositions and methods
11/28/2002WO2002094770A2 Aminoalcohol derivatives
11/28/2002WO2002094268A1 Tetrahydroquinolin derivatives for the inhibition of diseases associated with estrogen deprivation or with an aberrant physiological response to endogenous estrogen
11/28/2002WO2002094261A1 Cxcr4-antagonistic drugs comprising nitrogen-containing compound
11/28/2002WO2002094203A2 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
11/28/2002WO2002094187A2 Novel use
11/28/2002US20020177716 Intermediates of CETP inhibitors
11/28/2002US20020177715 Quinone-indicator antibiotics; controlling gene expression
11/28/2002US20020177637 Polymers and oligomers, their synthesis, and electronic devices incorporating same
11/28/2002US20020177601 Inhibit the signal transduction by tyrosine kinases; e.g. 4-(3-chloro-4-fluorophenylamino)-6-(3-(4-(methoxycarbonyl-methyl)-1 -piperazinyl)propyloxy)-7-methoxyquinazoline; use such as antitumor agent
11/28/2002US20020177594 Inhibitors of histone deacetylase
11/28/2002US20020177588 Selectivity
11/28/2002US20020177587 Treating sexual dysfunction including erectile dysfunction, diabetes melitus, gastrointestinal disorders, including gastric paresis and cardiovascular disorders; cyclic guanosine 3',5'-monophosphate (cGMP)
11/28/2002US20020177559 Inhibitors of cellular efflux pumps of microbes
11/28/2002CA2448080A1 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
11/28/2002CA2448076A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
11/28/2002CA2447103A1 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
11/28/2002CA2447063A1 Novel use
11/28/2002CA2446324A1 Quinoline derivatives as ligands for the neuropeptide y receptor
11/28/2002CA2444787A1 Tetrahydroquinolin derivatives for the inhibition of diseases associated with estrogen deprivation or with an aberrant physiological response to endogenous estrogen
11/27/2002EP1259497A1 Novel quinoline ligands and metal complexes for diagnosis and therapy
11/27/2002EP1259488A1 Ortho-sulfonamido aryl hydroxamic acids, process for their preparation and their use as matrix metalloproteinase inhibitors
11/27/2002EP1073639B1 Quinoline derivatives
11/27/2002EP0862557B1 SYMMETRICAL bis-HETEROARYLMETHOXYPHENYLALKYL CARBOXYLATES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS
11/27/2002CN1382124A Bicycle androgen and progesterone receptor modulator compounds and methods