Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
01/2004
01/08/2004US20040006137 Asymmetric synthesis of amino-pyrrolidinones and a crystalline, free-base amino-pyrrolidinone
01/08/2004US20040006103 Use of chloroquine, hydroxychloroquine and 4 amino-quinolinic derivatives to obtain a drug for the anti retroviral therapy, active towards HIV sensitive strains and towards HIV strains which are resistant to both nucleosidic and non-nucleosidic reverse transcriptase inhibitors and to proteases inhibitors
01/08/2004US20040006102 Alkoxy aryl beta2 adrenergic receptor agonists
01/08/2004CA2493854A1 Phosphodiesterase inhibitor
01/08/2004CA2489560A1 Substituted quinoline ccr5 receptor antagonists
01/08/2004CA2489433A1 Inhibitors of hcv ns5b polymerase
01/07/2004EP1377567A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
01/07/2004EP1377555A1 Novel compounds
01/07/2004EP1377554A1 Antagonism of immunostimulatory cpg-oligonucleotides by 4-aminoquinolines and other weak bases
01/07/2004EP1377553A1 Tetrahydroquinoline derivatives as stat6-modulators, preparation and use thereof
01/07/2004EP1377550A1 Phenyl heterocyclyl ether derivatives as serotonin re-uptake inhibitors
01/07/2004EP1377283A2 Compounds of the formula r1-x-y-z-nr2r3 as abca-1 elevating agents against coronary artery disease or atherosclerosis
01/07/2004EP1175417B1 Substituted benzolactam compounds
01/07/2004EP1056733B1 Histamine h3 receptor ligands
01/07/2004CN1466575A Quinolene derivatives as anti-inflammation agents
01/07/2004CN1133432C Aqueous liquid preparations
01/06/2004US6673801 Dihydroxyhexanoic acid derivatives
01/02/2004EP1375487A1 Process for producing quinoline-3-carboxylic acid compound
01/02/2004EP1375486A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity
01/02/2004EP1375485A1 Method for preparing 7-quinolinyl-3,5-dihydroxyhept-6-enoate
01/02/2004EP1374867A1 Use of chloroquine, hydroxychloroquine and 4 amino-quinolinic derivatives to obtain a drug for the anti retroviral therapy, active towards hiv sensitive strains and towards hiv strains which are resistant to both nucleosidic and non-nucleosidic reverse transcriptase inhibitors and to proteases inhibitors
01/02/2004EP1373240A2 Retinoid x receptor modulators
01/02/2004EP1373233A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
01/02/2004EP1373211A1 Quinoline derivatives and their use as antibiotics
01/02/2004EP1373192A1 N-phenpropylcyclopentyl-substituted glutaramide derivatives as nep inhibitors for fsad
01/02/2004EP1373191A1 Acylated indanyl amines and their use as pharmaceuticals
01/02/2004EP1372655A2 Cathepsin cysteine protease inhibitors
01/02/2004EP1372654A2 Quinoline inhibitors of hyak1 and hyak3 kinases
01/02/2004EP1044187B1 N-benzyl-3-indenylacetamides derivatives for treating neoplasia
01/01/2004US20040002604 Phenylalkynes
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
01/01/2004US20040002506 Antiproliferative agents; antitumor agents
01/01/2004US20040002493 Benzoic acid derivatives and pharmaceutical agents comprising the same as active ingredient
01/01/2004US20040002123 Detection of transmembrane potentials by optical methods
01/01/2004US20040001970 Organic electroluminescent materials and devices made from such materials
12/2003
12/31/2003WO2004000828A1 New compounds useful for the treatment of obesity, type ii diabetes and cns disorders
12/31/2003WO2004000814A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003WO2004000797A1 Alpha-sulfonylamino-acetonitriles
12/31/2003CN1132818C 用作抗病毒剂的4-氧代-1,4-二氢-3-喹啉甲酰胺 As antiviral agents 4-oxo-1,4-dihydro-3-quinoline carboxamide
12/31/2003CA2490043A1 8-(biaryl) quinoline pde4 inhibitors
12/31/2003CA2486989A1 New compounds useful for the treatment of obesity, type ii diabetes and cns disorders
12/30/2003US6670645 Bright, efficient, stable; increased volatility for lower temperature vacuum deposition preventing decomposition
12/30/2003US6670377 Quinoline derivatives, having in particular antiviral properties, preparation and biological applications thereof
12/30/2003US6670376 Aryl aniline β2 adrenergic receptor agonists
12/29/2003CA2433983A1 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
12/28/2003CA2433237A1 Use of chloroquine, hydroxy chloroquine and 4 amino-quinolinic derivatives to obtain a drug for the anti retroviral therapy, active towards hiv sensitive strains and towards hiv strains which are resistant to both nucleosidic and nonnucleosidic reverse transcriptase inhibitors and to proteases inhibitors
12/25/2003WO2003106424A1 Process for the manufacture of quinoline derivatives
12/25/2003US20030236281 Quinoline derivatives(2)
12/25/2003US20030236280 Aminotetralin-derived urea modulators of vanilloid VR1 receptor
12/25/2003US20030236259 Novel aryl- and heteroarylpiperazines
12/24/2003WO2003106425A2 Phenyl- and pyridyl-diazaheterocycles having a tnf-modulating activity
12/24/2003WO2003106423A1 Cyclic amine and medicinal composition containing the same
12/24/2003WO2003106422A1 BLUE EMITTING TRIS (8-OXOQUINOLINE) ALUMINUM (III) (AlQ3)
12/24/2003WO2003106421A2 Phenylalkylamines and pyridylalkylamines
12/24/2003WO2003106390A1 Polymerisation inhibitor
12/24/2003WO2003105851A1 Novel crystalline forms of gatifloxacin
12/24/2003WO2003105850A1 2-aminoquinolines as melanin concentrating hormone receptor antagonists
12/24/2003WO2003105849A1 Tetrahydroquinolines for modulating the expression of exogenous genes via an ecdysone receptor complex
12/24/2003WO2003074025A3 Pressurised metered dose inhalers containing solutions of beta-2 agonists
12/24/2003WO2003068760A3 Compounds possessing affinity at 5ht1-type receptors and use thereof in therapy of cns disorders
12/24/2003WO2003039454A3 Beta-secretase inhibitors and methods of use
12/24/2003CN1463191A Low hygroscopic aripiprazole drug substance and processes for prepn. thereof
12/24/2003CA2489377A1 Novel crystalline forms of gatifloxacin
12/24/2003CA2488407A1 Tetrahydroquinolines for modulating the expression of exogenous genes via an ecdysone receptor complex
12/23/2003US6667307 HIV protease
12/18/2003WO2003104221A1 Inhibitors of the gpib -vwf interaction, their preparation and use
12/18/2003WO2003104195A1 4-(aryl or heteroaryl) -2-butylamine derivatives and their use as glucocorticoid ligans
12/18/2003WO2003103671A1 Basic non-peptide bradykinin antagonists and pharmaceutical compositions therefrom
12/18/2003WO2003103668A1 Pyridin-2-one and quinolin-2-one derivatives, preparation thereof and use thereof as antibacterials
12/18/2003US20030233001 Process for the manufacture of organic compounds
12/18/2003US20030232990 For therapy of arteriosclerosis and dyslipidaemias
12/18/2003US20030232989 Process for the preparation of specific aromatic aldehydes
12/18/2003US20030232868 Cyclic carboxylic acids as integrin antagonists
12/18/2003US20030232863 Cathepsin cysteine protease inhibitors
12/18/2003US20030232859 Antiinflammatory agents; for treatment of rheumatoid arthritis and multiple sclerosis
12/18/2003US20030232854 Such as 3-methyl-5-(2-chloro-6-fluorophenyl)-4-isoxazole-carboxylic acid ethyl ester for inhibiting multidrug resistance protein (MRP1)
12/18/2003US20030232846 Caspase inhibitors and uses thereof
12/18/2003US20030232844 Dihydrobenzopyrans, dihydrobenzothiopyrans, and tetrahydroquinolines for the treatment of cox-2 mediated disorders
12/18/2003US20030232808 Sulfonyl derivatives
12/18/2003US20030232807 Dietetic agents
12/18/2003US20030232802 Aryl and heteroaryl sulfonates
12/18/2003US20030232801 Identification of compounds for the treatment or prevention of proliferative diseases
12/18/2003US20030232792 Useful for male contraception, treatment of a variety of hormone-related conditions such as sexual disorders, prostate cancer
12/18/2003DE10215316C1 Chinolin- und Isochinolin-Derivate, ein pharmazeutisches Mittel und ihre Verwendung als Entzündungshemmer Quinoline and isoquinoline derivatives, to a pharmaceutical agent and their use as anti-inflammatory agents
12/18/2003CA2488193A1 Inhibitors of the gpib -vwf interaction, their preparation and use
12/18/2003CA2486491A1 4-(aryl or heteroaryl)-2-butylamine derivatives and their use as glucocorticoid ligans
12/17/2003EP1370532A1 Method for producing cyclopentadiene compounds
12/17/2003EP0934276B1 Anthranilic acid derivatives as multi drug resistance modulators
12/17/2003CN1462273A Bicyclic heteroaromatic compounds
12/17/2003CN1461748A Synthesis process of jiatisasin
12/17/2003CN1131214C Tetrahy droquimoline derivatives as EAA antagonists
12/17/2003CN1131213C Carbostyril derivatives as antithrombotic agents
12/17/2003CN1131211C Heteraryl diazacy cloa lkanes as cholinergic ligands at nicotinic acetylcholine receptors
12/17/2003CN1131202C Calcium receptor-active compounds
12/16/2003US6664393 N-guanidinoalkylamides, their preparation, their use, and pharmaceutical preparations comprising them
12/16/2003CA2269547C Process for converting nitrogen-containing hydroxy heteroaromatics to arylamines
12/11/2003WO2003101941A2 Alpha acyloxyacetamides for kallikrein and urokinase inhibition
12/11/2003WO2003101442A1 Peptide deformylase inhibitors
12/11/2003WO2003064382A3 Process for the manufacture of organic compounds
12/11/2003WO2003024395A3 Linked biaryl compounds