Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
07/2005
07/21/2005WO2005066115A2 Disubstituted chalcone oximes having rarϝ retinoid receptor antagonist activity
07/21/2005WO2005043124A3 Chiral 1,8-diarylnaphthalenes, methods of making them, and their use as sensors
07/21/2005WO2005042712A3 Heterocyclic compounds and methods of making and using thereof
07/21/2005WO2005033119A9 Supramolecular compounds and their use as antitumour and antiviral agents
07/21/2005WO2004050609A8 Substituted ureas and carbamates
07/21/2005US20050159480 Preparation of statins by reacting (trisubstituted phosphoranylidenecarbonyl)acetates with benzaldehydes, reduction with diamino-group 8 metal coordinates, condensation with 1-hydroxy-1-alkoxyethylenes, hydrolysis, and optionally converting the carboxy acid product into a salt or a lactone
07/21/2005US20050159448 Aryl aniline derivatives as beta2 adrenergic receptor agonists
07/21/2005US20050159447 Quinoline derivative anticarcinogenic compounds; based on herbicides
07/21/2005US20050159446 of preparing 4-substituted quinoline compounds as intermediates in the manufacture of receptor tyrosine kinase inhibitors and intermediate compounds used in the methods thereof, wherein the 4-substituted quinoline compound has the following general formula (I):
07/21/2005US20050159429 Novel crystalline forms of aripiprazole
07/21/2005US20050159421 Ethylene diamine derivatives and their use as orexin-receptor antagonists
07/21/2005DE10360154A1 New 2-(hetero)aryl-tetrahydroquinoline derivatives and 1,2,3,4-tetrahydro-1,5-naphthyridine derivatives are mitotic motor protein Eg5 inhibitors used as anticancer agents for treating carcinoma or leukemia
07/21/2005CA2552090A1 Disubstituted chalcone oximes as selective agonists of rar.gamma. retinoid receptors
07/21/2005CA2551294A1 Disubstituted chalcone oximes having rary retinoid receptor antagonist activity
07/20/2005EP1554260A1 Aryloxyalkylamine derivatives as h3 receptor ligands
07/20/2005EP1554249A2 1-pyridin-4-yl-urea derivatives
07/20/2005EP1554243A1 Bicyclic benzamide compounds as histamine h3 receptor ligand useful in the treatment of neurological diseases
07/20/2005EP1554239A2 Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists
07/20/2005CN1642931A Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
07/20/2005CN1642917A Non-peptide GnRH antagonists
07/20/2005CN1642915A Benzamide derivatives useful as histone deacetylase inhibitors
07/20/2005CN1642580A Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
07/20/2005CN1211369C L-amino acid acyl-(8-quinolyl) amine platinum (II) complex and prep. and use thereof
07/20/2005CN1211331C Method for isomerisation of allyl alcohols
07/19/2005US6919470 Aryl and heteroaryl sulfonates
07/19/2005US6919353 Enzyme inhibitors of phosphordiesterase 4 having minimal side effects; antiinflammatory agents; antiallergens; asthma; neurodegenerative disorders; antidiabetic agents; pain; anti-tumor, -carcinogenic and -arthritic agents
07/19/2005US6919347 Antidiabetic agents; antiinflammatory agents; analgesics; antiallergens
07/19/2005US6919339 ABCA-1 elevating compounds
07/19/2005US6919335 Heterocycles that are inhibitors of IMPDH enzyme
07/14/2005WO2005064006A1 OPTICALLY ACTIVE, HETEROAROMATIC β-HYDROXY ESTERS, PROCESSES FOR THEIR PREPARATION FROM β-KETO ESTERS AND PROCESSES FOR THE PREPARATION OF THESE β-KETO ESTERS
07/14/2005WO2005063713A1 Crystal of salt of 4-(3-chloro-4-(cyclopropylaminocarbonyl)amino-phenoxy)-7-methoxy-6-quinolinecarboxamide or of solvate thereof and processes for producing these
07/14/2005WO2005063712A1 5-ht2 receptors modulators, their pharmaceuticals compositions and their use for the treatment of cardiovascular and muscle diseases
07/14/2005WO2005063711A1 Crystal form of quinoline compound and process for its production
07/14/2005WO2005063689A1 Benzamide derivative
07/14/2005WO2005063244A1 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
07/14/2005WO2005063239A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/14/2005WO2005035514A3 Modulators of atp-binding cassette transporters containing cycloalkyl or pyranyl groups
07/14/2005WO2005017185A3 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS
07/14/2005US20050154230 Urea derivatives
07/14/2005US20050154202 Substituted aryl amides
07/14/2005US20050154013 Pressurised metered dose inhalers containing solutions of beta-2 agonists
07/14/2005US20050154008 Aryl fused substituted 4-oxy-pyridines
07/14/2005US20050153974 Heterocyclymethylpiperidines and -piperazines possessing affinity at 5ht-1 type receptors
07/14/2005US20050153964 Novel compounds
07/14/2005US20050153957 Beta2-adrenoceptor agonists
07/14/2005US20050153942 Heterocyclic inhibitors of MEK and methods of use thereof
07/14/2005US20050152981 jet crystallization utilizes two jet streams that strike each other head-on; streams carries a solution rich in the aripiprazole and the other carries an anti-solvent, such as water
07/14/2005US20050152846 Hydrofluoroalkane (HFA) propellant and co-solvents; inhalants; storage stability; deep lung penetration
07/14/2005CA2551552A1 5-ht2 receptors modulators, their pharmaceuticals compositions and their use for the treatment of cardiovascular and muscle diseases
07/14/2005CA2551227A1 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
07/14/2005CA2551050A1 Crystal form of quinoline compound and process for its production
07/14/2005CA2550649A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/14/2005CA2546981A1 Optically active, heteroaromatic .beta.-hydroxy esters, processes for their preparation from .beta.-keto esters and processes for the preparation of these .beta.-keto esters
07/13/2005EP1553092A1 Aralkyl formyl-alkyl piperazine derivatives and their uses as cerebral nerve protective agent
07/13/2005EP1551829A2 Novel compounds with antibacterial activity
07/13/2005EP1551807A1 Improved reagents for n-amination
07/13/2005EP1551798A1 Novel sulphones for inhibition of gamma secretase
07/13/2005EP1448529B1 Sulfone derivatives suitable for the treatment of autoimmune diseases and allergies
07/13/2005EP1161415B1 N-cyanomethylamides as protease inhibitors
07/13/2005CN1639130A Process for producing fused imidazole compound, reformatsky reagent in stable form, and process for producing the same
07/13/2005CN1639119A Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
07/13/2005CN1639096A Process for producing trans-4-amino-1-cyclohexanecarboxylic acid derivative
07/13/2005CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
07/13/2005CN1638730A Formoterol superfine formulation
07/13/2005CN1638729A Pressurised metered dose inhalers containing solutions of beta-2 agonists
07/13/2005CN1636986A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636985A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636984A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636976A Mutilin derivatives and their use as antibacterials
07/13/2005CN1636597A Compounds for the treatment of female sexual dysfunction
07/13/2005CN1210263C N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
07/12/2005US6916957 Antiinflammatory agents; antihistamines; antiallergens
07/12/2005US6916831 Oxo acids and salts such as 2-Phenyl-4-quinolone-8-acetic acid, used for prophylaxis of cancers; antitumor agents
07/12/2005US6916812 Dietetic agents
07/12/2005CA2319542C The treatment of sexual dysfunction in certain patient groups
07/12/2005CA2094494C A 4-quinolone antibiotic compound as gamma ray scintigraphy diagnostic imaging agent
07/07/2005WO2005061475A2 Ornithine derivatives as prostaglandin e2 agonists or antagonists
07/07/2005WO2005061459A1 Biaryl sulfonamides and methods for using same
07/07/2005WO2005060963A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
07/07/2005WO2005060748A1 Fungicide
07/07/2005WO2005060456A2 Method for treating adamts-5-associate disease
07/07/2005WO2005047258A3 Methods and compositions for selectin inhibition
07/07/2005WO2005047257A3 Methods and compositions for selectin inhibition
07/07/2005WO2005042498A3 4-amino (aza) quinoline derivatives as capsaicin receptor agonists
07/07/2005WO2005034869A3 Compounds and compositions as protein kinase inhibitors
07/07/2005US20050148777 (2R)-6-chloro-7-isobutyl-2-(trifluoromethyl)-2H-chromene-3-carboxylic acid; cyclooxygenase-2 mediated disorders
07/07/2005US20050148648 Cystic fibrosis transmembrane conductance regulator; ABC transporter mediated diseases like cystic fibrosis; 5-methoxy-N-((1-(3,4-dimethoxyphenyl)-cyclohexyl)methyl)benzofuran-2-carboxamide; or sulfonamide analogs; chloride or bicarbonate channel modulators
07/07/2005US20050148631 Modulation of steroid enzymes in mammals as antidiabetic agents, for treatment of obesity, vision defects, lowering fats in blood, for treatment of osteoporosis, tuberculosis or atherosclerosis in mammals
07/07/2005US20050148627 Benzopyran compounds for use in the treatment and prevention of inflammation related conditions
07/07/2005US20050148626 Novel thromodulin expression promoters
07/07/2005US20050148605 Modulation of protein tyrosine kinases for treatment of diseases with prodrugs
07/07/2005US20050148595 heterocylcyclic amines used for treating or preventing conditions ameliorated by monoamine reuptake such as vasomotor symptoms, sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
07/07/2005US20050148590 4-[3-Hydroxyimino-3-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-propenyl]-benzoic acid; emphysema; respiratory system and skin disorder; acne and psoriasis; side effect reduction; improved pharmacology
07/07/2005US20050148581 Quinolines; 1-(6-bromo-2-methoxy-quinolin-3-yl)-4-dimethylamino-2-naphthalen-1-yl-1-phenyl-butan-2-ol; Mycobacterium tuberculosis, M. bovis, M. avium and M. marinum; reduces the total length of treatment and the frequency of drug administration; multi-drug and antibiotic resistance
07/07/2005CA2550958A1 Ornithine derivatives as prostaglandin e2 agonists or antagonists
07/07/2005CA2549651A1 Benzenesulfonylamino-pyridin-2-yl derivatives and related compounds as inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1 (11-beta-hsd-1) for the treatment of diabetes and obesity
07/07/2005CA2548513A1 Biaryl sulfonamides and methods for using same
07/07/2005CA2547575A1 Method for treating adamts-5-associated disease
07/06/2005EP1549613A1 Sulfonamides having antiangiogenic and anticancer activity
07/06/2005CN1636004A Process for the manufacture of hmg-coa reductase inhibitory mevalonic acid derivatives