Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273) |
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09/08/2000 | WO2000051975A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors |
09/08/2000 | WO2000051974A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7 - receptor antagonists |
09/08/2000 | WO2000051973A1 Cyclobutene-3,4-dione derivatives, preparation method and therapeutic use |
09/08/2000 | WO2000051972A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy |
09/08/2000 | WO2000051970A1 Amide compounds for the potentiation of cholinergic activity |
09/08/2000 | CA2366954A1 Dihetero-substituted metalloprotease inhibitors |
09/08/2000 | CA2365032A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy |
09/08/2000 | CA2364878A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors |
09/08/2000 | CA2361164A1 Nitroxyderivatives having antiinflammatory, analgesic and antithrombotic activity |
09/08/2000 | CA2361162A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7-receptor antagonists |
09/07/2000 | DE19908938A1 Übergangsmetallverbindung, Katalysatorsystem, Verfahren zu seiner Herstellung und seine Verwendung zur Polymerisation von Olefinen Transition metal compound catalyst system, to methods for its production and its use for the polymerization of olefins |
09/06/2000 | EP1033371A1 Transition metal compound, catalyst system, process for the preparation thereof and its use for the polymerization of olefins |
09/06/2000 | EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists |
09/06/2000 | EP1032562A2 Advanced glycation end-product intermediaries and post-amadori inhibition |
09/06/2000 | EP1032559A1 Aminoalkylphenol derivatives and related compounds |
09/06/2000 | EP1032556A1 Pharmaceutically active compounds and methods of use |
09/06/2000 | EP1032377A1 Substituted 2-aminoacetamides and the use thereof |
09/06/2000 | EP0824514B1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production |
09/06/2000 | CN1265669A Compounds which inhibit leukocyte adhesion mediated by VLA-4 |
09/06/2000 | CN1265654A 1-(N-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of phenyl ring |
09/06/2000 | CN1265647A Acrylic metalloprotease inhibitor |
09/06/2000 | CN1265645A Urokinase inhibitors |
09/06/2000 | CN1265642A Aryloxyaniline derivatives |
09/06/2000 | CN1265393A Process for preparing N-(amino-4,6-dihalopyrimidine) formamide |
09/06/2000 | CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease |
09/05/2000 | US6114580 Catalyst for making herbicides |
09/05/2000 | US6114535 Process and intermediates for the manufacture of pyridine-2,3-dicarboxylate compounds |
09/05/2000 | US6114524 Process for producing halogenated heteroaryl compounds |
09/05/2000 | US6114493 Contacting a compound to be phosgenated with an excess of a phosgene source in the form of a solid phase reagent; supports in combinatorial synthesis for the creation of libraries of compounds for lead identification |
09/05/2000 | US6114386 1-((substituted)alkylcarbonylamino),2-(hydroxyl or amino)-substituted benzene compounds of given formula; treating and preventing bacterial or trypanosomal infection using the inhibitor |
09/05/2000 | US6114375 Substituted cyclopropyl phenoxymethyl phenyl carbamates and their use as fungicides |
09/05/2000 | US6114364 2-((substituted)alkyl(thio, sulfonyl, or sulfoxy)methyl), 3-(carboxyl or aliphatic hydrocarbonyl)cyclopentan-1-one derivatives, except cystacyclin; use as neuron differentiation accelerator |
09/05/2000 | US6114363 Pyridyl phenyl and benzyl ethers, process and intermediate products for their preparation and their use as fungicides and for controlling animal pests |
09/05/2000 | US6114357 Hemoregulatory compounds |
08/31/2000 | WO2000050872A2 A system for cell-based screening |
08/31/2000 | WO2000050431A1 Platinum (ii) compounds |
08/31/2000 | WO2000050408A1 Pyridazin-3-one derivatives and medicines containing the same |
08/31/2000 | WO2000050403A1 N-[2-hydroxy-3-(1-piperidinyl)propoxy]pyridine-1-oxide-3-carboximidoyl chloride and its use in the treatment of insulin resistance |
08/31/2000 | WO2000050402A1 Pde iv inhibiting compounds, compositions and methods of treatment |
08/31/2000 | WO2000050401A1 3-phenylpyridine derivatives and their use as nk-1 receptor antagonists |
08/31/2000 | WO2000050400A1 2-aminopyridines containing fused ring substituents |
08/31/2000 | WO2000050399A1 Inhibitors of cellular niacinamide mononucleotide formation and their use in cancer therapy |
08/31/2000 | WO2000050398A2 Phenyl- and pyridinyl derivatives as neurokinin 1 antagonists |
08/31/2000 | WO2000050392A1 2-mercaptocarboxylic acid derivatives |
08/31/2000 | WO2000050390A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production |
08/31/2000 | WO2000050389A1 Efficient carbamate synthesis |
08/31/2000 | WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines |
08/31/2000 | WO2000050376A2 Efficient synthesis of alkyl carbonates |
08/31/2000 | WO2000040558A8 Aspartic protease inhibitors |
08/31/2000 | DE10008042A1 Neurokinin-1-Rezeptorantagonisten Neurokinin-1 receptor antagonists |
08/31/2000 | CA2364804A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production |
08/31/2000 | CA2364712A1 Platinum (ii) compounds |
08/31/2000 | CA2364653A1 Pde iv inhibiting compounds, compositions and methods of treatment |
08/30/2000 | EP1031570A1 Immuno-modulator exhibiting anti-microbial and anti-mycobacterial activities, method for producing the same and pharmaceutical preparation for treating mycobacterioses as well as lung chronic and non specific conditions, sexually transmitted diseases and the resulting immuno-deficiency |
08/30/2000 | EP1031564A1 Inhibitors of cellular nicotinamide mononucleotide formation and their use in cancer therapy |
08/30/2000 | EP1031563A1 Sulfonyl derivatives |
08/30/2000 | EP1030842A1 Metalloproteinase inhibitors |
08/30/2000 | EP1030840A1 Cyclic amine derivatives and their use as drugs |
08/30/2000 | EP1030831A1 Process for the preparation of azacycloalkylalkanoyl pseudotetrapeptides |
08/30/2000 | EP0888297B1 N-arylsulfilimine compounds and their use as catalysts in the preparation of n-arylarylsulfonamide compounds |
08/30/2000 | CN1265098A Heterocyclic derivatives which inhibit factor XA |
08/30/2000 | CN1265096A Hydrazine derivatives |
08/29/2000 | US6111113 Reacting methacrolein and methyl ethyl ketone with ammonia in a gas phase in the presence of a catalyst comprising silica-alumina containg at least one metal selected from cadmium and lead; catalytic durability; by-product inhibition |
08/29/2000 | US6111112 Etherification of the reaction product, isopropylidene-malonitrile, with triethyl orthoformate; cyclization; diazotization; chlorination; acidolysis; and hoffman rearrangement; intermediate for |
08/29/2000 | US6110970 For treating or preventing or ameliorating cancer and other proliferative diseases as well as for inducing wound healing, treating cutaneous ulcers, treating gastrointestinal disorders, treating blood disorders such as anemias |
08/29/2000 | US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents |
08/29/2000 | US6110946 An enzyme inhibitors of retroviral aspartate protease for the treatment of aids |
08/29/2000 | US6110945 An antiinflammatory agent inhibiting the binding of integrins to their ligands; in the prophylaxis for treating immune or inflammatory disorders |
08/29/2000 | US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor |
08/29/2000 | US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
08/29/2000 | US6110871 2-((phenyl, pyridyl or pyrazolyl)(oxy or thio)), 6-((substituted)phenyl)-cyanopyridines; herbicidal activity with the necessary selectivity and enhanced soil degradation |
08/24/2000 | WO2000049015A1 Pyridine compounds and their pharmaceutical use |
08/24/2000 | WO2000049007A1 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s |
08/24/2000 | WO2000048998A1 Amino(thio)phenols and their therapeutic use |
08/24/2000 | WO2000048997A1 SUBSTITUTED ACETYLPYRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION OF INTERMEDIATES FOR OPTICALLY ACTIVE β3 AGONIST BY THE USE OF THE SAME |
08/24/2000 | WO2000048996A2 β-ALANINE DERIVATIVES |
08/24/2000 | WO2000048994A1 Thioamide derivatives |
08/24/2000 | WO2000048993A1 Arylaminoalkylamides |
08/24/2000 | WO2000048992A1 Acylated aminoacetonitriles as cysteine protease inhibitors |
08/24/2000 | WO2000048988A1 Phenylalaninol derivatives |
08/24/2000 | WO2000002887B1 Ligands for metals and metal-catalyzed processes |
08/24/2000 | CA2371824A1 .beta.-alanine derivatives |
08/24/2000 | CA2362070A1 Substituted acetylpyridine derivatives and process for the preparation of intermediates for optically active .beta.3 agonist by the use of the same |
08/23/2000 | EP1029909A1 Organic electroluminescence device and phenylenediamine derivative |
08/23/2000 | EP1029851A1 Piperazine compounds and medicinal use thereof |
08/23/2000 | EP1028945A1 Substituted pyridine compounds as anti-inflammatory agents |
08/23/2000 | EP1028944A1 Fluorinated naphthalene derivatives and their use in liquid crystal mixtures |
08/23/2000 | EP1028942A2 Dipeptide nitriles |
08/23/2000 | EP1028941A2 Compounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition |
08/23/2000 | EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation |
08/23/2000 | EP0876344B1 Pyridylacetic acid derivatives, method and intermediate products for producing them and agents containing them |
08/23/2000 | EP0876334B1 Phenylacetic acid derivatives, process for their preparation and their use as pesticides and fungicides |
08/23/2000 | EP0836596B1 Hydrazine derivatives |
08/23/2000 | EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides |
08/23/2000 | EP0763005B1 TETRAHYDROINDENO[1,2-d][1,3,2]OXAZABOROLES AND THEIR USE AS ENANTIOSELECTIVE CATALYSTS |
08/23/2000 | EP0711289B1 Piperazine compounds used in therapy |
08/23/2000 | EP0708772B1 IMIDAZO [4,5-c]PYRIDIN-4-AMINES |
08/23/2000 | EP0667859B1 Molecule labelling using 2-hydraninopyridine derivatives |
08/23/2000 | EP0640072B1 Derivatives of pyridine as hydroxylase and lyase inhibitors |
08/23/2000 | EP0637297B1 Compounds having selectivity for retinoid x receptors |