Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
09/2000
09/08/2000WO2000051975A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/08/2000WO2000051974A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7 - receptor antagonists
09/08/2000WO2000051973A1 Cyclobutene-3,4-dione derivatives, preparation method and therapeutic use
09/08/2000WO2000051972A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
09/08/2000WO2000051970A1 Amide compounds for the potentiation of cholinergic activity
09/08/2000CA2366954A1 Dihetero-substituted metalloprotease inhibitors
09/08/2000CA2365032A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
09/08/2000CA2364878A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/08/2000CA2361164A1 Nitroxyderivatives having antiinflammatory, analgesic and antithrombotic activity
09/08/2000CA2361162A1 Alpha-aminoacetic acid derivatives useful as alpha 4 beta 7-receptor antagonists
09/07/2000DE19908938A1 Übergangsmetallverbindung, Katalysatorsystem, Verfahren zu seiner Herstellung und seine Verwendung zur Polymerisation von Olefinen Transition metal compound catalyst system, to methods for its production and its use for the polymerization of olefins
09/06/2000EP1033371A1 Transition metal compound, catalyst system, process for the preparation thereof and its use for the polymerization of olefins
09/06/2000EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists
09/06/2000EP1032562A2 Advanced glycation end-product intermediaries and post-amadori inhibition
09/06/2000EP1032559A1 Aminoalkylphenol derivatives and related compounds
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000EP1032377A1 Substituted 2-aminoacetamides and the use thereof
09/06/2000EP0824514B1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production
09/06/2000CN1265669A Compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265654A 1-(N-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of phenyl ring
09/06/2000CN1265647A Acrylic metalloprotease inhibitor
09/06/2000CN1265645A Urokinase inhibitors
09/06/2000CN1265642A Aryloxyaniline derivatives
09/06/2000CN1265393A Process for preparing N-(amino-4,6-dihalopyrimidine) formamide
09/06/2000CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease
09/05/2000US6114580 Catalyst for making herbicides
09/05/2000US6114535 Process and intermediates for the manufacture of pyridine-2,3-dicarboxylate compounds
09/05/2000US6114524 Process for producing halogenated heteroaryl compounds
09/05/2000US6114493 Contacting a compound to be phosgenated with an excess of a phosgene source in the form of a solid phase reagent; supports in combinatorial synthesis for the creation of libraries of compounds for lead identification
09/05/2000US6114386 1-((substituted)alkylcarbonylamino),2-(hydroxyl or amino)-substituted benzene compounds of given formula; treating and preventing bacterial or trypanosomal infection using the inhibitor
09/05/2000US6114375 Substituted cyclopropyl phenoxymethyl phenyl carbamates and their use as fungicides
09/05/2000US6114364 2-((substituted)alkyl(thio, sulfonyl, or sulfoxy)methyl), 3-(carboxyl or aliphatic hydrocarbonyl)cyclopentan-1-one derivatives, except cystacyclin; use as neuron differentiation accelerator
09/05/2000US6114363 Pyridyl phenyl and benzyl ethers, process and intermediate products for their preparation and their use as fungicides and for controlling animal pests
09/05/2000US6114357 Hemoregulatory compounds
08/2000
08/31/2000WO2000050872A2 A system for cell-based screening
08/31/2000WO2000050431A1 Platinum (ii) compounds
08/31/2000WO2000050408A1 Pyridazin-3-one derivatives and medicines containing the same
08/31/2000WO2000050403A1 N-[2-hydroxy-3-(1-piperidinyl)propoxy]pyridine-1-oxide-3-carboximidoyl chloride and its use in the treatment of insulin resistance
08/31/2000WO2000050402A1 Pde iv inhibiting compounds, compositions and methods of treatment
08/31/2000WO2000050401A1 3-phenylpyridine derivatives and their use as nk-1 receptor antagonists
08/31/2000WO2000050400A1 2-aminopyridines containing fused ring substituents
08/31/2000WO2000050399A1 Inhibitors of cellular niacinamide mononucleotide formation and their use in cancer therapy
08/31/2000WO2000050398A2 Phenyl- and pyridinyl derivatives as neurokinin 1 antagonists
08/31/2000WO2000050392A1 2-mercaptocarboxylic acid derivatives
08/31/2000WO2000050390A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/31/2000WO2000050389A1 Efficient carbamate synthesis
08/31/2000WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines
08/31/2000WO2000050376A2 Efficient synthesis of alkyl carbonates
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/31/2000DE10008042A1 Neurokinin-1-Rezeptorantagonisten Neurokinin-1 receptor antagonists
08/31/2000CA2364804A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/31/2000CA2364712A1 Platinum (ii) compounds
08/31/2000CA2364653A1 Pde iv inhibiting compounds, compositions and methods of treatment
08/30/2000EP1031570A1 Immuno-modulator exhibiting anti-microbial and anti-mycobacterial activities, method for producing the same and pharmaceutical preparation for treating mycobacterioses as well as lung chronic and non specific conditions, sexually transmitted diseases and the resulting immuno-deficiency
08/30/2000EP1031564A1 Inhibitors of cellular nicotinamide mononucleotide formation and their use in cancer therapy
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030842A1 Metalloproteinase inhibitors
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030831A1 Process for the preparation of azacycloalkylalkanoyl pseudotetrapeptides
08/30/2000EP0888297B1 N-arylsulfilimine compounds and their use as catalysts in the preparation of n-arylarylsulfonamide compounds
08/30/2000CN1265098A Heterocyclic derivatives which inhibit factor XA
08/30/2000CN1265096A Hydrazine derivatives
08/29/2000US6111113 Reacting methacrolein and methyl ethyl ketone with ammonia in a gas phase in the presence of a catalyst comprising silica-alumina containg at least one metal selected from cadmium and lead; catalytic durability; by-product inhibition
08/29/2000US6111112 Etherification of the reaction product, isopropylidene-malonitrile, with triethyl orthoformate; cyclization; diazotization; chlorination; acidolysis; and hoffman rearrangement; intermediate for
08/29/2000US6110970 For treating or preventing or ameliorating cancer and other proliferative diseases as well as for inducing wound healing, treating cutaneous ulcers, treating gastrointestinal disorders, treating blood disorders such as anemias
08/29/2000US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents
08/29/2000US6110946 An enzyme inhibitors of retroviral aspartate protease for the treatment of aids
08/29/2000US6110945 An antiinflammatory agent inhibiting the binding of integrins to their ligands; in the prophylaxis for treating immune or inflammatory disorders
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110871 2-((phenyl, pyridyl or pyrazolyl)(oxy or thio)), 6-((substituted)phenyl)-cyanopyridines; herbicidal activity with the necessary selectivity and enhanced soil degradation
08/24/2000WO2000049015A1 Pyridine compounds and their pharmaceutical use
08/24/2000WO2000049007A1 Acetamido acetonitrile derivatives as inhibitors of cathepsin l and/or cathepsin s
08/24/2000WO2000048998A1 Amino(thio)phenols and their therapeutic use
08/24/2000WO2000048997A1 SUBSTITUTED ACETYLPYRIDINE DERIVATIVES AND PROCESS FOR THE PREPARATION OF INTERMEDIATES FOR OPTICALLY ACTIVE β3 AGONIST BY THE USE OF THE SAME
08/24/2000WO2000048996A2 β-ALANINE DERIVATIVES
08/24/2000WO2000048994A1 Thioamide derivatives
08/24/2000WO2000048993A1 Arylaminoalkylamides
08/24/2000WO2000048992A1 Acylated aminoacetonitriles as cysteine protease inhibitors
08/24/2000WO2000048988A1 Phenylalaninol derivatives
08/24/2000WO2000002887B1 Ligands for metals and metal-catalyzed processes
08/24/2000CA2371824A1 .beta.-alanine derivatives
08/24/2000CA2362070A1 Substituted acetylpyridine derivatives and process for the preparation of intermediates for optically active .beta.3 agonist by the use of the same
08/23/2000EP1029909A1 Organic electroluminescence device and phenylenediamine derivative
08/23/2000EP1029851A1 Piperazine compounds and medicinal use thereof
08/23/2000EP1028945A1 Substituted pyridine compounds as anti-inflammatory agents
08/23/2000EP1028944A1 Fluorinated naphthalene derivatives and their use in liquid crystal mixtures
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP1028941A2 Compounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
08/23/2000EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation
08/23/2000EP0876344B1 Pyridylacetic acid derivatives, method and intermediate products for producing them and agents containing them
08/23/2000EP0876334B1 Phenylacetic acid derivatives, process for their preparation and their use as pesticides and fungicides
08/23/2000EP0836596B1 Hydrazine derivatives
08/23/2000EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
08/23/2000EP0763005B1 TETRAHYDROINDENO[1,2-d][1,3,2]OXAZABOROLES AND THEIR USE AS ENANTIOSELECTIVE CATALYSTS
08/23/2000EP0711289B1 Piperazine compounds used in therapy
08/23/2000EP0708772B1 IMIDAZO [4,5-c]PYRIDIN-4-AMINES
08/23/2000EP0667859B1 Molecule labelling using 2-hydraninopyridine derivatives
08/23/2000EP0640072B1 Derivatives of pyridine as hydroxylase and lyase inhibitors
08/23/2000EP0637297B1 Compounds having selectivity for retinoid x receptors