Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
06/2005
06/02/2005WO2005049087A1 Remedy for chronic pelvic pain syndrome
06/02/2005WO2005049023A1 Glyt1 transporter inhibitors
06/02/2005WO2005049009A1 Methods and agents for inhibiting dynamin-dependent endocytosis
06/02/2005WO2005023794A3 Compound libraries of 4-carboxamidopiperidine derivatives
06/02/2005WO2005009961B1 Fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions
06/02/2005WO2004063150A3 Diagnostic and therapeutic alkyl piperidine/piperazine compounds and process
06/02/2005WO2004039781A9 Platinum complexes
06/02/2005WO2003075847A3 NOVEL CURCUMINOID-FACTOR VIIa CONSTRUCTS AS SUPPRESSORS OF TUMOR GROWTH AND ANGIOGENESIS
06/02/2005US20050119332 Substituted thiophene compounds as modulators of protein tyrosine phosphatases (PTPases)
06/02/2005US20050119256 Aromatic amino acid derivates and medicinal compositions
06/02/2005US20050119252 Ligands of melanocortin receptors and compositions and methods related thereto
06/02/2005US20050119250 Amino-derivatives as novel inhibitors of histone deacetylase
06/02/2005US20050119245 Alpha -, beta -, and gamma -amino acid derivatives, e.g., S)-2-{N'-[4-(4-Fluoro-phenoxy)-phenyl]-N''-cyano-guanidino}-3-phenyl-N-(3-pyrrolidin-1-yl-propyl)-propionamide for the treatment of central nervous system conditions such as muscle spasticity, tinnitus, epilepsy and neuropathic pain.
06/02/2005US20050119225 Phosphodiesterase 4 inhibitors, including N-substituted aniline and diphenylamine analogs
06/02/2005US20050119157 Organic compounds
06/02/2005US20050118619 Dark quenchers for fluorescence resonance energy transfer (FRET) in bioassays
06/02/2005DE10123573B4 N-Oxidanthranylamid-Derivate und deren Verwendung als Arzneimittel N-Oxidanthranylamid derivatives and their use as medicaments
06/02/2005CA2556801A1 Methods and agents for inhibiting dynamin-dependent endocytosis
06/02/2005CA2545048A1 Androgen receptor modulators
06/02/2005CA2543247A1 Benzannelated compounds as ppar activators
06/01/2005EP1535919A2 Synthesis and use of retinoid compounds having negative hormone and/or antagonist activities
06/01/2005EP1535909A2 Cyclic amine derivatives and their use as drugs
06/01/2005EP1534693A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
06/01/2005EP1534689A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
06/01/2005EP1534680A1 Prenylation inhibitors and methods of their synthesis and use
06/01/2005EP1534679A2 Inhibitors of post-amadori advanced glycation end products
06/01/2005EP1534671A2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
06/01/2005EP1534664A1 N-bisaryl- and n-aryl-cycloalkylidenyl-alpha-hydroxy-and alpha-alkoxy acid amides
06/01/2005EP1534658A2 Ketone ligands for modulating the expression of exogenous genes via an ecdysone receptor complex
06/01/2005EP1534276A2 Non-nucleoside reverse transcriptase inhibitors
06/01/2005EP1534273A2 Modulators of the glucocorticoid receptor and method
06/01/2005EP1351959B1 Novel pleuromutilin derivatives
06/01/2005EP1345902B1 Substituted heterocyclo-norbornylamine derivatives, method for producing the same, their use as medicament or diagnostic agent and medicament containing the same
06/01/2005EP1254136A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF
06/01/2005EP1115695B1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity
06/01/2005EP1114030B1 Pyridine ketones useful as herbicides
06/01/2005EP1109965B1 Method of treating a textile
06/01/2005EP1095015B1 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
06/01/2005EP0994862B1 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
06/01/2005EP0993441B1 INHIBITORS OF p38
06/01/2005EP0946499B1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
06/01/2005EP0708756B1 Substituted 2-phenylpyridines with herbicidal action
06/01/2005CN1622942A HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
06/01/2005CN1622832A Labeled macrophage scavenger receptor antagonists for imaging atherosclerosis and vulnerable plaque
06/01/2005CN1204138C Pyrazolo [4, 3-d] pyrimidine derivs.
06/01/2005CN1204137C Uracil compound and its appliance
06/01/2005CN1203852C Valdecoxib compositions
05/2005
05/31/2005US6900345 Antibiotics; mutilin 14-[N-(2-carbamoyloxyethoxycarbonyl)]carbamate; therapy for bacteria infections; chemical synthesis
05/31/2005US6900332 Converting alpha- isocyanoalkanoate esters in the presence of assistants at temperatures above 80 degrees C. into the 5-alkoxy-substituted oxazoles, and removing the reaction product from the reaction mixture
05/31/2005US6900330 Process for producing 2,3-pyridinedicarboxylic acid
05/31/2005US6900321 Substituted pyridyl amine complexes, and catalysts
05/31/2005US6900319 Carbo- and heterocyclic amidines
05/31/2005US6900244 Controlling lipid, cholesterol metabolism; anticholesterol agents
05/31/2005US6900237 Sulfonamide compounds as protease inhibitors
05/31/2005US6900232 For therapy of tumor metastasis, solid tumor growth (neoplasia), osteoporosis, Paget's disease, humoral hypercalcemia of malignancy, osteopenia, angiogenesis, including tumor angiogenesis and lymphangiogenesis
05/31/2005US6900231 Aminopyridyl-substituted phenyl acetamides as protease inhibitors
05/31/2005US6900218 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
05/31/2005US6900210 Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers
05/31/2005US6900202 Nicotinic acetylcholine receptor activators; treating neurodegenerative disorders
05/31/2005US6900180 Mixture of folic acid, vitamin b6 and b12 with carbohydrates, fats and proteins; infant formula; sleep disorders
05/31/2005US6899739 Hair dyes
05/26/2005WO2005047256A1 The derivatives of pyridone and the use of them
05/26/2005WO2005047255A1 Substituted nicotinoylcarbamates as pesticides
05/26/2005WO2005047254A1 Octahydrophenanthrene hydrazinde derivatives useful as glucocorticoid receptor modulators
05/26/2005WO2005047249A1 Benzylether amine compounds useful as ccr-5 antagonists
05/26/2005WO2005047233A1 Novel herbicides
05/26/2005WO2005047230A1 Bis-cationic compounds and use thereof
05/26/2005WO2005046683A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
05/26/2005WO2005046604A2 Heteroaryl-hydrazone compounds
05/26/2005WO2005046603A2 Pyridine compounds
05/26/2005WO2005046599A2 Alpha, beta-unsaturated sulfoxides for treating proliferative disorders
05/26/2005WO2004106363A3 A tag for purification of peptides
05/26/2005WO2003054145A3 Dinuclear copper-based compound and ligand for nucleic acid scission and anticancer treatment
05/26/2005US20050113595 C2-substituted idan-1-ols and their derivatives, processes for their preparation and their use as pharmaceuticals
05/26/2005US20050113580 2-(3-{3-[[2-chloro-3-(trifluoromethyl)benzyl](2,2-dephenylethyl)amino]propoxy}phenyl)-ethanol; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
05/26/2005US20050113578 Process for preparing substituted pyridines
05/26/2005US20050113450 method of sterilization, sanitation, antisepsis, and disinfection, includes applying antimicrobial compounds to a surface; e.g. 2-[(3-{[4-chloro(methyl)anilino]sulfonyl}benzoyl)amino]-5-(trifluoromethyl)benzoic acid
05/26/2005US20050113447 Selective retinoid agonists
05/26/2005US20050113440 Compounds that modulate PPAR activity and methods for their preparation
05/26/2005US20050113424 E.g., 4-{3-[4-(3-{4-[amino(imino)methyl]phenoxy}propyl)-1-piperazinyl]propoxy}benzamidine; an antifungal agent with good pharmacokinetics and excellent antifungal action; side effect reduction such as nephrotoxicity; action to Mycomycetes
05/26/2005US20050113416 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
05/26/2005US20050113396 Na+/H++exchanger-3 (NHE-3) inhibitors; antiischemic agents
05/26/2005US20050113373 medicine to inhibit proliferative conditions, such as cancer and psoriasis; detecting or identifying a histone deactylase (HDAC) in a biological sample
05/26/2005US20050113366 Derivatives of 4-hydroxybutanoic acid and of its higher homologue as ligands of $g(g)-hydroxybutyrate (ghb) receptors, pharmaceutical compositions containing same and pharmaceutical uses
05/26/2005US20050113346 making sulfur compounds such as 2-((4-But-2-ynyloxy-benzenesulfonyl)-methyl-amino)-N-hydroxy-3-methyl -butyramide, used as tumor necrosis factor-alpha converting enzyme (TACE) inhibitors, for prophylaxis of rheumatic diseases, sepsis or inflammation
05/26/2005US20050113344 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
05/26/2005US20050112407 Organic electroluminescent device
05/26/2005CA2545259A1 Heteroaryl-hydrazone compounds
05/26/2005CA2545258A1 Pyridine compounds
05/26/2005CA2545020A1 Octahydrophenanthrene hydrazinde derivatives useful as glucocorticoid receptor modulators
05/26/2005CA2543913A1 Benzylether amine compounds useful as ccr-5 antagonists
05/26/2005CA2541949A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
05/25/2005EP1533303A1 Substituted Aminosalicylacid Amides ( intermediates )
05/25/2005EP1533294A1 Beta-alanine derivative and use thereof
05/25/2005EP1533292A1 Dibenzylamine compound and medicinal use thereof
05/25/2005EP1532310A1 Method for delivering biologically active substances
05/25/2005EP1532209A2 Charge transport compositions and electronic devices made with such compositions
05/25/2005EP1532158A1 Neutral metallic dendrimer complexes
05/25/2005EP1532112A1 Process for the preparation of modification i of n-(1-methylethylaminocarbonyl)-4-(3-methylphenylamino)-3-pyridinesulfonamide
05/25/2005EP1532111A1 2,5-disubstituted 3-mercaptopentanoic acid