Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273) |
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12/22/2005 | WO2005121073A1 Inhibitors of histone deacetylase |
12/22/2005 | WO2005121069A1 Levodopa prodrugs, and compositions and uses thereof |
12/22/2005 | WO2005120515A2 Novel sulfonamides as inhibitors of histone deacetylase for the treatment of disease |
12/22/2005 | WO2005120477A2 N- (2-benzyl) -2-phenylbutanamides as androgen receptor modulators |
12/22/2005 | WO2005103041A9 Treatment of cns disorders using cns target modulators |
12/22/2005 | WO2005061443A3 Benzoyl-substituted phenylalanine amides |
12/22/2005 | WO2004106296A3 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators |
12/22/2005 | US20050282908 Substituted aminopropoxyaryl derivatives useful as agonists for LXR |
12/22/2005 | US20050282905 Hydroxamic acid derivative and mmp inhibitor containing the same as active ingredient |
12/22/2005 | US20050282891 Parkinson's disease, depression, attention deficit disorder; schizophrenia, manic depression, cognitive impairment disorders, restless legs syndrome, periodic limb movement disorders, Huntington's disease, Tourette's syndrome, congestive heart failure, sustained release |
12/22/2005 | US20050282882 Diamines as modulators of chemokine receptor activity |
12/22/2005 | US20050282881 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
12/22/2005 | US20050282872 Novel thyroid receptor ligands and method II |
12/22/2005 | US20050282871 3-(3,5-Disubstituted-4-hydroxyphenyl)propionamide derivatives as cathepsin b inhibitors |
12/22/2005 | US20050282869 Use of a compound in the treatment of sleep disorders and the like, in providing refreshedness on waking and a method for the treatment of grogginess therewith |
12/22/2005 | US20050282862 Aromatic amides |
12/22/2005 | US20050282858 Substituted cycloalkylcarboxamides: 1-((1-(4-Chlorophenyl)cyclopropyl)carbonyl)pyrrolidin-3-ol and 1-Acetyl-4-(4-{1-[(3-phenylpyrrolidin-1-yl)carbonyl]cyclopropyl}phenyl)piperazine; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; antidiabetic agents |
12/22/2005 | US20050282846 Compounds capable of activating cholinergic receptors |
12/22/2005 | US20050282817 4-(3-Phenyl-3-carbocycloylpropyl)-1-phenyl- or pyridylpiperazine derivatives: 1-(2-methoxyphenyl)-4-[3-(benzoyl)-3-(phenyl)propyl]piperazine oxalate; serotonin receptor antagonists; obesity |
12/22/2005 | US20050282809 Heteroaryl-hydrazone compounds |
12/22/2005 | US20050282787 Synthesis of tetracyclines and analogues thereof |
12/22/2005 | US20050282707 Pyridinylisoxazoles and their use as herbicides |
12/22/2005 | CA2569883A1 Aroyl-o-piperidine derivatives for the treatment of diabetes-related problems |
12/22/2005 | CA2568632A1 Levodopa prodrugs, and compositions and uses thereof |
12/22/2005 | CA2567835A1 Novel sulfonamides as inhibitors of histone deacetylase for the treatment of disease |
12/22/2005 | CA2564499A1 Tetrahydropyranyl cyclopentyl tetrahy-dropyridopyridine modulators of chemokine receptor activity |
12/21/2005 | EP1607388A1 An improved manufacturing process for methylphenidate and intermediates thereof |
12/21/2005 | EP1606261A1 Novel process for the preparation of roflumilast |
12/21/2005 | EP1606260A1 Oxamide derivatives useful as raf-kinase inhibitors |
12/21/2005 | EP1606237A1 2-(butyl-1-sulfonylamino)-n- 1(r)-(6-methoxy-pyridin-3-yl)-propyl]-benzamid, the use thereof in the form of drug an pharmaceutical preparations containing said compound |
12/21/2005 | EP1362039B1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands |
12/21/2005 | EP0579819B1 Novel pyridone derivative having an affinity for the angiotensine ii receptor |
12/21/2005 | CN1711257A Aryl sulfonamides |
12/21/2005 | CN1711252A 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders |
12/21/2005 | CN1711245A Process for the preparation of 2-aminomethylpyridine derivative |
12/21/2005 | CN1711244A Novel process for the preparation of 2-aminomethylpyridine derivative |
12/21/2005 | CN1711239A Novel biaromatic compounds which activate PPARy type receptors and cosmetic/pharmaceutical compositions comprised thereof |
12/20/2005 | US6977266 Pyridone derivatives having affinity for cannabinoid 2-type receptor |
12/20/2005 | CA2302412C Aminoalkylphenol derivatives and related compounds |
12/20/2005 | CA2181569C Ep2-receptor agonists as agents for lowering intraocular pressure |
12/20/2005 | CA2174127C Phenylsulfonyl ureas, processes for their preparation, and their use as herbicides and plant growth regulators |
12/15/2005 | WO2005118606A1 Fluorine-substituted iridium complex and luminescent material made with the same |
12/15/2005 | WO2005118545A1 Gas-phase oxidation of alkyl-substituted heterocyclic compounds |
12/15/2005 | WO2005118544A2 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/15/2005 | WO2005118543A1 Kinase inhibitor and use thereof |
12/15/2005 | WO2005118542A1 Glucagon receptor antagonists, preparation and therapeutic uses |
12/15/2005 | WO2005118541A2 Heterocyclic compounds and their use as aldosterone synthase inhibitors |
12/15/2005 | WO2005117904A2 Phosphonate analogs of hiv integrase inhibitor compounds |
12/15/2005 | WO2005117883A1 Modulators of muscarinic receptors |
12/15/2005 | WO2005117867A2 Monocyclic heterocycles as kinase inhibitors |
12/15/2005 | US20050277681 N-(2-benzyl)-2-phenylbutanamides as androgen receptor modulators |
12/15/2005 | US20050277680 tyrphostin-like compounds that display a significant potency as kinase inhibitors, cause the downregulation of c-myc proto-oncogene and inhibit the growth and survival of cancerous cell lines; antiproliferative agents |
12/15/2005 | US20050277678 5-(4-Fluorophenyl)-1-(4-methylsulfoximinylphenyl)-3-trifluoromethyl-1H-pyrazole; prostaglandin and cyclooxygenase inhibitor; antiinflammatory, analgesic, and antipyretic agent |
12/15/2005 | US20050277667 Manufacturing process for methyl phenidate and intermediates thereof |
12/15/2005 | US20050277663 3-Aryl-3-hydroxy-and 3-aryl-3-oxopropionic acid esters as fungicides |
12/15/2005 | US20050277662 such as: 1-(2, 4-difluorobenzyl) -N-hydroxy-3-(morpholin-4-ylmethyl)-1H-pyrrolo[2,3-c]pyridine-5-carboxamide; acquired immunodeficiency syndrome ("AIDS"), and AIDS related complex ("ARC") |
12/15/2005 | US20050277652 Hepatocyte growth factor receptor inhibitors; Antitumor agents, anticarcinogenic agents, angiogenesis inhibitors; pyrimidine derivatives like Pyrrolidine-1-carboxylic acid [6-(2-fluoro-4-{3-[2-(4-fluorophenyl)acetyl]thioureido}phenoxy)pyrimidin-4-yl]amide |
12/15/2005 | US20050277649 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors; potentiation; diabetes and obesity; 2-(4-{4-[1-(6-chloro-pyridin-3-yl)cyclopropylmethyl]-2-(R)-methyl-piperazine-1-sulfonyl}phenyl)-1,1,1-trifluoro-propan-2-ol |
12/15/2005 | US20050277646 N-[4-({5-(4-fluorophenyl)-4-[4-(trifluoromethyl)phenyl]pyridin-2-yl}oxy)-1,3-benzothiazol-2-yl]acetamide; vanilloid (capsaicin) receptor antagonist/agonist; antiinflammatory, analgesic, antiarthritis, antirheumatic; diseases involving sensory nerve function |
12/15/2005 | US20050277631 Vanilloid receptor ligands and their use in treatments |
12/15/2005 | DE4332964B4 Verfahren zur Herstellung von aromatischen Polyetherketonen A process for the preparation of aromatic polyetherketones |
12/15/2005 | DE102004024565A1 Verfahren zur Herstellung von α-Chloralkylpyridylketonen und/oder deren Hydrochloriden A process for preparing α-Chloralkylpyridylketonen and / or their hydrochlorides |
12/15/2005 | CA2568524A1 Modulators of muscarinic receptors |
12/15/2005 | CA2568164A1 Heterocyclic compounds and their use as aldosterone synthase inhibitors |
12/15/2005 | CA2566531A1 Cycloalkyl substituted pyrimidinediamine compounds and their uses |
12/15/2005 | CA2563831A1 Monocyclic heterocycles as kinase inhibitors |
12/15/2005 | CA2562713A1 Phosphonate analogs of hiv integrase inhibitor compounds |
12/14/2005 | EP1603923A1 Metal complexes |
12/14/2005 | EP1603879A2 Substituted pyridine derivatives useful in the treatment of cancer and other disorders |
12/14/2005 | EP1603878A1 Processes for the preparation of n-heteroaryl-n-aryl-amines by reacting an n-aryl carbamic acid ester with a halo-heteroaryl and analogous processes |
12/14/2005 | EP1603877A1 NOVEL AMINOPYRIDINE DERIVATIVES AS mGIuR5 ANTAGONISTS |
12/14/2005 | EP1603876A1 Process for the preparation of pyridinyl and pyrimidinyl mono-fluorinated beta keto esters |
12/14/2005 | EP1603858A2 Kcnq channel modulating compounds and their pharmaceutical use |
12/14/2005 | EP1603572A1 Lactam-containing cyclic diamines and derivatives as factor xa inhibitors |
12/14/2005 | EP1603570A2 Aminoheteroaryl compounds as protein kinase inhibitors |
12/14/2005 | EP1603562A2 Sulfonyl-amidino containing and tetrahydropyrimidino containing compounds as factor xa inhibitors |
12/14/2005 | EP1326858B1 Piperidine compounds as anti-allergic |
12/14/2005 | EP1263712B1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds |
12/14/2005 | EP1224165B1 Novel compounds |
12/14/2005 | EP1200411B1 Process for synthesis of heteroaryl-substituted urea compounds |
12/14/2005 | CN1708482A N-sulfonyl-4-methyleneamino-3-hydroxy-2-pyridones as antimicrobials |
12/14/2005 | CN1708481A N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones as antimicrobials |
12/14/2005 | CN1708478A P-(sulfonyl)-aryl and heteroaryls amines |
12/14/2005 | CN1708476A Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds |
12/14/2005 | CN1231476C Substd. pyridine herbicides |
12/14/2005 | CN1231465C Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament |
12/14/2005 | CN1231464C Novel 3-substituted urea derivatives and medicinal use thereof |
12/14/2005 | CN1231440C Novel tricyclic compound |
12/14/2005 | CN1231431C Process for preparing substituted 2-3-dihydro-1-indanones |
12/14/2005 | CN1231212C Multicyclic compounds which inhibit beukocyte adhesion mediated by VLA-4 |
12/13/2005 | US6974876 Method for preparing intermediates useful in synthesis of retroviral protease inhibitors |
12/13/2005 | US6974836 Diamines as modulators of chemokine receptor activity |
12/13/2005 | US6974830 For therapy of atherosclerosis, gallstone disease, lipid disorders, obesity or a cardiovascular disorder |
12/13/2005 | US6974828 3-((2-((3-((Amino(imino)methyl)amino)benzoyl)amino)phenyl)sulf anyl)- 3-(3-pyridinyl)propanoic acid, for example; angiogenic inhibitors; antitumor, -carcinogenic, -metastatic, -diabetic, -arthritic and inflammatory agents; bone disorders |
12/13/2005 | US6974817 CCR1 receptor antagonists; inhibitors of MIP-1 alpha (CCL3) binding to its receptor CCR1 found on inflammatory and immunomodulatory cells; macrophage inflammatory protein (MIP) |
12/13/2005 | US6974802 Treatment of viral infections using prodrugs of 2′,3-dideoxy,3′-fluoroguanosine |
12/13/2005 | US6974567 Labeled macrophage scavenger receptor antagonists for imaging atherosclerosis and vulnerable plaque |
12/08/2005 | WO2005116198A2 Methods of 1,3-enyne preparation using copper (i) catalysts |
12/08/2005 | WO2005116010A1 Ep4 receptor agonist, compositions and methods thereof |
12/08/2005 | WO2005115992A1 Theramutein modulators |