Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
04/2008
04/10/2008US20080085893 N-Hydroxy (2S)-2-hydroxy phenyl or heteroaryl sulfonamide derivatives; for example, N-Hydroxy (2S)-2-hydroxy-3-{N-[4-(4- chlorophenoxy)phenyl], N- methanesulfonylamino}propionamide; for treating disorders related to matrix metalloproteases, particularly useful for treating strokes;
04/10/2008US20080085891 Asthma and allergic inflammation modulators
04/10/2008US20080085884 Eating disorders, psychological disorders, sexual disorders, nervous system disorders, sleep disorders, autism; 4-(Benzyloxy)-6'-[3-methyl-3-(methylamino)pyrrolidin-1-yl]-2H-1,3'-bipyridin-2-one for example
04/10/2008CA2665428A1 Hdac inhibitors
04/10/2008CA2664119A1 3-pyridinecarboxamide and 2-pyrazinecarboxamide derivatives as hdl-cholesterol raising agents
04/09/2008EP1908751A1 N-hydroxy benzamides with antitumour activity
04/09/2008EP1907387A1 An oxime derivative and preparations thereof
04/09/2008EP1907382A1 Nitrocatechol derivatives as comt inhibitors
04/09/2008EP1907372A1 Substituted cyclohexyl derivatives as nk-3 receptor antagonists
04/09/2008EP1907363A1 Phenyl substituted piperazine-derivatives as inhibitors of plaminogenic activator inhibitors-i (pai-i)
04/09/2008EP1907362A1 Amide derivatives as kinase inhibitors
04/09/2008EP1907361A1 Amide derivatives as kinase inhibitors
04/09/2008EP1907360A1 Improved process for the manufacture of flecainide
04/09/2008EP1907120A1 Catalyst with bimodal distribution of the particles of the catalytically active material, method for the production thereof and for the regeneration thereof and the use of the catalyst
04/09/2008EP1594867B1 Phenylacetamides and their use as glucokinase modulators
04/09/2008EP1572651A4 Compounds useful as pesticides
04/09/2008EP1309565B1 Heterocyclic mutilin esters and their use as antibacterials
04/09/2008EP0958287B2 Sulfamide-metalloprotease inhibitors
04/09/2008CN101160288A Method for producing nicotinic acid derivative or its salt
04/09/2008CN101160287A 吡啶基非芳香族含氮杂环-1-羧酸酯衍生物 Pyridyl non-aromatic nitrogen-containing heterocyclic-1-carboxylate derivative
04/09/2008CN101160285A Substituted sulfonylaminoarylmethyl cyclopropanecarboxamide as vr1 receptor antagonists
04/09/2008CN101157654A Preparation method of 2-chlorin-3-amido-4-methyl pyridine
04/09/2008CN101157653A Method for preparing 2,6-diacetyl pyridine
04/09/2008CN101157652A Antitumor activity bipyridine methyl amine compound and preparation method thereof
04/09/2008CN100379725C Immunoassay detection method for neonicotinyl insecticides
04/09/2008CN100379416C Stable solid medicinal composition for oral administration.
04/08/2008US7355049 Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
04/08/2008US7355048 Process for preparing 1-(6-methylpyridin-3-yl)-2-[4- (methylsulphonyl)phenyl]ethanone
04/08/2008US7355042 Sleep disorders; side effect reduction
04/08/2008US7354946 Biarylurea derivatives
04/08/2008US7354943 Statine derivatives for the treatment of Alzheimer's disease
04/08/2008US7354942 Benzylether and benzylamino beta-secretase inhibitors for the treatment of Alzheimer's disease
04/08/2008US7354940 2,5-dioxoimidazolidin-4-yl acetamines and analogues as inhibitors of metalloproteinase mmp12
04/08/2008US7354895 Phosphinyloxy, oxime and carboxylic acid derivatives which are useful as carboxypeptidase U inhibitors
04/03/2008WO2008039645A1 Compounds which modulate the cb2 receptor
04/03/2008WO2008038955A1 Benzophenone derivatives useful for inhibiting formation of microtubule
04/03/2008WO2008037604A1 Novel polybenzofulvene derivatives, synthesis and uses thereof
04/03/2008WO2008014199A3 Sulfonyl compounds which modulate the cb2 receptor
04/03/2008US20080081926 Sulfonylaminobenzoic acid and salt
04/03/2008US20080081912 Near-infrared absorptive image-forming composition, ink and electrophotographic toner using the same, and inkjet-recording method, electrophotographic-recording method and near-infrared-ray-reading method using those
04/03/2008US20080081825 5-((2,4-difluorophenyl) {[(1-methyl-4-piperidinyl)oxy]imino}methyl)-1-(2,6-dimethylphenyl)-2(1H)-pyridinone; p38 MAP kinase and tumor necrosis factor inhibitor; inflammatory cytokines or chemokine, respiratory diseases, cardiovascular diseases and bone diseases
04/03/2008US20080081822 N-(5-tert-Butyl-isoxazol-3-yl)-2-cyclohexanesulfonyl-2-methyl-propionamide; cannabinoid receptor agonist, antagonist; analgesic, antiinflammatory and antitumor agent; neuropatic pain
04/03/2008US20080081812 and inverse agonist; 2-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazol-3-yl)-5-(pyridin-4-yl)-1,3,4-oxadiazole; obesity and obesity-related metabolic disorders
04/03/2008CA2664310A1 Compounds which modulate the cb2 receptor
04/02/2008EP1905761A1 An improved process for the preparation of 4-[2-(methyl-2-pyridinylamino) ethoxy] benzaldehyde, an intermediate for the preparation of rosiglitazone
04/02/2008EP1905438A2 Hypoglycemic agent
04/02/2008EP1904537A1 Polymerisation catalyst system based on dioxime ligands
04/02/2008EP1904471A1 Heteroarylethenyl derivatives, their manufacture and use as pharmaceutical agents
04/02/2008EP1904439A2 Sphingosine kinase inhibitors
04/02/2008EP1765771A4 Formation of tetra-substituted enamides and stereoselective reduction thereof
04/02/2008EP1201648B1 Carbamate derivatives and agricultural/horticultural bactericides
04/02/2008CN101155782A Potentiator for radiation therapy comprising pyridine derivative as active ingredient
04/02/2008CN101155781A Pyridine-3-carboxamide derivatives as cb1 inverse agonists
04/02/2008CN100378100C Pyrazolo(4,3-d)pyrimidine derivatives
04/02/2008CN100378076C Pyridine carboxamide derivatives and their use as pesticides
04/02/2008CN100378075C Aniline derivative using as phosphodiesterase 4 inhibitor
04/02/2008CN100378072C Heterocyclic methyl sulfone derivative
04/02/2008CN100378063C Novel compounds and medicinal use thereof
04/02/2008CN100378059C Diastereoselective method of preparing olefins by means of the Horner-Wadsworth-Emmons reaction, comprising the addition of a tris-(polyoxaalkyl)-amine sequestering agent
04/01/2008US7351865 Synthesis of sterically hindered secondary aminoether alcohols from acid anhydride and/or acid halide and sulfur trioxide
04/01/2008US7351861 Halo-substituted N-arylanilides with one or more hydroxy groups that may be esterified; N-benzilideneiminoarylamides; antibacterial agents
04/01/2008US7351835 Organic molecular cataylst having binaphthol skeleton and processes for producing the same and application thereof
04/01/2008US7351834 Sorafenib and salts such as tosylate (N-(4-chloro-3-(trifluoromethyl)phenyl)-N'-(4-(2-(N-methylcarbamoyl)-4-pyridyloxy)phenyl)urea); serine-threonine kinase inhibitor; antitumor and anticarcinogenic agent
04/01/2008US7351826 Aryl acid pyrimidinyl methyl amides, pyridazinyl methyl amides and related compounds
04/01/2008US7351825 4-[5-((1S,2R)-1-Carboxy-2-phenyl-cyclopropylsulfamoyl)-thiophen-2-yl]-3,6-dihydro-2H-pyridine-1-carboxylic acid tert-butyl ester; aggrecanase and matrix metalloproteinase (with zinc in the catalytic active center) (MMP) inhibitor; antiarthritic agent: osteoarthritis, rheumatoid arthritis
04/01/2008US7351822 Serine protease inhibitors
04/01/2008US7351738 e.g., phenyl ((1S,2R)-1-(3,5-difluorobenzyl)-3-{[(1S)-7-ethyl-1,2,3,4-tetrahydronaphthalen-1-yl]amino}-2-hydroxypropyl)carbamate; inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide
04/01/2008US7351733 Tetrahydrocarbazole derivatives and their pharmaceutical use
04/01/2008US7351721 Amino acid derivatives and pharmaceutical composition comprising, as active ingredients, them
04/01/2008US7351719 Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds
04/01/2008US7351703 Which modulate the endogenous production of cyclic guanosine monophosphate (cGMP); for therapy and prophylaxis of cardiovascular disorders such as high blood pressure, angina pectoris, cardiac insufficency, thromboses, and/or atherosclerosis
04/01/2008CA2332713C Hydroxamic acid derivatives as antibacterials
03/2008
03/27/2008WO2008034886A1 Pyridine borane complexes
03/27/2008WO2008034272A1 Stilbazolium salt
03/27/2008WO2008008660A3 Cyclopentane derivatives as antiglaucoma agents
03/27/2008WO2008008431A3 Heteroaryl sulfonamides and ccr2/ccr9
03/27/2008WO2007141200A8 Novel n-aryl and n-heteroaryl substituted pyridinone derivatives for use in mch-1 mediated diseases
03/27/2008WO2007136573A3 Antidiabetic bicyclic compounds
03/27/2008WO2007134038A3 Salt forms of (2s)-(4e)-n-methyl-5-[3-(5-isopropoxypyridin)yl]-4-penten-2-amine
03/27/2008WO2007132179A3 Therapeutics comprising pyridinium derivatives
03/27/2008US20080076930 Novel stereoselective synthesis of benzimidazole sulfoxides
03/27/2008US20080076805 Antagonists and/or inverse agonists of CB1; N'-[1-(3-chlorophenyl)-2-(4-chlorophenyl)ethyl]-N'-methyl-N-(2-methyl-2-[5-(trifluoromethylpyridin-2-yl)oxy]propanoyl)hydrazide for example; obesity, psychological disorders, analgesics, drug abuse, constipation, asthma, cirrhosis
03/27/2008US20080076801 Indolylalkylpyridin-2-amines for the inhibition of beta-secretase
03/27/2008US20080076800 Anticancer, inflammation, arthritis, angiogenesis, neurodegenerative diseases, fungal infections, malaria; Heat-shock protein 90 inhibitors; 4-(6,6-Dimethyl-4-oxo-3-methyl-4,5,6,7-tetrahydro-indazol-1-yl)-2-(3,4,5-trimethoxyanilino)-benzamide
03/27/2008US20080076794 Hyperaldosteronism
03/27/2008US20080076738 antiviral: improved pharmacokinetics
03/27/2008DE102006043520A1 2-Phenoxynikotinsäure-Derivate und ihre Verwendung 2-Phenoxynikotinsäure derivatives and their use
03/27/2008DE102006043519A1 4-Phenoxynikotinsäure-Derivate und ihre Verwendung 4-Phenoxynikotinsäure derivatives and their use
03/27/2008CA2663901A1 Pyridine derivatives for the treatment of metabolic disorders related to insulin resistance or hyperglycemia
03/27/2008CA2663677A1 Pyridine borane complexes
03/26/2008EP1903030A1 Method for catalytic manufacture of aromatic or heteroaromatic nitriles
03/26/2008EP1903023A1 Method for manufacturing arylamines
03/26/2008EP1902714A1 Prodrugs of gaba analogs, compositions and uses thereof
03/26/2008EP1902074A1 Single site catalyst systems having a scorpion-like structure
03/26/2008EP1902028A2 Histamine h3 receptor antagonists
03/26/2008EP1902022A1 Piperazine heteroaryl derivates as gpr38 agonists
03/26/2008EP1902017A1 Antiviral compounds and methods
03/26/2008EP1902004A2 Onium-alkylsulfonate production method
03/26/2008EP1556342B1 Phenethanolamine derivative for the treatment of respiratory diseases
03/26/2008EP1509218A4 Peptide deformylase inhibitors