Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
10/2008
10/15/2008EP1979322A1 Cyclohexyl sulfonamide derivatives having h3 receptor activity
10/15/2008EP1979321A1 Novel pyridinylaminoalkylene- and pyridinyloxyalkylene-cyclopropanamines, process for the preparation thereof and pharmaceutical compositions containing them
10/15/2008EP1979320A2 PIPERAZINES AND PIPERIDINES AS mGluR5 POTENTIATORS
10/15/2008EP1979311A2 Phenoxy acetic acids as ppar delta activators
10/15/2008EP1896416B1 Substituted heterocycles, their use as medicament, and pharmaceutical preparations comprising them
10/15/2008EP1781297B1 Novel biaromatic compounds that activate ppar type receptors, and use thereof in cosmetic or pharmaceutical compositions
10/15/2008EP1742642B1 Phosphonate analogs of hiv integrase inhibitor compounds
10/15/2008EP1532158B1 Neutral metallic dendrimer complexes
10/15/2008EP1476423B1 Arylsulfonamidobenzylic compounds
10/15/2008EP1385912B1 Pyridone dyes, a process for their preparation and their use in the production of coloured plastics or polymeric colour particles
10/15/2008EP1373257B9 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
10/15/2008EP1308436B1 Calcium receptor antagonists
10/15/2008CN101287718A Substituted heteroaryl- and phenylsulfamoyl compounds
10/15/2008CN101287708A Pyridinaminosulfonyl substituted benzamides as inhibitors of cytochrome p450 3a4 (cyp3a4)
10/15/2008CN101287707A 激酶抑制剂 Kinase inhibitors
10/15/2008CN101287702A N-phenyl phenylacetamide non-nucleoside reverse transcriptase inhibitors
10/15/2008CN101284865A New compound and its medicine use
10/15/2008CN101284779A Preparation method of (E)-4-(beta-bromovinyl)phenol ester
10/15/2008CN101284247A Dinuclear nickel cross-coupling reaction catalyst supported by nitrogen heterocycle carbine ligand and preparation method thereof
10/15/2008CN100425609C N-heteroarylnicotinamide derivatives
10/15/2008CN100425607C Method for controlling particular insects by applying anthranilamide compounds
10/14/2008US7435844 Fungicides; 2-methoxyacrylic acid esters or amides, 2-substituted with o-(phenoxymethyl)phenyl- groups, e.g., methyl (E)-2-{2-[3,5-dichloro-4-(3,3-dimethylbutoxy)phenoxymethyl]phenyl}-3-methoxyacrylate; agriculture, horticulture, animal husbandry
10/14/2008US7435843 Thiobenzoic acid, N-malonylhydrazide in which the free carboxy group is protected; enhances the desirable tumor attacking properties of anticancer agents without further increasing undesirable side-effects
10/14/2008US7435823 2,3-Dihydro-4H-1,4-benzoxazine derivatives containing an optionally fused pyridine or pyrimidine ring; 7-((6,7-bis(methyloxy)-4-quinolinyl)oxy)-N-phenyl-2,3-dihydro-4H-1,4-benzoxazine-4-carboxamide; kinase inhibitors; inflammation, angiogenesis and cancer
10/14/2008US7435815 Sulfonylamino-acetic acid derivatives
10/14/2008US7435743 I kappa B kinase beta inhibitors that are 2-amino-4,6-disubstituted nicotinic acid ester analogs; antiinflammatory, antitumor and antiischemic effects; asthma; nuclear factor kappa B inhibitors; 7-(2-hydroxyphenyl)-5-(3-piperidinyl)-1,4-dihydro-2H-pyrido[2,3-d][1,3]oxazin-2-one
10/14/2008CA2333089C Processes and intermediates for preparing 2-substituted piperidine stereoisomers
10/14/2008CA2309328C Cyclic amine derivatives and their use as drugs
10/09/2008WO2008120810A1 Compound, photoelectric converter and photoelectrochemical cell
10/09/2008WO2008120759A1 Urea compound and use thereof
10/09/2008WO2008120754A1 Picolinamide compound
10/09/2008WO2008120235A1 Novel benzophenone hybrids as potential anticancer agents and a process for the preparation thereof
10/09/2008WO2008119773A1 Amide derivatives as inhibitors of aspartyl proteases
10/09/2008WO2008101682A3 Iminipyridine derivatives and their uses as microbiocides
10/09/2008WO2008062276A8 Acetylene derivatives as stearoyl coa desaturase inhibitors
10/09/2008WO2008024304A3 Compounds for treatment of proliferative disorders
10/09/2008WO2007124424A3 Il-8 receptor antagonists
10/09/2008WO2007107706A3 Dimers of heterocyclic compounds for the treatment of copd
10/09/2008US20080249314 Using isopropanol solvent and dibenzolytartaric acid; forming salt; reacting with a base
10/09/2008US20080249313 Heating mixture of trichloromethylpyridine with sulfuric acid in liquid phase
10/09/2008US20080249306 Method for the Production of Statins
10/09/2008US20080249166 Inhibiting hepatic fatty acid and sterol synthesis; use with statins; compounds such as cyclopropyl or cyclobutyl-functional hydroxy-functional alpha,gamma-alkanediacids
10/09/2008US20080249140 Quaternary 3 -Amido, N-Methylpyridinium Salts as Anti-Inflammatory Agents
10/09/2008US20080249139 N-((1S,2R)-1-(3,5-difluorobenzyl)-3-{[(1S)-7-ethyl-1,2,3,4-tetrahydronaphthalen-1-yl]amino}-2-hydroxypropyl)pyrazine-2-carboxamide for example; or corresponding sulfonamides; beta-secretase inhibitors; dementia; Alzheimer's disease
10/09/2008US20080249138 Pyridine Compounds For The Treatment Of Prostaglandin Mediated Diseases
10/09/2008US20080249137 e.g. {3-butoxy-5-[4-(4-trifluoromethoxy-phenoxy)-benzenesulfonyl]-phenyl}-acetic acid; peroxisome proliferator activated receptor modulator; antidiabetic agent; obesity, hyperlipidemia, dyslipidemia, hypertriglyceridemia, Syndrome X, insulin resistance, diabetic neuropathy, atherosclerosis, eczema
10/09/2008US20080249102 Hiv Protease Inhibitors
10/09/2008US20080249093 immunosuppressive, anti-inflammatory and hemostatic agents to modulate leukocyte trafficking, sequestering lymphocytes in secondary lymphoid tissues, and enhancing vascular integrity; safer and more effective; 3-(4-(5-(3-Cyano-4-isopropyloxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid
10/09/2008US20080249071 inhibitory activity against the activation of inflammatory cytokines such as interleukin (IL)-1, IL-6, IL-8 and tumor necrosis factor (TNF- alpha ), NF- kappa K B; inflammatory disorders, autoimmune diseases; side effects reduction; immuno suressants; N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxybenzamide
10/09/2008US20080248329 Light sources comprising organic light emmiters between electrodes, used in displaying, electrophotography, recording, exposure, signs or optical communications; brightness; efficiency; durability; iridium complex
10/09/2008US20080246002 Polar liquid crystal
10/09/2008CA2682384A1 Benzophenone hybrids as potential anticancer agents and a process for the preparation thereof
10/08/2008EP1977749A1 Use of cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia
10/08/2008EP1976840A1 Cyclohexyl piperazinyl methanone derivatives and their use as histamine h3 receptor modulators
10/08/2008EP1654233A4 Method for the manufacture of cyanopyridines and catalysts suitable therefor
10/08/2008EP1539693B9 Cannabinoid receptor agonists
10/08/2008EP1341785B1 Hydrolysis of r(r*,r*)-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4- [(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid esters with calcium hydroxide
10/08/2008EP1335902B1 Heteroarylacryloylaminoalkyl-substituted benzenesulfonamide derivatives, their preparation, their use and pharmaceutical preparations comprising them
10/08/2008CN101282953A Therapeutic agents
10/08/2008CN101282937A Therapeutic agents
10/08/2008CN101282934A Triarylcarboxylic acid derivative
10/08/2008CN101282933A Novel NK1 and NK2 antagonists
10/08/2008CN101282786A Catalyst with bimodal distribution of the particles of the catalytically active material, method for the production thereof and for the regeneration thereof and the use of the catalyst
10/08/2008CN101279969A Organic electroluminescent material and application thereof
10/08/2008CN101279927A Arylene-carboxylic acid (2-amino-phenyl)-amide derivatives as pharmaceutical agents
10/08/2008CN100424083C Pyrimidine derivative compound and its preparing method
10/08/2008CN100423721C Thrombopoietin mimetics
10/07/2008US7432392 Ester derivatives and medical use thereof
10/07/2008US7432378 For example, 2-{2-Chloro-4-[3-(4-methyl-piperazin-1-yl)-propoxy]-phenyl}-4,5-dimethyl-1H-benzoimidazole; use in leukocyte recruitment inhibition, in modulating H4 receptor, and in treating conditions such as inflammation, H4 receptor-mediated conditions, and related conditions
10/07/2008US7432370 Mixing a racemic mixture of enantiomers of pyrrolo[2,3-d]pyrimidine compounds in a solvent, with a resolving compound having a defined stereospecificity, to form a solution and with resolving agent being capable of binding with enantiomers to form a precipitate collecting precipitate and purifying
10/07/2008US7432303 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states
10/07/2008US7432289 5-Acylamino-1,1′-biphenyl-4-carboxamide derivatives and their use as P38 kinase inhibitors
10/07/2008US7432287 e.g. 3-(6-ethanesulfonylpyridin-3-yloxy)-5-(2-hydroxy-1-methyl-ethoxy)-N-(1-methyl-1H-pyrazol-3-yl)benzamide; glucokinase activator; antidiabetic agent; obesity, insulin resistance
10/07/2008US7432286 Pharmaceutically active sulfonyl hydrazide derivatives
10/07/2008US7432281 4-(2,2-dichloro)-N-(quinolin-3-yl)benzamide; (1R,2R)2-methyl-N-(quinolin-3-yl)-4-(2-(trifluoromethyl)cyclopropyl)benzamide; inflammation-related conditions in mammals, arthritis, Parkinson's/Alzheimer's diseases, stroke, asthma; acute/chronic or neuropathic pain; VR1 agonist/antagonist
10/07/2008US7432268 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
10/07/2008US7432264 Antibacterial compounds such as (S)-2-cyano-1-(trans-4-(5-nitro-2-pyridylamino)cyclohexylamino )acetylpyrrolidine; activity against Gram-negative and Gram-positive pathogens, including a methicillin-resistant S. aureus strain
10/07/2008US7432228 Applying a N-aryl(methyl)-p-hydroxy- or p-alkoxy--phenylalkylamine, e.g., 4-[2-(2-hydroxy-benzylamino)-ethyl]-phenol to inhibit 9-cis-epoxycarotenoid dioxygenase; plant growth regulators
10/07/2008US7432227 6-alkyl or alkenyl-4-aminopicolinates and their use as herbicides
10/07/2008CA2362831C Thioamide derivatives
10/02/2008WO2008119015A2 Synthesis of thiohydantoins
10/02/2008WO2008117862A1 Novel (2-aminophenyl)pyridinecarboxamide derivative having urea structure
10/02/2008WO2008117861A1 Intraocular pressure lowering agents containing phenylenediamine derivatives as the active ingredient
10/02/2008WO2008116663A2 Heterocyclyl-substituted-tetrahydro-naphthalen-amine derivatives, their preparation and use as medicaments
10/02/2008WO2008116301A1 Fluorinated derivatives of deferiprone
10/02/2008WO2008093024A3 N-(amino-heteroaryl)-1h-pyrrolopyridine-2-carboxamides derivatives, preparation thereof and their use in therapy
10/02/2008WO2008084223A3 Chemical compounds 637: pyridopyrimidinediones as pde4 inhibitors
10/02/2008WO2008082500A3 Process for the synthesis of 2,6-diaminopyridines from glutarimidines
10/02/2008WO2008075172A3 Nicotinamide derivatives as inhibitors of h-pgds and their use for treating prostaglandin d2 mediated diseases
10/02/2008WO2008053194A3 Pyridine carboxamides as 11-beta-hsd1 inhibitors
10/02/2008WO2007149163A3 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors
10/02/2008WO2007082098A8 6-(poly-substituted aryl)-4-aminopicolinates and their use as herbicides
10/02/2008US20080242866 Synthesis of anthranilamides
10/02/2008US20080242706 neurodegenerative diseases; to remove free iron or iron accumulation in neural tissues; iron chelators; improved chemical stability, penetration through blood brain barrier; reacting 3-hydroxy-4-pyridinone/3-hydroxy-4-pyranone derivatives; 1-cyclopropyl-2-difluoromethyl-5-hydroxy-1H-pyridin-4-one
10/02/2008US20080242705 Fluridone as an Anti-Inflammatory Agent
10/02/2008US20080242702 Paclitaxel enhancer compound
10/02/2008US20080242698 Antiepilrptic agents; antiischemic agents; vision defects; skin disorders; muscular disorders; anticonvulsants;analgesics; Parkinson's disease; huntington's disease; amyotrophic lateral sclerosis; multiple sclerosis
10/02/2008US20080242656 N-Substituted-N-Sulfonylaminocyclopropane Compounds and Pharmaceutical Use Thereof
10/02/2008US20080242593 Such as 2-(((9H-fluoren-9-yl)methoxy)carbonylamino)-3-(6-(2-ethylphenyl)pyridin-3-yl)propanoic acid; stability to proteolytic cleavage
10/02/2008DE102007016139A1 Verfahren zur regioselektiven Oxygenierung von N-Heterozyklen Method for the regioselective oxygenation of N-heterocycles