Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
01/1999
01/12/1999US5859029 Heterocyclic compounds method of preparing them and pharmeutical compositions in which they are present
01/12/1999US5859011 Dihydropyridine derivatives as bradykinin antagonist
01/12/1999US5859002 HIV protease inhibitors
01/12/1999US5858925 Heterocyclylbenzonitriles
01/12/1999US5858736 Contacting dinitrile in aqueous mixture with enzyme catalyst having aliphatic nitrilase activity or combination of nitrile hydratase and amidase activity, contacting product with hydrogen and hydrogenation catalyst to produce lactam
01/07/1999WO1999000376A1 Novel heterocyclic compounds
01/07/1999WO1999000369A1 Process for preparing nifedipine
01/07/1999WO1999000368A1 Substituted 3-(benzylamino)piperidine derivatives and their use as therapeutic agents
01/07/1999WO1999000367A1 Novel heterocyclic compounds
01/07/1999WO1999000366A1 Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives
01/07/1999WO1999000365A1 Novel nitroxyl compounds and drugs and reagents containing the same as the active ingredient
01/07/1999WO1999000362A1 Synthesis of aminocarbonyl substituted lactams
01/07/1999WO1999000127A1 Antithrombotic agents
01/07/1999WO1999000121A1 Antithrombotic agents
01/07/1999EP0889036A1 HIV protease inhibitors
01/07/1999EP0888320A1 Novel n-aminoalkyl-2-anthracenecarboxamides; new dopamine receptor subtype specific ligands
01/07/1999EP0888319A1 Substituted 1,2,3,4-tetrahydronaphthalene derivatives
01/07/1999EP0888304A1 Substituted 3-aryl-3-carboxyalkyl glutaramides, method for preparing same by 4-arylo-4-cyanoheptane dicarboxylic acid cyclisation, and use thereof for preparing 3-aryl-3-hydroxyalkylpiperidines
01/07/1999EP0888303A1 Synthetic derivatives of rapamycin as multimerizing agents for chimeric proteins with immunophilin-derived domains
01/07/1999EP0888302A1 N- (r)-1- 3-(4-piperidyl)propionyl-3-piperidylcarbonyl]-2(s)-acetylamino-beta-alanine as fibrinogen receptor antagonist
01/07/1999EP0888114A1 USE OF (+)-$g(a)-(2,3-DIMETHOXYPHENYL)-1- 2-(4-FLUOROPHENYL)ETHYL]-4-PIPERIDINEMETHANOL IN TREATING DEPRESSIVE DISORDERS AND BIPOLAR DISORDERS
01/07/1999DE19829229A1 Hydrazinderivate Hydrazine
01/07/1999DE19812066A1 Catalytic system for oligomerisation of ethylene@ to linear alpha olefin
01/07/1999CA2294312A1 Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives
01/07/1999CA2294126A1 Antithrombotic agents
01/07/1999CA2294042A1 Antithrombotic agents
01/07/1999CA2291734A1 Substituted 3-(benzylamino)piperidine derivatives and their use as therapeutic agents
01/06/1999CN1204319A Processes and intermediates for preparing 1-benzyl-4-((5,6-dimethoxy-1-indanon)-2-Yl) methyl piperidine
01/06/1999CN1204315A New phenylamidine derivatives process for preparing the same and their use as medicaments
01/06/1999CN1203923A Catalytic system
01/05/1999US5856505 Intermediates for the manufacture of dicarboxamides having thrombin inhibiting activity
01/05/1999US5856494 From acetone or condensates and ammonia
01/05/1999US5856491 Reacting secondary amine with terminally unsaturated electrophilic compound in presence of n-methylpyrrolidinone solvent
01/05/1999US5856346 Short-acting dihydropyridines
01/05/1999US5856338 Sulfonamide-substituted compounds, processes for their preparation, their use as a medicament or diagnostic, and pharmaceutical preparation comprising them
01/05/1999US5856318 Nitrogen-containing cyclohetero cyclo-heteroaminoaryl derivatives for CNS disorders
01/05/1999US5856311 Derivatives of β-aminopropionic acid with a fungicidal activity
01/05/1999US5856307 Peptide derivatives as kininogenase inhibitors
01/05/1999US5856273 Controlling weeds
01/05/1999CA2157117C Spirocyclic piperidine derivatives
12/1998
12/30/1998WO1998058949A1 Treatment of insulin resistance with growth hormone secretagogues
12/30/1998WO1998058934A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
12/30/1998WO1998058901A1 3-anilino-2-cycloalkenone derivates
12/30/1998EP0886637A1 Inhibitors of microsomal triglyceride transfer protein and method
12/30/1998EP0886636A1 Novel piperidines derived from 1-/(piperazin-1-yl)aryl(oxy/amino)carbonyl/-4-aryl-piperidine as selective 5-ht-1d.beta. receptor antagonists
12/30/1998EP0666848B1 Substituted n-phenylglutarimides and n-phenylglutaric acid amides, their preparation and use in agriculture
12/30/1998EP0648130B1 Radioiodinated benzovesamicol analogs for cholinergic nerve mapping
12/30/1998CN1203226A Paroxetine and process for preparing medical salts thereof
12/30/1998CA2294464A1 Treatment of insulin resistance
12/29/1998US5854249 Opioid diarylmethylpiperazines and piperidines
12/29/1998US5854234 Amidino dervatives useful as nitric oxide synthase inhibitors
12/24/1998DE19725664A1 3-Benzylpiperidine 3 Benzylpiperidine
12/23/1998WO1998057959A1 Benzo(5,6)cyclohepta(1,2-b)pyridine derivatives for the inhibition of farnesyl protein transferase
12/23/1998WO1998057953A1 3-benzylpiperidine
12/23/1998WO1998057909A1 Process for the production of radioiodinated neuroreceptor agents
12/23/1998WO1998057640A1 Alpha 1a adrenergic receptor antagonists
12/23/1998WO1998057639A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998WO1998057638A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998EP0885215A1 Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
12/23/1998EP0885213A1 Fibrinogen receptor antagonists
12/23/1998EP0885205A1 Fibrinogen receptor antagonists
12/23/1998EP0885204A1 Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds
12/23/1998EP0885192A1 Dihydropyridine-, pyridine-, benzopyran- one- and triazoloquinazoline derivative, their preparation and their use as adenosine receptor antagonists
12/23/1998EP0885191A1 Resolution of threo-methylphenidate
12/23/1998EP0885190A1 Novel n-substituted 4-((4'-aminobenzoyl)-oxymethyl)-piperidines having gastric prokinetic properties
12/23/1998EP0885180A1 Stabilized monomer composition
12/23/1998EP0885004A1 Use of 4-phenyl-3,6-dihydro-2h-pyridyl derivatives as nmda receptor subtype blockers
12/23/1998CN1202882A New LH-RH antigonists with improved effectiveness
12/23/1998CN1202826A Use of 1-(2-naphth-2-ylethyl)-4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridine for preparing drugs for treating amyotrophic lateral scherosis
12/23/1998CN1041317C Olefin polymer compositions including at least one monomeric ester and its use
12/23/1998CN1041309C Method for preparing piperidine derivatives
12/23/1998CA2294590A1 Alpha 1a adrenergic receptor antagonists
12/23/1998CA2294379A1 3-benzylpiperidine
12/23/1998CA2294349A1 Alpha 1aadrenergic receptor antagonists
12/23/1998CA2294346A1 Alpha 1a adrenergic receptor antagonists
12/23/1998CA2293317A1 Process for the production of radioiodinated neuroreceptor agents
12/22/1998US5852221 Optically active β-aminoalkoxyborane complex
12/22/1998US5852192 Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
12/22/1998US5852044 Use of NK1 receptor antagonists for preparing cardio-regulatory drugs
12/22/1998US5852043 HIV protease inhibitors
12/17/1998WO1998056787A1 4-Phenylpiperidine compounds
12/17/1998WO1998056763A1 Reagents for assaying central local acetylcholinesterase activity
12/17/1998WO1998056746A1 Polymerization inhibition of acrylates using blends of nitroxides
12/17/1998WO1998056249A1 Method for enhancing the activity of glaucoma drugs
12/17/1998CA2293539A1 Reagents for assaying central local acetylcholinesterase activity
12/16/1998EP0883608A1 Optical resolution of methylphenidate by 0,0'-bisaroyl tartaric acids
12/16/1998EP0883607A1 Processes and intermediates for preparing 1-benzyl-4-((5,6-dimethoxy-1-indanon)-2-yl)methylpiperidine
12/16/1998EP0883405A1 Amidino protease inhibitors
12/16/1998EP0883403A1 Method for treating sexual dysfunctions
12/16/1998EP0703902B1 Process for the production of piperidine derivatives
12/16/1998CN1202153A 3-(4-subst.-piperidinyl-1)-1-(3,4-dichlorophenyl) propyl carbamates and ureas and derivatives as neurokinin antagonists
12/16/1998CN1202152A 4-(oxyalkoxyphenyl)-3-oxy-piperidines for treating heart and kidney insufficiency
12/15/1998US5849924 Highly selective process for the preparation of enantiomerically pure phenyl-substituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives
12/15/1998US5849860 Polyethylene-protein conjugates
12/15/1998US5849762 Peripherally acting anti-pruritic opiates
12/15/1998US5849761 Peripherally active anti-hyperalgesic opiates
12/15/1998US5849760 2-(arylalkenyl)azacycloalkane derivatives as ligands for sigma receptors
12/15/1998US5849755 3-amidochromanylsulfonyl(thio)ureas, processes for their preparation, their use, and pharmaceutical preparations comprising them
12/15/1998US5849732 Phenol compound having antioxidative activity and the process for preparing the same
12/15/1998CA1340223C 3,3-diphenylpropyl amines and pharmaceutical compositions and cholinergic uses thereof