Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
10/2001
10/03/2001CN1315861A Use of R(+)-alpha-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol for treatment of sleep disorders
10/03/2001CN1315319A Process for preparing ethyl-sulfonylpiperidine derivatives
10/02/2001USH1996 Agriculture
10/02/2001US6297374 Nitroimino-nitromethylene—azole or-azine heterocyclic compounds, insecticidal compositions containing them, and insecticidal methods of using them
10/02/2001US6297260 Nitrosated and nitrosylated nonsteroidal antiinflammatory compounds, compositions and methods of use
10/02/2001US6297259 Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl) benzamides useful for the treatment of allergic diseases
10/02/2001US6297247 Particularly stromelysin-1 and gelatinase a (72 kd gelatinase)
10/02/2001US6297233 Lactam inhibitors of FXa and method
10/02/2001CA2212451C Stereoselective and useful preparation of 3-substituted 4-aryl piperidine compounds
10/02/2001CA2037541C Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment
09/2001
09/27/2001WO2001070736A1 N-(heterocyclyl)benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
09/27/2001WO2001070734A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
09/27/2001WO2001070691A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors
09/27/2001WO2001070690A1 Heterocyclic side chain containing metalloprotease inhibitors
09/27/2001WO2001070688A2 N-(2,6-dioxo-piperidin-3-yl) benzamides and their use as immune modulators
09/27/2001WO2001070677A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
09/27/2001WO2001070670A1 Novel phenylalanine derivative
09/27/2001WO2001070230A2 Compounds with 5-ht activity useful for controlling visual field loss
09/27/2001WO2001070223A1 Compounds with 5-ht2 and 5-ht1a agonist activity for treating glaucoma
09/27/2001WO2001070222A2 Compounds with 5-ht1a activity useful for treating disorders of the outer retina
09/27/2001WO2001017972A3 Novel herbicides
09/27/2001US20010025106 Antiallergens, bronchodilator
09/27/2001US20010025052 Novel nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
09/27/2001US20010025041 Amidino protease inhibitors
09/27/2001DE10013499A1 New N-(2,6-dioxo-piperidin-3-yl)-benzamide derivatives, useful as immunomodulators causing no general immunosuppression, is useful for the treatment of inflammatory or autoimmune disease
09/27/2001CA2404131A1 Heterocyclic side chain containing, n-substituted metalloprotease inhibitors
09/27/2001CA2404076A1 Heterocyclic side chain containing metalloprotease inhibitors
09/27/2001CA2400637A1 Compounds with 5-ht2 and 5-ht1a agonist activity for treating glaucoma
09/27/2001CA2400168A1 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
09/27/2001CA2399985A1 Compounds with 5-ht activity useful for controlling visual field loss
09/26/2001EP1136490A1 New forms of paroxetin hydrochloride
09/26/2001EP1136475A1 Piperidine and piperazine compounds for use in the treatment of Alzheimer
09/26/2001EP1135379A1 Antitumor dibenzofluorene derivatives
09/26/2001EP1135370A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
09/26/2001EP0799201B1 Process for the preparation of substituted 4-ethyl-piperidines
09/26/2001CN1314888A Crystalline forms of osanetant
09/26/2001CN1314887A Ester of (+)-alpha-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol and their use as prodrugs of the 5HT2A receptor antagonist MDL 110,907
09/26/2001CN1314883A Amino acid derivatives and drug containing the same as the active ingredient
09/26/2001CN1071738C Carboxylic derivatives exhibiting phospholipase A2 inhibitory activity
09/25/2001US6294673 Mixing methyl 2-(2-nitrobenzylidene) acetoacetate and methyl 3-aminocrotonate in alkanol solvent in absence of catalylst; heating reaction mixture in closed container; isolating nifedipine
09/25/2001US6294556 Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds
09/25/2001US6294555 1-[(1-Substituted-4-piperidinyl)methyl]-4-piperidine derivative, process for producing the same, medicinal compositions containing the same and intermediates of these compounds
09/25/2001US6294554 Muscarinic antagonists
09/25/2001US6294551 N-linked sulfonamides of heterocyclic thioesters
09/25/2001US6294544 Blood flow increased in vessels for eyes in mammals
09/25/2001US6294542 Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
09/25/2001US6294533 Calcium channel blockers
09/25/2001US6294517 Compositions and kits comprising alpha-adrenergic receptor antagonists and nitric oxide donors and methods of use
09/25/2001CA2213404C Use of angiogenesis suppressors for inhibiting hair growth
09/20/2001WO2001068645A2 N-cyanomethylcarboxamides and their use as protease inhibitors
09/20/2001WO2001068619A1 5-amide substituted diarylamines as mex inhibitors
09/20/2001WO2001068606A1 Process for preparing sterically hindered n-oxyl compounds
09/20/2001WO2001068605A1 Polycyclic aryl and heteroaryl substituted benzenes useful for selective inhibition of the coagulation cascade
09/20/2001WO2001068604A2 3-substituted piperidines comprising urea functionality, and methods of use thereof
09/20/2001WO2001068588A1 POLYMER-IMMOBILIZED α-IMINOESTER
09/20/2001WO2001068575A1 Fluoroalkylonium salt type cation or acid generator generating cation or acid upon irradiation with energy ray
09/20/2001WO2001068140A2 Opioid formulations
09/20/2001WO2000071506A9 Naphthalene ureas as glucose uptake enhancers
09/20/2001US20010023269 Materials handling; fluid flow
09/20/2001US20010023249 Calcium channel blockers
09/20/2001CA2403017A1 5-amide substituted diarylamines as mex inhibitors
09/20/2001CA2402865A1 Opioid formulations
09/19/2001EP1133489A1 Isonipecotamides for the treatment of integrin-mediated disorders
09/19/2001EP1133473A1 New manufacturing process
09/19/2001EP0869954B1 Heterocyclic compounds for use in the treatment of neurogenic inflammation
09/19/2001EP0800516B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME
09/19/2001CN1313855A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta
09/19/2001CN1313847A Method for preparing alkoxyamines from nitroxides
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/19/2001CN1071329C Aryl glycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds
09/18/2001US6291722 Contacting grignard reagent of formula r.sup.7--mgx with an aryl compound of the formula r.sup.1--x in the presence of a catalytic amount of coordination comprising trasition metal complexed to phosphine oxide to prepare bisaryl compound
09/18/2001US6291672 Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
09/18/2001US6291657 N-butyldeoxygalactonojirimycin; suppression of glycolipid biosynthesis; microbiocides; treatment of gaucher's disease
09/18/2001US6291481 Conditions related to a hampered or impaired gastric emptying and more generally to treat conditions related to a hampered or impaired gastrointestinal transit.
09/18/2001US6291478 Compounds of the benzylaminodiacetamide family, compositions comprising them, preparation process and uses
09/18/2001US6291450 Carboxylic acid substituted heterocycles, derivatives thereof and methods of use
09/18/2001US6291417 Cleaning process
09/18/2001US6289745 High temperature insertion type flow element and mounting extension
09/13/2001WO2001066521A1 Azacyclic compounds for use in the treatment of serotonin related diseases
09/13/2001WO2001066114A1 Novel methods using cholinesterase inhibitors
09/13/2001WO2001009138A3 Chemokine receptor antagonists and methods of use therefor
09/13/2001US20010021791 Cyclopropyl phenyl ketone compound
09/13/2001US20010021778 Oxidizing a 4-phenyl-N-acyldihydropyridine
09/13/2001US20010021715 Gastrointestinal disorders
09/12/2001EP1132379A1 Novel thiol derivatives, process for producing the same and utilization thereof
09/12/2001EP1132370A2 Process for producing n-substituted polyhydroxy nitrogen-containing heterocyles
09/12/2001EP1132085A1 Drugs and reagents containing n-acyloxylated cycloalkyl compounds as the active ingredient
09/12/2001EP1131291A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii
09/12/2001EP1131290A1 Piperidine ccr-3 receptor antagonists
09/12/2001EP1131289A1 Processes for preparing 2-piperidineethanol compounds
09/12/2001EP0820450B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof
09/12/2001EP0682514B1 Use of topical anesthetics for the manufacture of a medicament for the treatment of bronchial asthma
09/12/2001CN1312802A Cycloalkyl-substituted aryl-piperazines, piperidines and tetrahydropyridines as serotonergic agents
09/12/2001CN1312799A Bispiperidines as antithrombotic agents
09/12/2001CN1312716A Use of optically pure (-)-norcisapride in treatment of apnea, bulimta and other disorders
09/12/2001CN1070831C Stabilized monomer composition
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
09/11/2001US6288231 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
09/11/2001US6288123 Therapeutic guanidines
09/11/2001US6288086 N-hydroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors