Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/1996
10/29/1996US5569800 Reacting phosphonic acid ester compound containing a pyrene ring with a carbonyl compound in the presence of a basic compound
10/29/1996US5569777 Process for the preparation of a substituted 2,5-diamino-3-hydroxyhexane
10/29/1996US5569768 Angiotensin II antagonists
10/29/1996US5569668 Nematophin: 3-indoleethyl-3-methyl-2-oxo-pentanamide; antibiotics
10/29/1996US5569659 4-arylpiperazines and 4-arylpiperidines
10/29/1996CA2057912C (1,2n) and (3,2n)-carbocyclic-2-amino tetralin derivatives
10/24/1996WO1996033184A1 Thf-containing sulfonamide inhibitors of aspartyl protease
10/24/1996WO1996033171A1 1h-pyrrol-1-yl and 1h-indol-1-yl aryl sulphones, processes for their preparation and use for the therapy of hiv-1 infections
10/24/1996WO1996033160A1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production
10/24/1996WO1996032968A1 Compounds for cancer imaging and therapy
10/24/1996WO1996032946A1 Compositions and methods to prevent toxicity induced by nonsteroidal antiinflammatory drugs
10/24/1996WO1996023769A3 Heterocyclic compounds possessing 5ht2c receptor antagonist activity
10/24/1996CA2215839A1 Compounds for cancer imaging and therapy
10/23/1996EP0738724A2 Process for the preparation of an N-terbutylamide derivative
10/23/1996EP0738258A1 Process for preparing n-substituted glycinic acids or glycine esters and use of said process in indigo synthesis
10/23/1996EP0646110B1 N-substituted 3-azabicyclo[3.2.0]heptane derivatives useful as neuroleptic agents
10/23/1996EP0574383B1 Color modified melanins and methods for their preparation and use
10/23/1996CN1134153A Matrix metalloprotease inhibitors
10/23/1996CN1033089C Process for preparation of aryl piperazinyl-heterocyclic compounds
10/22/1996US5567844 Process for preparing 1-phenyl-2-amino-3-fluoro-1-propanols
10/22/1996US5567827 4-Hydroxyphenylthio derivatives, their preparation and their use for the preparation of aminoalkoxyphenylsulphonyl derivatives
10/22/1996US5567713 Hypoglycemic agents
10/22/1996US5567692 9-[(substituted glycyl) amido)]-6-demethyl-6-deoxytetracyclines
10/22/1996CA1338671C Light-induced killing of carcinoma cells
10/17/1996WO1996032381A1 Carbazole derivative
10/17/1996WO1996032380A1 Substituted indolylmethylene-oxindole analogues as tyrosine kinase inhibitors
10/17/1996WO1996032379A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS
10/17/1996WO1996032366A1 Naphthol derivatives and process for producing the same
10/17/1996CA2217707A1 Indole derivatives as cgmp-pde inhibitors
10/17/1996CA2192542A1 Naphthol derivatives and process for producing the same
10/16/1996EP0737678A1 4-Indolylpiperazinyl derivatives
10/16/1996EP0737677A1 4-Indolylpiperazinyl derivates
10/16/1996EP0737670A1 Tricyclic amides, processes for their preparation, and pharmaceutical compositions containing them
10/16/1996EP0737232A1 Modular design and synthesis of aminimide containing molecules
10/16/1996EP0526529B1 An improved process for the preparation of substituted indolone derivatives
10/16/1996CN1133284A Method of systhesizing diphenylamine from aniline
10/16/1996CN1033029C Prepn. of indenoindole compound
10/16/1996CN1033028C Process for preparing new derivatives of 2,2-dimethyl cyclopropane carboxylic acid
10/15/1996US5565604 Chemical intermediate for hiv protease inhibitor
10/15/1996US5565580 Treatment of central nervous system disorders
10/15/1996US5565579 Neuroprotective agent
10/15/1996US5565484 Cardiovascular disorders
10/15/1996US5565483 3-substituted oxindole derivatives as potassium channel modulators
10/15/1996US5565470 Cycloaminoalkoxyphenyl derivatives, a process for their preparation as well as the compositions containing them
10/15/1996US5565447 Almotriptan malate; treating headaches, movement disorders, depression, anxiety
10/15/1996US5565418 Retroviral protease inhibiting compounds
10/15/1996CA1338647C Inhibitors of lysyl oxidase
10/11/1996CA2173693A1 4-indolylpiperazinyl derivatives
10/11/1996CA2173690A1 4-indolylpiperazinyl derivatives
10/10/1996WO1996031527A1 Protease inhibiting succinic acid derivatives
10/10/1996WO1996031209A1 Pharmaceutical agents for the treatment of alzheimer's disease
10/09/1996EP0736525A1 Benzonitriles and -fluorides as 5-HT agonists and antagonists
10/09/1996EP0736036A1 Kininogen inhibitors
10/09/1996EP0736008A1 Indole derivatives as anti-estrogens
10/09/1996EP0736007A1 Non-peptide tachykinin receptor antagonists
10/09/1996EP0735821A1 Methods for the treatment or prevention of conditions associated with amyloidogenic reptides
10/09/1996EP0354921B1 Use of melatonin for the manufacture of a contraceptive composition
10/09/1996CN1132756A Antiviral ethers of aspartate protease substrate isosteres
10/08/1996US5563168 Fungicides, insecticides
10/08/1996US5563142 Diaromatic substituted compounds as anti-HIV-1 agents
10/08/1996US5563115 Pre- and postemergence herbicides
10/03/1996WO1996030348A1 Synthesis of bis-indolylmaleimides
10/03/1996WO1996030340A1 Method for the preparation of a n-alkoxy-(tetra- or hexahydro)-phthalimide and method for the preparation of a n-alkoxyamine
10/03/1996WO1996030014A1 Inhibitors of farnesyl-protein transferase
10/03/1996WO1996029974A2 Compositions and methods utilizing nitroxides in combination with biocompatible macromolecules
10/03/1996WO1996024348A3 Use of carbazole compounds for the treatment of congestive heart failure
10/03/1996CA2216651A1 Compositions and methods utilizing nitroxides in combination with biocompatible macromolecules
10/03/1996CA2216526A1 Inhibitors of farnesyl-protein transferase
10/02/1996EP0734384A1 3-substituted 1-arylindole compounds
10/01/1996US5561733 Thermally stable electro-optic device and method
10/01/1996US5561149 For nasal administration
10/01/1996US5561142 Substituted sulfonamides as selective β3 agonists for the treatment of diabetes and obesity
10/01/1996US5561141 MDR reversal agents
09/1996
09/26/1996WO1996029304A1 Nonpeptides as tachykinin antagonists
09/26/1996CA2211191A1 Nonpeptides as tachykinin antagonists
09/25/1996EP0733680A2 Reactive dyes with a benzo-anellated heterocycle as reactive group
09/25/1996EP0733042A1 Process for preparing spirocyclic lactams
09/25/1996EP0733041A1 Anthracene spiro-pyrrolidines as immuno-modulators
09/25/1996EP0733040A1 Piperazine-substituted pyrroloanthracene as immuno-moderators
09/25/1996EP0733039A1 Substituted pyrroloanthracenes and pyrroloanthracene diones as immunomodulators
09/25/1996EP0733038A1 Bleach activator preparation
09/25/1996EP0733035A1 Tricyclic derivatives, pharmaceutical compositions containing them
09/25/1996CN1131942A HIV protease inhibitors
09/25/1996CN1131898A Use of indenoindole compounds
09/24/1996US5559256 Aminediol protease inhibitors
09/24/1996US5559247 Carboxylate and heat-sensitive recording material using same
09/24/1996US5559245 Intermediates to 4-amino- hexahydrobenz (cd) indoles and processes therefor
09/24/1996US5559228 Synthesis of bisindolylmaleimides
09/24/1996US5559143 Anxiolytics, antidepressants, hypotensive agents, treatment of migraine
09/24/1996US5559127 Fibrinogen receptor antagonists
09/19/1996WO1996028441A1 Heterocyclic substituted piperazinone derivatives as tachykinin receptor antagonists
09/19/1996WO1996010999A3 Lta4 hydrolase inhibitor pharmaceutical compositions and methods of use
09/18/1996EP0732332A1 Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation
09/18/1996EP0731802A1 N-substituted azabicycloalkane derivatives as neuroleptika asf
09/18/1996EP0731790A1 Tachykinin antagonists
09/18/1996CN1131418A Novel fused-ring carboxylic acid compound or salt thereof, and medicinal use thereof
09/18/1996CN1131417A Substituted 4-carbamoyl pyrrolin-2-one and dihydrofuran-2-one derivatives and their use as pesticides
09/18/1996CN1131144A Glycinamide derivatives, processes for their preparation and medicines containing them
09/18/1996CA2171695A1 Substituted benzothienylpiperazines their use as medicaments, and processes for their preparation
09/17/1996US5556989 Indoline compounds useful for dyeing keratinous fibres