Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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10/16/2008 | WO2008122105A1 Novel amorphous form of carvedilol phosphate and processes for the preparation thereof |
10/16/2008 | WO2008106125A3 Deuterated derivatives of silodosin as alpha la-adrenoceptor antagonists |
10/16/2008 | WO2008021745A3 Hepatitis c virus entry inhibitors |
10/16/2008 | WO2007109178A9 Indole derivatives as inhibitors of histone deacetylase |
10/16/2008 | WO2007070892A3 Useful indole compounds |
10/16/2008 | US20080255350 Substituted aza-indoles as inhibitors of poly(adp-ribose) polymerase (parp) |
10/16/2008 | US20080255221 Novel hydroxamates as therapeutic agents |
10/16/2008 | US20080255214 Novel hydroxamates as therapeutic agents |
10/16/2008 | US20080255201 Ppar active compounds |
10/16/2008 | US20080255189 using an thiourea compound or carbonyl thiourea compound; therapy for drug resistant infections |
10/16/2008 | US20080255169 4'-Fluoro-biphenyl-3-sulfonic acid benzo[1,3]dioxol-5-ylamide, for example; for use as an alpha 2 beta 1 integrin I domain inhibitor; use as a medicament for treating thrombosis and cancer spread |
10/16/2008 | US20080255154 Cycloalkylcarbonyl-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-ones: N-methyl-5-[4-(1-{[3-oxo-1'H,3H-spiro[2-benzofuran-1,3'-pyrrolidin]-1'-yl]carbonyl}cyclopropyl)phenyl]pyridine-2-carboxamide; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; diabetes |
10/16/2008 | US20080255149 1-Oxopiperidine derivatives; amides derived from fused and/or spiro polyheterocycles such as decahydro-(iso)quinoline, tetrahydro(iso)quinoline, piperazine, piperidine, indole, or (iso)indole; histone deacetylase inhibitors; antiproliferative, antitumor, and antitumor agents; hyperplasia; immune diseases |
10/16/2008 | US20080255144 (3'-Chloro-4-methanesulfonyl-biphenyl-2-yl)-[4-(3,4-dichloro-phenyl)-piperazin-1-yl]-methanone; neurological and neuropsychiatric disorders including schizophrenia |
10/16/2008 | US20080255129 3-Heteroaryl-3,5-dihydro-4-oxo-4H-pyridazino[4,5-b]indole-1-acetamide derivatives, their preparation and their application in therapeutics |
10/16/2008 | US20080255117 Sulfonyltryptophanols |
10/16/2008 | US20080255111 (4'-{[2-(tert-Butoxycarbonyl)-3-hydroxy-4-(trifluoromethyl)benzyl]oxy}-1,1'-biphenyl-4-yl)acetic acid; vascular restenosis following angioplasty, endarterectomy, percutaneous transluminal coronary angioplasty (PTCA) or stent implantation, blood coagulation diseases |
10/16/2008 | US20080255102 1-(2,3-dihydro-4H-1,4-benzoxazin-4-yl)-3-(methylamino)-1-phenylpropan-2-ol; fluctuations of sex steroid lelels; monoamine reuptake modulator; antidepressant, sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue and fibromylagia syndrome, stress and urinary incontinence |
10/16/2008 | US20080254546 Arsenic complexes; transmetallization |
10/16/2008 | US20080254318 Charge generating and charge transfer compounds;applying carbazole compound; reducing drive voltage ; emission efficiency; accuracy |
10/16/2008 | US20080254128 Process for the precipitation and isolation of 6,6-dimethyl-3-aza-bicyclo [3.1.0] hexane-amide compounds by controlled precipitation and pharmaceutical formulations containing same |
10/16/2008 | CA2681861A1 Ornithine derivative |
10/15/2008 | EP1979317A1 Benzoisoindole derivatives for the treatment of pain |
10/15/2008 | EP1979316A1 Benzo (f) isoindol-2-ylphenyl acetic acid derivatives as ep4 receptor agonists |
10/15/2008 | EP1979315A2 Methods for treating hepatitis c |
10/15/2008 | EP1979314A2 Indole sulfonamide modulators of progesterone receptors |
10/15/2008 | EP1742642B1 Phosphonate analogs of hiv integrase inhibitor compounds |
10/15/2008 | EP1708998B1 Indol-alanine derivatives as selective s1p4-agonists |
10/15/2008 | EP1692124B1 Biaryl sulfonamides as mmp inhibitors |
10/15/2008 | EP1660455B1 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
10/15/2008 | EP1587585B1 Acylsulfonamide compounds as inhibitors of rna-dependent rna (viral) polymerases |
10/15/2008 | EP1569901B1 ARYL, ARYLOXY, AND ALKYLOXY SUBSTITUTED i 1H /i -INDOL-3-YL GLYOXYLIC ACID DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1) |
10/15/2008 | EP1530572B1 Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents |
10/15/2008 | EP1411940B1 Bridged piperidine derivatives as melanocortin receptor agonists |
10/15/2008 | CN101284865A New compound and its medicine use |
10/15/2008 | CN101284811A Synthetic method for chiral carbocyclic ring intermediate of abacavir |
10/15/2008 | CN100425610C Method for preparing phthalocyanines |
10/15/2008 | CN100425592C Indole derivatives |
10/14/2008 | US7435843 Thiobenzoic acid, N-malonylhydrazide in which the free carboxy group is protected; enhances the desirable tumor attacking properties of anticancer agents without further increasing undesirable side-effects |
10/14/2008 | US7435832 Preparing an anhydrous crystal of a malic acid salt of N-[2-(diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide by reacting the acid and amine in a solvent and crystallizing under various process conditions |
10/14/2008 | US7435815 Sulfonylamino-acetic acid derivatives |
10/14/2008 | US7435729 using estrogen antagonist ; anticancer agents |
10/14/2008 | CA2309328C Cyclic amine derivatives and their use as drugs |
10/09/2008 | WO2008121800A1 Methods of separation and detection of bazedoxifene acetate in pharmaceutical compositions |
10/09/2008 | WO2008121686A1 Sub-type selective azabicycloalkane derivatives |
10/09/2008 | WO2008121150A1 Methods for producing and purifying 2-hydrocarbyl-3,3-bis(4-hydroxyaryl)phthalimidine monomers and polycarbonates derived therefrom |
10/09/2008 | WO2008121149A1 Methods for producing and pruifying 2-hydrocarbyl-3.3-bis(4-hydroxyaryl) phthalimidine monomers and polycarbonated derived therefrom |
10/09/2008 | WO2008120899A1 Naphthyl carbazole derivatives, kl host material, the organic light emitting device employing the same, the display device and the illumination device employing the same |
10/09/2008 | WO2008120818A1 Indole derivative having cpla2 inhibitory activity, use of the same and method for producing the same |
10/09/2008 | WO2008120661A1 Novel fused pyrrole derivative |
10/09/2008 | WO2008120241A2 Novel alcohol solvates of perindopril erbumine |
10/09/2008 | WO2008079159A3 Chemicals, compositions, and methods for treatment and prevention of orthopoxvirus infections and associated diseases |
10/09/2008 | WO2008076316A3 Bisulfite purification of an alpha-keto amide |
10/09/2008 | WO2008021625A3 Combination faah inhibitor and analgesic, anti-inflammatory or anti-pyretic agent |
10/09/2008 | WO2008013856A3 Methods and compositions for production, formulation and use of 1 aryl -3-azabicyclo[3.1.0 ] hexanes |
10/09/2008 | US20080249318 Splitting of the corresponding phenylindole compound containing lactam group; cyclooxygenase inhibitor |
10/09/2008 | US20080249317 Novel amorphous form of carvedilol phosphate and processes for the preparation thereof |
10/09/2008 | US20080249315 Having an acylsulfonamide amine-reactive groups; crosslinker for amine containing material such as gel and hydrgels |
10/09/2008 | US20080249306 Method for the Production of Statins |
10/09/2008 | US20080249302 neuronal nitric oxide synthase (nNOS) isoform inhibitors; 2-ethyl-1-(1H-indol-5-yl)-isothiourea; neurogenerative disorders, stroke, reperfusion injury, head trauma, migraine headache, neuropathic pain, drug abuse, hyperalgesia |
10/09/2008 | US20080249155 5-Hydroxyindole-3-Carboxylate Derivatives and Uses Thereof |
10/09/2008 | US20080249135 Compounds for alzheimer's disease |
10/09/2008 | US20080249110 Novel Substituted 3-Sulfur Indoles |
10/09/2008 | US20080249098 peripheral benzodiazepine receptors; 7-fluoro-N,N,5-trimethyl-4-oxo-3-(pyridin-2-yl)-3,5-dihydro-4H-pyridazino[4,5-b]indole-1-carboxamide; for the treatment of various types of peripheral neuropathies, amyotrophic lateral sclerosis |
10/09/2008 | US20080249091 Indoles Useful in the Treatment of Inflammation |
10/09/2008 | US20080249071 inhibitory activity against the activation of inflammatory cytokines such as interleukin (IL)-1, IL-6, IL-8 and tumor necrosis factor (TNF- alpha ), NF- kappa K B; inflammatory disorders, autoimmune diseases; side effects reduction; immuno suressants; N-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxybenzamide |
10/09/2008 | US20080248511 Methods to quench light from optical reactions |
10/09/2008 | CA2682185A1 Methods of separation and detection of bazedoxifene acetate in pharmaceutical compositions |
10/09/2008 | CA2681979A1 Indole derivatives having cpla2 inhibiting activity and applications and production methods of the same |
10/09/2008 | CA2679728A1 Sub-type selective azabicycloalkane derivatives |
10/08/2008 | EP1978016A1 Asymmetric reduction method |
10/08/2008 | EP1976840A1 Cyclohexyl piperazinyl methanone derivatives and their use as histamine h3 receptor modulators |
10/08/2008 | EP1976829A2 N-(6-membered aromatic ring)-amido anti-viral compounds |
10/08/2008 | EP1606351A4 Cyanine dye labelling reagents with meso-substitution |
10/08/2008 | EP1539693B9 Cannabinoid receptor agonists |
10/08/2008 | EP1379246B1 Nociceptin analogs |
10/08/2008 | EP1341785B1 Hydrolysis of r(r*,r*)-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4- [(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid esters with calcium hydroxide |
10/08/2008 | CN101282932A Carboxyamine compounds and their use in the treatment of HDAC dependent diseases |
10/08/2008 | CN101282931A Tanaka Hiroaki |
10/08/2008 | CN101282930A Fab I inhibitor and process for preparing same |
10/08/2008 | CN101282929A Compounds and compositions as tpo mimetics |
10/08/2008 | CN101279969A Organic electroluminescent material and application thereof |
10/08/2008 | CN101279888A 9,10-divinyl anthracene derivate and application thereof to organic electroluminescent devices |
10/08/2008 | CN100424084C (Zinc) porphyrin - perylene diimide ( PDI) - C60 ternary system and its synthesis method |
10/08/2008 | CN100424074C N-isoindole dione substituted phenylurea compound with herbicidal activity |
10/08/2008 | CN100424073C Synthesis of DL-tryptophane-alpha-N |
10/07/2008 | US7432392 Ester derivatives and medical use thereof |
10/07/2008 | US7432380 Crystalline form of Fluvastatin sodium |
10/07/2008 | US7432285 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use |
10/07/2008 | US7432281 4-(2,2-dichloro)-N-(quinolin-3-yl)benzamide; (1R,2R)2-methyl-N-(quinolin-3-yl)-4-(2-(trifluoromethyl)cyclopropyl)benzamide; inflammation-related conditions in mammals, arthritis, Parkinson's/Alzheimer's diseases, stroke, asthma; acute/chronic or neuropathic pain; VR1 agonist/antagonist |
10/07/2008 | US7432255 Histamine 3 receptor antagonists/inverse agonists ; (4-isopropyl-piperazin-1-yl)-[1-(1-isopropyl-pyrrolidin-3-yl)-1H-indol-5-yl]-methanone; obesity, metabolic syndrome (syndrome X), and other eating disorders |
10/07/2008 | US7431997 Luminescent 2,2'-aryliminobis(5-phenylcarbazole) derivatives; electrically stable, has the ability to transport charges and a high glass transition temperature, and is not susceptible to crystallization |
10/07/2008 | CA2331461C Analogs of 2-phthalimidinoglutaric acid and their use as inhibitors of angiogenesis |
10/02/2008 | WO2008117815A1 Inhibitor for cell death caused by endoplasmic reticulum stress or oxidation stress |
10/02/2008 | WO2008117773A1 Process for production of asymmetric tetrasubstituted quinolonecarboxylic acids and intermediates for the production |
10/02/2008 | WO2008117303A1 Indole derivatives and their metal conjugates and uses thereof |
10/02/2008 | WO2008116926A1 Tetrahydroindole derivatives as nadph oxidase inhibitors |
10/02/2008 | WO2008116814A1 Pyrrole and isoindole carboxamide derivatives as p2x7 modulators |
10/02/2008 | WO2008116671A1 2,3,4,9-tetrahydro-1h-carbazoles |
10/02/2008 | WO2008116308A1 Quinolone and tetrahydroquinoline and related compounds having nos inhibitory activity |