Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
06/2006
06/15/2006US20060128974 Cyclometallated complexes of a group 9 or 10 element prepared from an iminated thiophenecarboxaldehyde and a monoanionic beta-diketone ligand or a monoanionic bidentate chelate ligand having a carboxyl group or a phenolic hydroxyl group; used in devices that operate at low voltage with high efficiency
06/15/2006US20060128973 N-[4-[(1E)-3-amino-1-propenyl]phenyl]-4'-(trifluoromethyl)-[1,1'-biphenyl]-2-carboxamide; for treatment of hyperlipidemia, obesity and type II diabetes
06/15/2006US20060128972 N-(p-(2-alpha-carboxybenzylamino)ethylamino)phenyl)p-(p-trifluoromethylphenyl)benzamide; antiobesity and anti-type II diabetic agents
06/15/2006US20060128971 Process for the preparation of the amorphous form of atorvastatin calcium salt
06/15/2006US20060128970 3-Pyrrolidin-2-yl-propionic acid derivatives
06/15/2006US20060128957 Fluorous tagging and scavenging reactants and methods of synthesis and use thereof
06/15/2006US20060128948 obtained by modifying carboxyl groups of biological low-molecular-weight compounds having two or more carboxyl groups with N-hydroxysuccinimide, N-hydroxysulfosuccinimide; used to treat medical devices and the like are non-natural, artificially synthesized products; low toxicity and easily assimilated
06/15/2006US20060128789 Especially 4-(hydroxymethyl)pyrrolidin-3-ol, forming camphor sultam from camphorsulfonic acid, SO2Cl2 and NH3 or forming diethyl 2-(benzyloxymethoxy)-3-(benzyloxymethyl)succinate from diethyl maleate and benzyl chloromethyl ether as an intermediate
06/15/2006US20060128779 Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1H-pyrrol-2-yl)acrylonitrile derivatives
06/15/2006US20060128704 2-Hydroxy-1,2,3,4-tetrahydronaphthalenes substituted in the 8-position with a biphenylcarbonylamino-, biphenylcarbonylaminoalkyl-, biphenylaminocarbonylamino-, or biphenylaminocarbonylaminoalkyl- group; vanilloid receptor antagonists
06/15/2006US20060128632 Peptide inhibitors of smac protein binding to inhibitor of apoptosis proteins (iap)
06/15/2006US20060124017 New compounds, a process for their preparation and their use as dyes and pigments
06/15/2006CA2590220A1 2-alkyl-cycloalk(en)yl-carboxamides
06/15/2006CA2588633A1 Novel anthranilic acid derivative or salt thereof
06/15/2006CA2587318A1 Pyrrolidin-2-one derivatives for use as dp1 receptor agonists
06/14/2006EP1669435A1 Dispersant reaction product with antioxidant capability
06/14/2006EP1667967A1 Process for preparing 2-oxo-1-pyrrolidine derivatives
06/14/2006EP1667966A1 N-alkylated diaminopropane derivatives as modulators of chemokine receptor activity
06/14/2006EP1667955A2 Cycloalkylidene compounds as modulators of the estrogen receptor
06/14/2006EP1667675A1 Entry inhibitors of the hiv virus
06/14/2006EP1667647A2 Monocyclic and bicyclic lactams as factor xa inhibitors
06/14/2006EP1667635A2 Sulfonylaminovalerolactams and derivatives thereof as factor xa inhibitors
06/14/2006EP1620495A4 Imide-linked maleimide and polymaleimide compounds
06/14/2006EP1427702B1 Method for the production of 2-pyrrolidone
06/14/2006EP1268418B1 Pharmaceutically active pyrrolidine derivatives as bax inhibitors
06/14/2006CN1787994A 2,4,6-phenyl substituted cyclic ketoenols
06/14/2006CN1787989A Imino ether derivative compounds and drugs containing the compounds as the active ingredient
06/14/2006CN1787817A 免疫抑制剂化合物及组合物 Immunosuppressant compounds and compositions
06/14/2006CN1785974A (4S)-1-tert butoxy carbonyl-4-amino-L-ethyl prolinate and its synthesis technology
06/14/2006CN1259307C Acylated indanyl amines and their use as pharmaceuticals
06/13/2006USRE39128 Antibacteria drug; respiratory system disorders; otitis
06/13/2006US7060850 Fluorous tagging and scavenging reactants and methods of synthesis and use thereof
06/13/2006US7060845 Stabilized activated derivatives of carbamic acid, their process of preparation and their use for the preparation of ureas
06/13/2006US7060722 Proline derivatives and use thereof as drugs
06/13/2006US7060719 Glutaminyl based DPIV inhibitors
06/13/2006US7060697 Immunosuppressant compounds and compositions
06/13/2006CA2260777C Pentafluorobenzenesulfonamides and analogs
06/08/2006WO2006060810A1 Sulfonamide compounds as cysteine protease inhibitors
06/08/2006WO2006060225A2 Process for asymmetric synthesis of hexahydropyrimido[1,2-a] azepine-2-carboxamides and related compounds
06/08/2006WO2006010095A3 Oxime derivative substituted hydroxyethylamine aspartyl protease inhibitors
06/08/2006WO2005052016B1 Bottom antireflective coatings
06/08/2006US20060122404 Novel compounds comprising a thiocarbonyl-sulfanyl group, which can be used for the radical synthesis of-alpha-perfluoroalkylamines
06/08/2006US20060122403 Atorvastatin calcium form vi or hydrates thereof
06/08/2006US20060122390 Boronic ester and acid compounds, synthesis and uses
06/08/2006US20060122255 Derivatives of N-methyl-N-[(1S)-1-phenyl-2-((3S)-3-hydroxypyrrolidin-1-yl)ethyl]-2,2-diphenylacetamide; for preparation of drugs
06/08/2006US20060122239 Lipid diseases; metabolism diosrders; antiproliferative agents
06/08/2006US20060122235 Amine oxidase inhibitor; use in treating Alzheimer's disease; for example, (RS)-1-[6-(4-fluoro-benzyloxy)-pyridin-3-yl]-5-oxo-pyrrolidine-3-carboxylic acid methylamide
06/08/2006US20060122230 1,5-Diaryl-pyrrole-3-carboxamide derivatives and their use as cannabinoid receptor modulators
06/08/2006US20060122182 Bioassay of testing the compound on the biological system or sample; antihistamines; bronchodilator agents, anticholinergic agents; respiratory system disorders; 2-{(S)-1-[5-(2-methylamino)acetylamino)pentyl]pyrrolidin-3-yl}-2,2-diphenylacetamide
06/08/2006US20060122166 Chemokine receptors; inhibition of HIV replication; acquired immune deficiency syndrome (AIDS); cis N-(4-{2-[3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-4-phenylcyclohexyl)-1H-pyrazole-4-carboxamide
06/08/2006US20060122126 (1S)-1,5-anhydro-1-[3-(1-benzothiene-2-ylmethyl)phenyl-D-glucitol and derivatives are Na+-glucose cotransporter inhibitors and are used to treat diabetes and related diseases such as insulin-resistance and obesity
06/08/2006US20060122124 Therapeutic agent
06/08/2006US20060122100 Melanin extinguisher
06/08/2006US20060122061 Arylphenyl-substituted cyclic ketoenols
06/08/2006US20060120959 Method for the selective and quantitative functionalization of immunoglobulin fab fragments, conjugate compounds obtained with the same and compositions thereof
06/08/2006US20060117497 Azo dye for hair; thickener is anionic amphiphilic polymer
06/07/2006EP1666466A2 Mutilin derivatives and their use as Antimicrobials
06/07/2006EP1666461A2 Polyaspartimides useful as reactive components for polyisocyanates in two-component polyurethane coating compositions
06/07/2006EP1666460A1 Preventive for cerebral stroke recurrence
06/07/2006EP1666459A2 Aminocyclohexyl ether compounds and uses thereof
06/07/2006EP1666047A1 Pharmaceutical compositions comprising nitric oxide-releasing pyrrolidones
06/07/2006EP1664323A1 Enzymatic synthesis of enatiopure intermediates by means of cholesterolesterase from yeasts
06/07/2006EP1664088A2 Hemiasterlin derivatives and uses thereof
06/07/2006EP1664084A1 Process for the manufacture of an enantiopure compound
06/07/2006EP1664031A2 Adamantane and azabicyclo-octane and nonane derivatives process of their preparation and their use as dpp-iv inhibitors
06/07/2006EP1663975A1 Novel gamma secretase inhibitors
06/07/2006EP1663969A1 Crystalline forms of [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid
06/07/2006EP1663968A1 Process for the preparation of pure levetiracetam
06/07/2006EP1663967A1 PROCESS FOR CONVERTING a-ANGELICA LACTONE TO 5-METHYL-N-ALKYL -2-PYRROLIDONE USING ALKYL AMINES
06/07/2006EP1663962A2 Compositions and methods for the treatment of disease associated with trp-p8 expression
06/07/2006EP1663953A1 Inhibitors of histone deacetylase
06/07/2006EP1663232A1 1-(2-amino-benzoyl)-piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses
06/07/2006EP1663204A2 C-kit modulators and methods of use
06/07/2006EP1425029A4 Peptidomimetics of biologically active metallopeptides
06/07/2006EP1369416B1 Stable crystals of pyrrole compound
06/07/2006EP1311478B1 Novel (thio)urea compounds and the pharmaceutical compositions containing the same
06/07/2006EP1280847B1 Oligo/polysuccinimides, process for producing thereof and their use
06/07/2006CN1784457A Imide-linked maleimide and polymaleimide compounds
06/07/2006CN1784381A Method for crystallizing guanidinium salts
06/07/2006CN1781890A 糖皮质激素受体调制剂 Glucocorticoid receptor modulators
06/07/2006CN1258532C Compound of poly-amide macrocyclic polyamine and its preparation process and application
06/07/2006CN1258528C Method for the production of 2-pyrrolidone
06/07/2006CN1258362C Use of substituted acryloyl stallimycin derivatives in treatment of tumors associated with high levels of glutathione
06/06/2006US7057053 for treatment of arrhythmia and the production of analgesia and local anesthesia
06/06/2006US7057036 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
06/06/2006US7057035 reacting aryl/heteroaryl triflate/halide with carbon monoxide and N-hydroxysuccinimide in solvent in presence of palladium catalyst and base
06/06/2006US7056944 Pyrazole compositions useful as inhibitors of erk
06/06/2006US7056935 Administering to the animal suffering from neurological disorders an amide compound having an affinity for FKBP-type immunophilins
06/06/2006US7056915 Compounds useful as reversible inhibitors of cysteine proteases
06/06/2006US7056907 Mandelic acid derivatives and their use as thrombin inhibitors
06/06/2006CA2232913C Process for the preparation of azide derivatives
06/06/2006CA2136903C Acetic acid derivatives
06/01/2006WO2006056884A1 N- [ (3s)- pyrrolidin-3-yl]- benzamide derivatives as monoamine re-uptake inhibitors
06/01/2006WO2006056752A1 Phenoxyacetic acid derivatives useful for treating respiratory diseases
06/01/2006WO2006056696A2 2-alcoxy-3,4,5-trihydroxy-alkylamides, preparation thereof, compositions containing them and use thereof
06/01/2006WO2006056282A1 2,6-diethyl-4-methyl-phenyl-substituted tetramic acid derivatives
06/01/2006WO2006056281A1 2-alkoxy-6-alkyl-phenyl-substituted spirocyclic tetramic acid derivatives
06/01/2006WO2006056166A2 Method for the addition of amides ureas lactams and carbamates to alkynes
06/01/2006WO2005118537A3 Arylpiperazine derivatives as adrenergic receptor antagonists
06/01/2006WO2005034940A8 Dual alanyl aminopeptidase and dipeptidyl peptidase iv inhibitors for functionally influencing different cells and for treating immunological, inflammatory, neuronal and other diseases