Patents
Patents for C07C 311 - Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups (17,647)
11/1999
11/16/1999US5986102 Hydroxypropylamide peptidomimetics as inhibitors of aspartyl proteases
11/16/1999US5985900 Treating tumor growth, invasion or metastasis, osteoarthritis, rheumatoid arthritis, osteoporosis, periodontitis, gingivitis, chronic dermal wounds, corneal ulceration, degenerative skin disorders, multiple sclerosis, stroke, atherosclerosis,
11/16/1999US5985899 Selective thrombin inhibitors
11/16/1999US5985870 Sulfonylalkanoylamino hydroxyethylamino sulfonamide retroviral protease inhibitors
11/16/1999US5985838 Peptide analogs as irreversible interleukin-1β protease inhibitors
11/16/1999CA2010272C Benzenesulfonamides and a process for their preparation
11/11/1999WO1999057102A1 Substituted sulphonyl cyanamides, method for producing same and their use as medicament
11/11/1999WO1999057098A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999WO1999056765A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME
11/11/1999DE19820064A1 Substituierte Sulfonylcyanamide, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament Substituted Sulfonylcyanamide, processes for their preparation and their use as a medicament
11/11/1999CA2331863A1 Substituted sulphonyl cyanamides, method for producing same and their use as medicament
11/11/1999CA2329704A1 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999CA2327507A1 Succinamide inhibitors of interleukin-1.beta. converting enzyme
11/10/1999CN1234792A Nitric ester derivatives and use in treatment of urinary incontinence and other diseases
11/10/1999CN1234786A Nitrification process
11/10/1999CN1234396A Process for alkylation of hindered sulfamide
11/10/1999CN1234177A Amino-acetonitrile derivative, pesticides containing same for farm and gardening and use thereof
11/09/1999US5981758 Preparation of saccharincarbonyl halides
11/09/1999US5981595 Sulfonyl urea and carbamate ACAT inhibitors
11/09/1999US5981584 Useful in the manufacture of a medicament for inhibiting the aggregation of blood platelets, inhibiting angiogenesis, inhibiting osteoclast mediated bone resorption, preventing platelet thrombosis
11/04/1999WO1999055687A2 Hydroxypropylamide peptidomimetics as inhibitors of aspartyl proteases
11/04/1999WO1999055667A1 N-substituted aminotetralins as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders
11/04/1999WO1999055663A1 Inhibitors of impdh enzyme
11/04/1999WO1999055661A1 Aminomethyl-benzoic ester derivatives as tryptase inhibitors
11/04/1999WO1999055330A1 Ccr-3 receptor antagonists
11/04/1999WO1999031074A3 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
11/04/1999CA2329821A1 Ccr-3 receptor antagonists
11/03/1999EP0953565A2 Aminoacetonitrile derivative, agricultural and horticultural insecticide containing the same, and use thereof
11/02/1999US5977408 Preparation and use of β-sulfonamido hydroxamic acids as matrix metalloproteinase and TACE inhibitors
11/02/1999US5977390 Fluorinated diester melt additives for thermoplastic polymers
11/02/1999US5977384 Benzothiazolone derivatives
11/02/1999US5977178 Compounds with growth hormone releasing properties
11/02/1999US5977177 Substituted benzenesulfonylureas and-thioureas, processes for their preparation and use of pharmaceutical preparations based on these compounds, and medicaments containing them
11/02/1999US5977123 Oximether and acrylic acid derivatives and their use as fungicides
11/02/1999US5977122 Antiinflammatory, antiallergens, tumor necorsis factor inhibitor
11/02/1999US5977114 Selective thrombin inhibitors
11/02/1999US5977075 N-aroylamino acid amides as endothelin inhibitors
10/1999
10/28/1999WO1999054320A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999WO1999054294A1 New substituted amides, their production and their use
10/28/1999WO1999054293A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999WO1999054279A1 Substituted amino acids as erythropoietin mimetics
10/28/1999WO1999047497A3 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
10/28/1999CA2328720A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999CA2328435A1 New substituted amides, their production and their use
10/28/1999CA2328430A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999CA2236196A1 New improved ion exchange membranes, their methods of preparation and their uses
10/27/1999EP0952148A1 Cyclobutyl-aryloxyarylsulfonylamino hydroxamic acid derivatives
10/27/1999EP0951295A1 Methods and compositions useful for inhibition of angiogenesis
10/27/1999CN1233242A Substituted 2,4-diamino-1,3,5-triazines as herbicides
10/26/1999US5973167 Sulfonamide group, ether containing acid
10/26/1999US5973148 Combining an aromatic or heteroaromatic slufonyl chloride compound with an aromatic or heteroaromatic amine in presence of aromatic tertiary amine base and added catalytic amount of an n-arylsulfilimine compound to form n-arylarylsulfonamides
10/26/1999US5973111 Novel compounds that are capable of binding to the active site of interleukin-1b-converting enzyme (ice) and inhibiting activity of that enzyme; administering to treat inflammatory, autoimmune, and neurodegenerative diseases
10/26/1999US5973003 Treatment of thrombosis, stroke, myocardial infarction, inflammation and arteriosclerosis
10/26/1999US5972964 Aminomethylindans, -benzofurans and -benzothiophenes
10/21/1999WO1999053039A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/21/1999WO1999052878A1 Substituted phenyl pyridazinones
10/21/1999WO1999052862A1 Process for alkylating hindered sulfonamides useful in the production of matrix metalloproteinase inhibitors
10/21/1999WO1999044624A3 Pharmaceutical composition for prophylaxis and therapy of diseases associated with ocular fundus tissue cytopathy
10/21/1999WO1999026927A3 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
10/21/1999DE19818614A1 New benzamide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999DE19817461A1 New benzamide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999CA2327806A1 Substituted phenyl pyridazinones
10/21/1999CA2327282A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
10/20/1999EP0950656A1 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
10/20/1999EP0949916A1 Antitumor compositions and methods of treatment
10/20/1999EP0788476B1 Stilbene derivatives useful as cyclooxygenase-2 inhibitors
10/20/1999EP0778821B1 Ortho-substituted aromatic ether compounds and their use in pharmaceutical compositions for pain relief
10/20/1999CN1232443A Novel p-terphenyl compounds
10/20/1999CN1232023A Process for preparing hydroxamic acids
10/19/1999US5969204 Diazotizing substituted monoamino benzenes, then reacting products with substituted p-divinylbiphenyls
10/19/1999US5969182 Preparation of substituted guanidine derivatives
10/19/1999US5968982 2,2-Dichloroalkanecarboxylic acids, processes for their production and pharmaceutical agents containing these
10/19/1999US5968978 Antiarrythmia agents, antiischemic agents, inhibit proliferation of cells
10/19/1999US5968951 Benzenesulfonamide derivatives as bradykinin antagonists
10/19/1999US5968942 Inhibitors of hiv protease
10/19/1999US5968916 Agricultural insecticides, nematocides or miticides
10/14/1999WO1999051572A1 Sulfonamide derivatives
10/14/1999WO1999051569A1 Calcilytic compounds
10/14/1999WO1999051564A1 Propanolamine derivatives
10/14/1999CA2327290A1 Sulfonamide derivatives
10/14/1999CA2327279A1 Calcilytic compounds
10/13/1999EP0949245A1 Process for alkylating hindered sulfonamides
10/13/1999EP0949244A2 Process for preparing hydroxamic acids
10/13/1999EP0949238A1 Substituted propionyl derivatives
10/13/1999EP0948482A2 Method for producing trifluoroacetoacetic acid anilides
10/13/1999EP0948481A1 Aminobutyric acid fungicides
10/13/1999EP0948480A1 Sulphonyl compounds for use as linkers in solid phase and combinatorial synthesis
10/13/1999EP0783486B1 Novel prostaglandin synthase inhibitors
10/13/1999EP0763523B1 Naphthalene derivative
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999CN1045604C Process for the production of clavulanic acid salts
10/13/1999CN1045590C Hydrazine derivative and application of same
10/12/1999US5965741 Ortho-substituted aromatic ether compounds and their use in pharmaceutical compositions for pain relief
10/12/1999US5965592 Acyl compounds
10/12/1999US5965588 Sulfonylalkanoylamino hydroxyethylamimo sulfonamides useful as retroviral protease inhibitors
10/12/1999US5965579 Antagonists of the neurotensin receptors; increasing affinity for human neurotensin receptors
10/12/1999US5965121 Compounds and compositions for delivering active agents
10/10/1999CA2268680A1 Process for preparing hydroxamic acids
10/07/1999WO1999050237A1 Sulfonamide derivatives and drugs containing the same as the active ingredient
10/07/1999WO1999050205A2 Asymmetric grignard synthesis with cyclic 1,2 aminoalcohols