Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
02/2005
02/24/2005WO2005016264A2 Diamine derivatives of quinone and uses thereof
02/24/2005US20050043509 Peptoid compounds
02/24/2005US20050043371 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
02/24/2005US20050042274 Compounds and compositions for delivering active agents
02/23/2005EP1507783A1 Hydroxy diphosphines and their use in catalysis
02/23/2005EP1317421B1 2-amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
02/23/2005CN1585633A Phenethanolamine derivatives for treatment of respiratory diseases
02/22/2005US6858740 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
02/22/2005US6858602 Compounds for the treatment of metabolic disorders
02/22/2005US6858434 Using thin layer chromatography for rapid preparation and screening of lead structures for drug candidates; rational drug design
02/17/2005WO2005014534A1 Aryl and heteroaryl compounds, compositions, and methods of use
02/17/2005WO2005014533A2 Aryl and heteroaryl compounds, compositions, and methods of use
02/17/2005WO2005014532A1 Aryl and heteroaryl compounds, compositions and methods of use
02/17/2005WO2003099192A8 Bis-aromatic alkanols
02/17/2005US20050038081 amidation of a heteroary substituted oxoaminobenzoic acid with an amine; for treatment of psoriasis and rheumatoid arthritis using e.g. N-(3-dimethylaminophenyl)-3-(3-methoxybenzamido)-4-methylbenzamide
02/17/2005US20050038019 Hydroxy substituted amides for the treatment of alzheimer's disease
02/17/2005US20050038002 Bactericides; antitumor agents; moderators of gene expression; viricides; parasiticides; malaria therapy
02/17/2005US20050037953 Aspartyl protease inhibitor; antimalaria agents
02/17/2005US20050037934 Hair conditioner; flexibility; smoothness
02/17/2005CA2533173A1 Method for the production of cyclic phosphonic acid anhydrides
02/17/2005CA2531796A1 Aryl and heteroaryl compounds, compositions, and methods of use
02/16/2005EP1506168A2 Gelling agents
02/16/2005EP1506160A1 Production process of aminomethyl group-containing benzamide compound
02/16/2005EP1506158A2 Diamino-functional chalcones
02/16/2005EP1506157A2 Amino-functional chalcones
02/16/2005EP1339675B1 Ortho-substituted and meta-substituted bis-aryl compounds, method for the production thereof, their use as a medicament, and pharmaceutical preparations containing these compounds
02/16/2005EP1244617B1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
02/16/2005CN1189166C FC receptor modulators and uses thereof
02/15/2005US6855843 Antihistamines; rheumatic diseases; antidiabetic agents; inflammatory bowel disorders
02/15/2005US6855826 1,3-butadienes, perhydrobutadienes, ethylenes and ethanes as amino acid derivatives; hypotensive agents; antidiabetic agents and (pre)eclampsia treatments
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/10/2005WO2005012291A1 3-amino choman and 2-amino tetralin derivatives
02/10/2005WO2005012230A1 Amino acid diamides in non alpha position useful as adjuvants for the administration of active biological agents
02/10/2005WO2005011685A1 Aryl dicarboxamides
02/10/2005WO2003099338A3 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
02/10/2005US20050032873 3-Amino chroman and 2-amino tetralin derivatives
02/10/2005US20050032805 Antimicrobial biaryl compounds
02/10/2005US20050032794 For example, 2-Dimethylamino-N-(3-dimethylamino-1,4-dioxo-1,4-dihydro-naphthalen-2-yl)-N-methyl-acetamide; ability to function as gene expression modulators for genes found in cancer cells, especially genes involved in misregulated signal transduction pathways typical of cancers of colon and breast
02/10/2005US20050032790 For example, 1-(2-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4,4'-bispiperidine; for treatment of thrombosis, emphysema, cirrhosis; antiarthritic agents, anticancer agents, antihistamines
02/10/2005CA2533639A1 Amino acid diamides in non alpha position useful as adjuvants for the administration of active biological agents
02/10/2005CA2533363A1 3-amino choman and 2-amino tetralin derivatives
02/10/2005CA2529662A1 Aryl dicarboxamides
02/09/2005EP1503981A2 Substituted tetracycline compounds
02/09/2005CN1578768A Anthranilic acid amides and pharmaceutical use thereof
02/09/2005CN1578663A Inhibitors of histone deacetylase
02/09/2005CN1188420C Fungicides for preventing and curing full rot disease of plants
02/09/2005CN1188419C Fungicides for control of full-rot disease of plants
02/09/2005CN1188389C Benzamide derivatives for the treatment of diseases caused by cytokines
02/08/2005US6852755 This invention pertains to nitrogen mustard compounds (Formula (II)) and prodrugs therefor (Formula (I)), methods for their preparation, pharmaceutical compositions comprising such compounds, and the use of such compounds and
02/03/2005WO2005009944A1 Prodrugs of 9-aminomethyl tetracycline compounds
02/03/2005WO2005009943A2 Substituted tetracycline compounds
02/03/2005WO2005009940A1 Novel aminobenzophenone compounds
02/03/2005WO2004072102A3 Benzene acetamide compounds useful as serine protease inhibitors
02/03/2005WO2002096360A3 Single amino acid based compounds for counteracting effects of reactive oxygen species and free radicals
02/03/2005US20050027014 And other diseases such as Down's syndrome related to A beta peptide, a component of amyloid plaques; inhibitors of the beta-secretase enzyme
02/03/2005US20050026994 Treating proliferative diseases such as tumors; 4-[4-(2-Benzyloxycarbonylamino-3-methyl-butyrylamino)-3-hydroxy-2-(4-methoxy-benzylamino)-5-phenyl-pentanoylamino]4-(2-hydroxy-4-methoxy-benzylcarbamoyl)-butyric acid methyl ester for example
02/03/2005US20050026875 Treating bacterial, viral, or fungal infections, cancer, a lung injury, an eye disorder, neurological disorder or stroke
02/03/2005CA2744317A1 Substituted tetracycline compounds
02/03/2005CA2531728A1 Substituted tetracycline compounds
02/03/2005CA2530302A1 Novel aminobenzophenone compounds
02/02/2005EP1501801A1 2,6-quinolinyl and 2,6-naphthyl derivatives, processes for preparing them and their uses as vla-4 inhibitors
02/02/2005EP1501790A2 Novel sodium channel blockers
02/02/2005EP1501787A1 N-biphenylmethyl aminocycloalkanecarboxamide derivatives with a substiituent on the methyl useful as bradykinin antagonists
02/02/2005CN1575275A Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
02/02/2005CN1575273A 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor antagonists
02/01/2005US6849757 For example, Methyl 5-(((2S)-6-amino-2-((tert-butoxycarbonyl)amino)hexanoyl)amino)-4' -hydroxy(1,1'-biphenyl) -2-carboxylate for example; broadly claimed structure has an amido or carbamoyl substituted biphenyl skeleton
02/01/2005US6849743 Synthesis of clasto-lactacystin β-lactone and analogs thereof
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849615 13-substituted methacycline compounds
01/2005
01/27/2005US20050020689 Process and intermediates for the preparation of 3-(amino)-3-cyclobutylmethyl-2-hydroxy-propionamide or salts thereof
01/27/2005US20050020504 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
01/27/2005US20050020450 Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
01/26/2005EP1500643A1 Benzamide derivatives
01/26/2005EP1499898A2 Regulation of tnf-alpha
01/26/2005CN1569820A Process for synthesis of L-glutamine
01/25/2005US6846939 Minocycline compound substitued at 9-position by a group selected from nitro, alkyl, alkenyl, alkynyl, aryl, alkoxy, alkylthio, alkylsufinyl, alkylsulfonyl, amino, thionitroso, arylalkynyl or carbamate, urea, and sulfonamide
01/25/2005CA2231201C Toilet bowl cleaning tablet
01/20/2005WO2005004802A2 N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer's disease
01/20/2005US20050014925 Polyamic acid oligomer, polyimide oligomer, solution composition, and fiber-reinforced composite material
01/20/2005CA2529994A1 N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer's disease
01/20/2005CA2529739A1 Aspartyl protease inhibitors
01/19/2005EP1498428A1 Antibodies for detecting ecstasy-class analytes
01/19/2005EP1497260A1 Novel methoxybenzamide compounds for use in mch receptor related disorders
01/19/2005EP1497247A2 Mimics of acyl coenzyme-a, compositions thereof, and methods of cholesterol management and related uses
01/19/2005EP1496838A2 Substituted amides
01/19/2005EP1165493B1 Nitrogen mustard compounds and prodrugs therefor
01/19/2005CN1568312A Biphenylcarboxamides useful as lipid lowering agents
01/19/2005CN1185212C Salicylamide derivatives
01/19/2005CN1185211C Benzamide derivatives for the treatment of diseases resulted from cytokines
01/13/2005WO2005003080A1 Process for iohexol manufacture
01/13/2005US20050010060 Novel quinones as disease therapies
01/13/2005US20050009924 1,4-, 1,5- and 1,8-difunctionalized anthraquinones, useful for treating abnormal proliferation including cancer, for enhancing an anti-oxidation effect, human telomerase activity, and tissue engineering application, and for stem cell research
01/12/2005EP1496047A1 Method for producing enamines of acetoacetylated aromatic amines
01/12/2005EP1495034A2 Mimics of acyl coenzyme-a comprising pantolactone and pantothenic acid derivatives, compositions thereof, and methods of cholesterol management and related uses
01/12/2005EP1494997A1 Substituted aryl amides
01/12/2005EP1494642A1 Organosilicone derivatives of amino hydroxybenzophenones and their use as uv-a filters in cosmetic preparations
01/12/2005CN1564690A Tetracycline derivatives and methods of use thereof
01/11/2005US6841703 Polymerization of ethylenically unsaturated monomers with low dispersity
01/06/2005WO2005000794A1 Propionamide derivatives useful as androgen receptor modulators
01/06/2005WO2005000793A1 2-substituted cycloalkylcarboxylic acid derivative
1 ... 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 ... 162