Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
02/2012
02/02/2012WO2012014226A1 Process for preparation of lacosamide and some n-benzyl-propanamide intermediate derivatives
02/02/2012US20120029188 Substituted Aniline Derivatives
02/02/2012US20120029083 Polymorphic forms of aliskiren hemifumarate and process for preparation thereof
02/02/2012US20120029013 Derivatives of aminocyclobutane or aminocyclobutene, their method of preparation and their use as medical products
02/02/2012US20120028995 Novel compounds for medical use as peptidase effectors
02/02/2012US20120028928 Process for Isolating Tigecycline and Tigecycline Made Therefrom
02/02/2012US20120027844 Compounds, their syntheses, compositions, and methods to treat cancer
02/02/2012CA2805739A1 Drug-ligand conjugates, synthesis thereof, and intermediates thereto
02/01/2012CN1867581B Il-21衍生物 Il-21 derivatives
02/01/2012CN102341371A Bis aromatic compounds for use as lct4 synthase inhibitors
02/01/2012CN102341367A Method for producing halogen-substituted benzene dimethanol
02/01/2012CN102336681A Triiodobenzene compound contrast agent
02/01/2012CN102336680A Methods of preparing substituted tetracyclines with transition metal-based chemistries.
02/01/2012CN102336679A 7-substituted tetracycline compounds
02/01/2012CN102336676A New preparation method of dopexamine hydrochloride by ArCHR protection strategy
02/01/2012CN101445468B 对氨基苯甲酸拟二肽酯及其制备方法和应用 Ethanol intends dipeptide ester and preparation method and application
01/2012
01/31/2012US8106225 Catalytically reacting a 7(9)- arene tetracycline diazonium salt or an iodotetracycline and a reactive substituent precursor, e.g., (substituted) alkenes, vinyl monomers, aromatics, carbon monoxide; carboxylation, esterification, amidation carbonylation, cyanation; anhydriding; imidation; bactericides
01/31/2012CA2669849C Crystalline forms of (3s)-3-[n-(n'-(2-tert-butylphenyl)oxamyl)alaninyl]amino-5-(2',3',5',6'-tetrafluorophenoxy)-4-oxopentanoic acid
01/29/2012CA2746890A1 Novel compounds for medical use as peptidase effectors
01/26/2012WO2012010651A2 Method for the preparation of omega-amino-alkaneamides and omega-amino-alkanethioamides as well as intermediates of this method
01/26/2012WO2011109326A3 Crosslinking reagents, methods, and compositions for studying protein-protein interactions
01/26/2012US20120022263 3-aminoxalyl-aminobenzamide derivatives and insecticidal and miticidal agents containing same as active ingredient
01/26/2012US20120022230 Ionizable isotopic labeling reagents for relative quantification by mass spectrometry
01/26/2012US20120022086 Catecholamine derivatives for obesity and neurological disorders
01/26/2012US20120022025 Crystalline form c of tigecycline dihydrochloride and methods for its preparation
01/26/2012US20120021530 HETEROGENEOUS FOLDAMERS CONTAINING alpha, beta, and/or gamma-AMINO ACIDS
01/26/2012US20120021469 Amidases and methods of their use
01/26/2012US20120021044 Novel Cationic Lipid, A Preparation Method of the Same and A Delivery System Comprising the Same
01/25/2012EP2408735A1 Process for the preparation of triiodinated carboxylic aromatic derivatives
01/25/2012CN102333569A Amine or amino alcohols as glyt1 inhibitors
01/24/2012US8101591 9-aminoacyl tetracycline compounds and methods of use thereof
01/24/2012US8101590 9-aminocarbonylsubstituted derivatives of glycylcyclines
01/24/2012CA2435687C Omega-aminoalkylamides of r-2-aryl-propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells
01/19/2012WO2012009678A1 Therapeutically active compositions and their method of use
01/19/2012WO2012007644A1 Novel arylamide derivatives having antiandrogenic properties
01/19/2012US20120015992 Napthalene-Based Inhibitors of Anti-Apoptotic Proteins
01/19/2012CA2805669A1 Therapeutically active compositions and their methods of use
01/19/2012CA2804765A1 Novel arylamide derivatives having antiandrogenic properties
01/18/2012EP2407448A2 Processes and intermediates for preparing steric compounds
01/18/2012EP2406220A1 Bis aromatic compounds for use as ltc4 synthase inhibitors
01/18/2012EP2406213A1 Nitration of tetracyclines
01/18/2012CN102325748A Process for the preparation of triiodinated carboxylic aromatic derivatives
01/18/2012CN102320990A Method for recovering oxytetracycline from oxytetracycline hydrochloride waste liquid
01/18/2012CN102320989A Uvaria macrophylla bisamide derivative and preparation method and application thereof
01/18/2012CN102126986B Triiodobenzene compound and contrast medium with same
01/18/2012CN101531613B Aminopeptidase N inhibitor bestatin dino ester, synthesis and application thereof
01/17/2012US8097655 Methods for concomitant administration of colchicine and macrolide antibiotics
01/17/2012US8097654 Radiolabeled 3-[3-(benzoyl-amido)benzyloxy]aspartic acid derivative and method of producing the same
01/12/2012WO2011106574A9 Inhibitors for antiviral use
01/12/2012US20120010401 Method for manufacturing 1,5-benzodiazepine derivative
01/12/2012US20120010112 Acid-free quaternized nitrogen compounds and use thereof as additives in fuels and lubricants
01/11/2012EP2404897A1 Method for producing halogen-substituted benzene dimethanol
01/11/2012EP2404896A1 Cyclohexane derivative having npy y5 receptor antagonism
01/11/2012EP2404894A1 Mevalonic Acid Derivatives
01/11/2012CN101209976B Substituted tartaric acid derivatives and use thereof for preparing beta-secretase inhibitor
01/10/2012US8093298 Methods for concomitant administration of colchicine and macrolide antibiotics
01/10/2012US8093297 Methods for concomitant administration of colchicine and a second active agent
01/10/2012US8093296 Methods for concomitant administration of colchicine and macrolide antibiotics
01/10/2012CA2608180C Substituted acrylamide derivative and pharmaceutical composition comprising the same
01/05/2012WO2012001710A1 An improved process for the preparation of lacosamide
01/05/2012US20120004462 Intermediate compounds and their use in preparation of lacosamide
01/05/2012US20120004452 Intermediate compounds and their use in preparation of lacosamide
01/05/2012US20120004310 Non-peptide bdnf neurotrophin mimetics
01/05/2012US20120004243 Amide derivatives bearing a cyclopropylaminoacarbonyl substituent useful as cytokine inhibitors
01/04/2012CN102304075A Inhibitors of viral replication
01/04/2012CN102304056A 3-methyl-4-aryl-3-alkenyl-butyryl-pentafluoroaniline derivatives and preparation method thereof
01/04/2012CN101434559B Preparation of aceglutamide
01/03/2012US8088826 Tetrahydro-naphthalene derivatives
01/03/2012US8088763 e.g. N-[1-(2,6-dichloro-benzyl)-pyrrolidin-3-yl]-N'-[4-dimethylamino-4-(4-methyl-benzyl)-cyclohexyl]-succinamide; noradrenaline and serotonin reuptake ihibitor; opioid ORL-1 receptor ligand; analgesic, antidepressant, anxiolytic agent, neurodegenerative diseases
01/03/2012US8088762 Nitrosated nonsteroidal antiinflammatory compounds, compositions and methods of use
01/03/2012US8088755 11a, 12-derivatives of tetracycline compounds
01/03/2012CA2529464C Propionamide derivatives useful as androgen receptor modulators
12/2011
12/29/2011US20110319454 Derivatives of cycloalkyl- and cycloalkenyl-1,2-dicarboxylic acid compounds having formyl peptide receptor like-1 (fprl-1) agonist or antagonist activity
12/29/2011US20110319368 Once daily formulations of tetracyclines
12/29/2011US20110318771 Deuterium isobaric tag reagents for quantitative analysis
12/28/2011EP2399901A1 Intermediate for producing lacosamide and a process for its preparation and conversion to lacosamide
12/28/2011EP2399900A1 Geranyl compounds
12/28/2011EP2399899A1 Geranyl compounds
12/28/2011EP2399893A2 Compositions containing, methods involving, and uses of non-natural amino acids and polypeptides
12/28/2011EP2398558A1 Amine or amino alcohols as glyt1 inhibitors
12/28/2011CN102300840A (1s,2r)-米那普仑的合成方法 (1s, 2r) - synthesis method milnacipran
12/28/2011CN102295580A 一种制备2-氨基丁腈的工艺改进方法 2-amino-butyronitrile A process for preparing an improved method
12/28/2011CN102295576A 替加环素的晶型及其制备方法 Tigecycline crystal form and its preparation method
12/28/2011CN102295575A 一种动力学拆分2-氨基丁酰胺消旋体的方法 One kind of 2-amino-butanamide kinetic resolution method of racemic
12/28/2011CN102295574A 合成茶氨酸的方法 Theanine synthesis method
12/28/2011CN102295571A 甲醇或甲醛氨氧化合成酰胺的方法 Methanol or formaldehyde ammoxidation AMIDE method
12/28/2011CN101780381B 一种n-烷基天冬氨酰胺表面活性剂及其制备方法 One kind of n- alkyl aspartic acid amide surfactant and its preparation method
12/27/2011US8083973 Polychromic substances and their use
12/22/2011WO2011158249A1 Process for preparation of milnacipran intermediate and its use in preparation of pure milnacipran
12/22/2011WO2011158197A1 New cathepsin s protease inhibitors, useful in the treatment of e.g. autoimmune disorders, allergy and chronic pain conditions
12/22/2011WO2011084719A3 Soluble anion exchangers from hyperbranched macromolecules
12/22/2011US20110312964 Cysteine protease inhibitors
12/22/2011US20110312895 Dipeptide mimetics of ngf and bdnf neurotrophins
12/22/2011US20110312890 Acetylated amino acids as anti-platelet agents, nutritional and vitamin supplements
12/22/2011US20110312875 Peptidic compounds
12/22/2011US20110311813 Self-assembled nanostructures
12/22/2011CA2798150A1 New cathepsin s protease inhibitors, useful in the treatment of e.g. autoimmune disorders, allergy and chronic pain conditions
12/21/2011EP2396297A1 Androgen receptor modulating compounds, preparation and uses thereof
12/21/2011EP1483578B1 Artificial receptors, building blocks, and methods
12/21/2011CN102285899A 制备n-苯基吡唑-1-甲酰胺的方法 Preparation n- phenyl-pyrazol-1-carboxamide Method
1 ... 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 ... 162