Patents
Patents for C07C 229 - Compounds containing amino and carboxyl groups bound to the same carbon skeleton (21,416)
09/2002
09/25/2002EP1242589A2 Methods for producing enantiomerically pure alpha-substituted carboxylic acids
09/25/2002EP1242382A1 Tricyclic protein kinase inhibitors
09/25/2002EP1242069A2 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies
09/25/2002EP0975580B1 Contrast agent preparation
09/25/2002CN1371356A Enatiomerically-enriched compounds having photocleavable bond(s) and methods related thereto
09/24/2002US6455726 Starting materials for fungicides of lipopeptide type; isomer/impurity free
09/24/2002US6455572 Estrogen agonist/antagonist metabolites
09/24/2002US6455539 Autoimmune disease; antiinflammatory agents; antiproliferatory agents
09/24/2002US6455519 Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/19/2002WO2002072020A2 Novel anti-adhesive compounds and uses thereof
09/19/2002WO2002058680A3 Use of bicylic amino acids for preventing and treating visceral pain and gastrointestinal disorders
09/19/2002US20020133020 Efficient synthetic routes for the preparation of rhinovirus protease inhibitors and key intermediates
09/19/2002US20020132965 Stabilized monoaspartic acid esters and polyaspartic acid esters
09/19/2002US20020132849 2-Amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
09/19/2002US20020132796 Treatment or prevention of the diseases and conditions which respond to treatment by retinoids and or which in healthy mammals, including humans, are controlled by natural retinoic acid.
09/19/2002US20020131967 Such as melphalan and an anti-interleukin-6 receptor antibody, administering in synergistic amounts
09/19/2002CA2441174A1 Novel anti-adhesive compounds and uses thereof
09/18/2002EP1117633B1 Diaminocyclobutene-3,4-dione derivatives, their preparation and use
09/18/2002EP0823889B1 1,3-propane diol derivatives as bioactive compounds
09/18/2002EP0804427B1 Lta4 hydrolase inhibitors
09/18/2002CN1370151A Process for preparing 2-amino-4-(4-fluorophenyl)-6-alkylpyrimidine-5-carboxylate
09/18/2002CN1370143A Propanoic acid derivatives that inhibit binding of integrins to their receptors
09/18/2002CN1369496A Use of compound with structure similar to L-phenylalanine as medicine to treat skin diseases
09/18/2002CN1091097C Process for preparing N-substuted glacinic acids or glycinic esters
09/18/2002CN1090934C Prepn. of salts of pharmaceutical active substances which have acidic groups
09/17/2002US6452044 Benzenedicarboxylic acid derivatives
09/17/2002US6452030 Betaine compound and process for production thereof
09/17/2002US6452013 For treating conditions which are related to impairment of gastric emptying
09/17/2002US6451972 Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors
09/17/2002US6451858 Certain 5-alkyl-2-arylaminophenylacetic acids and derivatives
09/17/2002US6451854 α-amino acid phenyl ester derivatives
09/17/2002US6451830 Use of substituted N,N-disubstituted non-fused heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/17/2002US6451823 Use of substituted N-phenoxy-N-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
09/17/2002US6451543 Lipid matrix-assisted chemical ligation and synthesis of membrane polypeptides
09/17/2002CA2278878C Very large scale immobilized peptide synthesis
09/12/2002WO2002070510A2 Amino dicarboxylic acid derivatives with pharmaceutical properties
09/12/2002WO2002070462A1 Substituted amino dicarboxylic acid derivatives
09/12/2002WO2002070461A1 Side-chain halogenated amino carboxylic acid derivatives as medicaments for treating cardiovascular diseases
09/12/2002WO2002070460A1 Halogen-substituted amino dicarboxylic acid derivatives as medicaments for treating cardiovascular diseases
09/12/2002WO2002070459A1 Novel amino dicarboxylic acid derivatives
09/12/2002WO2002070458A1 Low colour nitrogen-containing surfactants
09/12/2002WO2002055480A3 6-substituted indanoyl amino acid conjugates as mimics to the biological activity of coronatine
09/12/2002WO2002050077A3 Triazolopyrimidines
09/12/2002US20020128510 Antiarthritic agents; rheumatic diseases; osteoarthritis; inhibition of the inducible nitric oxide synthase - induced after activation of vascular smooth muscle, macrophages, endothelial cells by enotoxin and cytokines
09/12/2002US20020127202 Compounds and compositions for delivering active agents
09/12/2002DE10110750A1 Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften Novel Aminodicarbonsäurederivate with pharmaceutical properties
09/12/2002DE10110749A1 Substituierte Aminodicarbonsäurederivate Substituted Aminodicarbonsäurederivate
09/12/2002DE10107528A1 Verfahren zur Herstellung der Enantiomere der 2-substituierten beta-Aminosäuren Process for preparing the enantiomers of the 2-substituted beta amino acids
09/12/2002CA2439945A1 Novel halogen-substituted aminodicarboxylic acid derivatives
09/12/2002CA2439939A1 Novel aminodicarboxylic acid derivatives
09/12/2002CA2439759A1 Substituted amino dicarboxylic acid derivatives
09/12/2002CA2439647A1 Side-chain-halogenated aminodicarboxylic acid derivatives as medicaments for treatment of cardiovascular disorders
09/11/2002EP1237848A1 Process for the preparation of 3-amino-3-cyclopropylpropanoate esters
09/11/2002EP1237847A1 Method for the stereoselective synthesis of cyclic amino acids
09/11/2002EP1237846A1 Preparation of 3-amino-3-cyclopropylpropanoate esters
09/11/2002EP1237845A1 Aminobenzophenones as inhibitors of il-1beta and tnf-alpha
09/11/2002EP0877561B1 Composition and method for producing a salty taste
09/11/2002EP0813529B1 Arginine analogues having nitric oxide synthase inhibitor activity
09/11/2002EP0748799B1 Process for producing 5,7-dichloro-4-hydroxyquinoline
09/11/2002CN1368951A Process for preparing betaines
09/11/2002CN1368498A Preparation method of o-chloromethyl phenyl glyoxalic acid derivative
09/11/2002CN1368497A Preparation method of o-chloromethyl phenyl glyoxalic acid derivative
09/11/2002CN1090637C Cross-link cinnamic acid derivative and its preparation method
09/10/2002US6448443 Synthesis of combinatorial libraries of compounds reminiscent of natural products
09/10/2002US6448442 Contrast media
09/10/2002US6448295 Treating cardiovascular disease; atherosclerosis, dyslipidema hypercholesterolaemia; decreasing concentrations of low density lipoprotein and raising level of high density lipoprotein
09/10/2002US6448293 Treatment or prevention of a disorder in which the regulation of monoamine transporter function is implicated, such as premature ejaculation.
09/06/2002WO2002068428A1 Method of preparing cephalosporins using 4-hydroxyphenylglycine derivatives
09/06/2002WO2002068393A1 Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors
09/06/2002WO2002068380A1 Synthetic excitatory amino acids
09/06/2002CA2434666A1 Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors
09/05/2002US20020123648 Containing an acid radical in such amount that the solubility of lysine therein has been increased; storage stability
09/05/2002DE10109861A1 Neuartige seitenkettenhalogenierte Aminodicarbonsäurederivate Novel side-chain halogenated Aminodicarbonsäurederivate
09/05/2002DE10109859A1 Neuartige Aminodicarbonsäurederivate Novel Aminodicarbonsäurederivate
09/05/2002DE10109858A1 Neuartige halogensubstituierte Aminodicarbonsäurederivate Novel halogen-substituted Aminodicarbonsäurederivate
09/04/2002EP1235792A1 Preparation of [4s-(4alpha,7alpha,10abeta)]-4-amino-octahydro-5-oxo-7h-pyrido 2,1-b] 1,3]thiazepine-7-carboxylic acid, methyl ester and salts thereof via novel disulfides
09/04/2002EP1235788A1 Process for the preparation of arylethanolamine derivatives having an anti-obesity and anti-diabetic properties
09/04/2002EP1235786A2 Method for the preparation of enantiomerically enriched compounds
09/04/2002EP0934278B1 Bis(acridinecarboxamide) and bis(phenazinecarboxamide) as antitumour agents
09/04/2002EP0832074B1 Amino acid derivatives of substituted quinoxaline 2,3-dione derivatives as glutamate receptor antagonists
09/04/2002CN1367775A Cubane derivatives as metabotropic glutamate receptor antagonists and process for their preparation
09/03/2002US6444701 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
08/2002
08/29/2002WO2002066456A2 Thiophene substituted amine derivatives as glyt-1 inhibitors
08/29/2002WO2002066418A2 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor
08/29/2002WO2002066417A1 Method for the production of the enantiomers of 2-substituted beta amino acids
08/29/2002WO2001012584A3 Pharmaceutical compounds
08/29/2002WO2000068188A9 Propanoic acid derivatives that inhibit the binding of integrins to their receptors
08/29/2002WO2000066104A9 Ace-2 inhibiting compounds and methods of use thereof
08/29/2002US20020120148 Benzocycloheptenylamino derivatives; treatment of pollakiuria or urinary incontinence
08/29/2002US20020120136 Method of preparing cephalosporins using 4-hydroxyphenylglycine derivatives
08/29/2002US20020120105 Polarization switching to control crystal form
08/29/2002US20020120096 Capable of stably fixing a water-soluble polymer onto a surface structure by taking advantage of intermolecular interaction, thereby enabling the water-soluble polymer to be carried thereon without giving any damage
08/29/2002US20020120011 Substituted N, N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity
08/29/2002US20020120009 Compounds and compositions for delivering active agents
08/29/2002US20020119965 Nitriloxy derivatives of (R) and (S)-carnitine
08/29/2002US20020119953 Sickle cell anemia
08/29/2002US20020119910 Drug delivery
08/29/2002CA2438367A1 Thiophene substituted amine derivatives as glyt-1 inhibitors
08/28/2002EP1097126A4 Crystalline salts of dodecyl 2-(n,n-dimethylamino)-propionate
08/28/2002EP1045828B1 Method for producing highly pure tetrasodium salt of ethylenediaminetetraacetic acid