Patents for A61P 27 - Drugs for disorders of the senses (53,017)
02/1993
02/18/1993WO1993003018A1 Compounds having angiotensine ii antagonistic activity
02/18/1993WO1992020651A3 N-(heteroaryl)-imidazolyl-alkenoic acids
02/18/1993CA2114621A1 Compounds having angiotensine ii antagonistic activity
02/17/1993EP0527534A1 Quinoline and azaquinoline angiotensin II antagonists
02/16/1993US5187179 Angiotensin II antagonists incorporating a substituted imidazo [1,2-b][1,2,4]triazole
02/16/1993US5187159 Angiotensin II antagonists incorporating a substituted 1,3-benzodioxole or 1,3-benzodithiole
02/16/1993CA2076057A1 N-acyl-n-heterocyclylalkylamino acids, processes, compositions and use
02/14/1993CA2075652A1 Quinoline and azaquinoline angiotensin ii antagonists incorporating a substituted benzyl element
02/10/1993EP0527042A2 3-deoxy-mannosamine derivatives and process for their preparation
02/10/1993EP0526865A1 Spongy material consisting essentially of hyaluronic acid or its derivatives, and its use in microsurgery
02/10/1993EP0526695A1 Stabilized PVP-I solutions
02/10/1993CN1019890C Process for preparation of 4-heterocyclic sulfonyl (or thio-) propyl-oxy-2-hydroxy-3-propyl-hypnone derivatives
02/09/1993US5185372 Sealed container of solution of retinol palmitate, boric acid, nonionic surfactant, chelating agent, preservative; adjusted pH; topical treatment of dry eye syndrome
02/09/1993US5185351 Hypotensive agents; for treatment of congestive heart failure, renal failure and glaucoma
02/09/1993US5185331 Triazolobenzodiazepines
02/07/1993CA2075336A1 3-deoxy-mannosamine derivatives and process for their preparation
02/06/1993CA2075340A1 Spongy material consisting essentially of hyaluronic acid or its derivatives, and its use in microsurgery
02/03/1993EP0526004A1 Pyrazolopyrimidinone antianginal agents
02/03/1993EP0526001A1 Substituted triazolinones
02/03/1993EP0525475A2 A beta-blocker and carbachol containing antiglaucoma composition
02/03/1993EP0525129A1 Substituted benzimidazoles
02/03/1993EP0525054A1 Modified heparin binding growth factors
02/03/1993EP0386076B1 Phosphoryled derivatives of cardiodilatine/anf peptides
02/03/1993EP0349545B1 New cardiodilatin fragment, process for preparing same and use thereof
02/02/1993CA1313371C Fused azepinone and azocinone derivatives, processes for their preparation, agents containing them and their use, and intermediates in their preparation
01/1993
01/27/1993EP0524696A1 Oral compositions containing dapiprazole
01/27/1993CN1068329A Pyrazolopyrimidinone antianginal agents
01/26/1993US5182288 Substituted n-biphenylyl lactams
01/26/1993US5182102 Mixture of a miotic and a beta-blocker, reduction of aqueous humor formation and improved outflow of humor
01/21/1993WO1993001177A1 Substituted triazolinones
01/20/1993EP0524004A1 Decahydro-8H-isoquino[2,1-g][1,6]naphthyridine and decahydrobenzo[a]pyrrolo[2,3-e]quinolizine derivatives
01/20/1993EP0523846A2 1,4-Benzodiazepines with 5-membered heterocyclic rings
01/20/1993EP0523845A2 New benzodiazepine analogs
01/20/1993EP0523141A1 Substituted pyrazoles, isoxazoles and isothiazoles
01/19/1993US5180837 Pilosinine derivatives
01/19/1993CA1312870C Alkanesulfonamides as antiglaucoma agents
01/18/1993CA2074038A1 Decahydro-8h-isoquino[2,1-g][1,6]naphthyridine and decahydrobenzo[a] pyrrol[2,3-e]quinolizine derivatives
01/13/1993EP0522226A1 Eyedrop solution for the treatment of ocular hypertension containing ketauserin
01/13/1993EP0522038A1 Substituted pyrimidines, pyrimidinones and pyridopyrimidines
01/13/1993EP0522000A1 5-lipoxygenase inhibitors
01/13/1993EP0521986A1 Topically active ocular gem-diacylthiadiazole sulfonamide carbonic anhydrase inhibitors
01/13/1993CA2072726A1 Anti-glaucoma compositions
01/12/1993US5179110 Adrenergic stimulants; antiulcer agents, bronchodilators, treatment of diarrhea, glaucoma, osteoporisis, prostate, diabetes, migraine
01/07/1993WO1993000341A1 4-(1-h-pyrrol-1-yl)imidazoles with angiotensin ii antagonist activity
01/07/1993WO1993000329A1 Chemical process
01/07/1993EP0521799A1 Ophthalmic compositions
01/07/1993EP0521009A1 5-trans-prostaglandin-2-alpha as an ocular hypotensive agent
01/06/1993CA2073141A1 Ophthalmic compositions
01/06/1993CA2072676A1 Azabicyclic compounds, pharmaceutical compositions containing them and their use in therapy
01/05/1993US5177074 Angiotensin ii antagonists incorporating a substituted thiophene or furan
01/05/1993US5177071 Tranquilizers
01/05/1993CA1312336C Aromatic polycyclic derivatives, their preparation process and their use in human and veterinary medicine as well as in cosmetics
01/04/1993CA2072775A1 Substituted triazolinones
12/1992
12/29/1992US5175166 Cognition activators
12/29/1992US5175164 Angiotensin ii antagonists incorporating a substituted indole or dihydroindole
12/29/1992US5175161 Occular hypotensive agents
12/29/1992CA1312083C Hydantoin derivatives
12/23/1992WO1992022569A1 Peptides with tachykinin antagonist activity
12/23/1992WO1992022300A1 Ocular compositions containing steroids and their use in treating glaucoma
12/23/1992EP0519831A1 N-Substituted heterocyclic derivatives, their preparation, and pharmaceutical compositions containing them
12/23/1992EP0519678A2 1,4-Benzodiazepines with 6-membered heterocyclic rings
12/23/1992CN1019544B Pharmaceutical composition for piperidinoalkanol derivatives
12/23/1992CA2111699A1 Ocular compositions containing steroids and their use for the glaucoma treatment
12/22/1992US5173496 Antiinflammatory agents
12/22/1992CA1311757C Acetylenes disubstituted with a heteroaromatic group and a tetralin group having retinoid like activity
12/22/1992CA1311754C Thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same
12/18/1992CA2071180A1 1,4-benzodiazepines with 6-membered heterocyclic rings
12/16/1992EP0518767A2 Derivatives of amide analogs of certain methano bridged quinolizines
12/16/1992EP0518722A1 Dithiane substituted retinoides, their use, process of their preparation, cosmetic and pharmaceutical compositions containing them and their use in therapeutics
12/16/1992EP0518676A2 Cyclic renin inhibitors
12/16/1992EP0518675A2 Cyclic renin inhibitors
12/16/1992EP0518672A2 Cyclic renin inhibitors
12/16/1992EP0517984A1 Derivatives of amide analogs of certain methano bridged quinolizines
12/16/1992EP0517812A1 Angiotensin ii antagonists incorporating a substituted benzyl element
12/16/1992EP0517789A1 Inhibitor of proliferation of endothelial cells.
12/16/1992CN1019490B Method for producing 3-(1h-tetrazol-5-yl) thieno 2,3-dlpyrimidin-4(3h)-ones
12/15/1992CA2071181A1 Benzodiazepine analogs
12/15/1992CA2071092A1 1,4-benzodiazepines with 5-membered heterocyclic rings
12/15/1992CA1311477C 1-hydroxy-5-oxo-5h-pyrido¬3,2-a|phenoxazine -3-carboxylic acid esters
12/12/1992CA2070983A1 Cyclic renin inhibitors
12/12/1992CA2070978A1 Cyclic renin inhibitors
12/12/1992CA2070972A1 Cyclic renin inhibitors
12/10/1992WO1992021360A1 Substituted n-carboxyalkylpeptidyl derivatives as antidegenerative active agents
12/10/1992CA2102890A1 Substituted n-carboxyalkylpeptidyl derivatives as antidegenerative active agents
12/09/1992EP0517484A2 Fermentation analogs of virginiamycin M1
12/09/1992EP0517357A1 Angiotensin II antagonists incorporating a substituted indole or dihydroindole
12/09/1992EP0517160A1 Extended-release ophthalmic preparations
12/09/1992EP0516685A1 Artificial tears
12/09/1992CN1066781A Ophthalmic compositions comprising combinations of carbonic anhydrase inhibitor and beta-adrenergic antagonist
12/08/1992US5169847 Aqueous solutions of piroxicam, sodium glycinecarboxylate, additives, for eye drops
12/06/1992CA2065078A1 Angiotensin ii antagonists incorporating a substituted indole or dihydroindole
12/04/1992CA2070242A1 Fermentation analogs of virginiamycin m1
12/02/1992EP0516392A2 Naphthyridine derivatives as angiotensin II inhibitors
12/02/1992EP0515548A1 Imidazole angiotensin ii antagonists incorporating a substituted benzyl element
12/02/1992EP0515535A1 Angiotensin ii antagonists incorporating a substituted benzyl element
12/02/1992CN1066654A Benzofuran derivatives
12/02/1992CN1019299B 1-hydroxy-5-oxo-5h-pyrido(3,2-a) phenoxazine-3-carboxylic acid esters
12/01/1992CA2068946A1 Heterocyclic derivatives
11/1992
11/30/1992WO1992021641A1 Dihydroxyindanone tyrosine kinase inhibitors
11/30/1992CA2109515A1 Dihydroxyindanone tyrosine kinase inhibitors