Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
07/1981
07/08/1981EP0031753A1 2-(4-Piperidyl)-1-(4-quinolyl)-ethanone derivatives, intermediates in and process for their preparation, and their use as medicines
07/08/1981EP0031727A2 Medicinal compositions comprising as an active ingredient substituted 1,4-benzoquinones
07/08/1981EP0031722A1 Water soluble guanidine derivatives of polyene macrolides and the esters thereof, processes for their preparation and pharmaceutical compositions containing them
07/08/1981EP0031708A2 Cephalosporin derivatives, processes for their manufacture, pharmaceutical compositions containing them and intermediates therefor
07/08/1981EP0031699A1 Benzimidazoline salts, their preparation and compositions containing them
07/08/1981EP0031653A1 N-Substituted alpha-amino acids, processes for making them and pharmaceutical compositions containing them
07/08/1981EP0031603A1 Pharmaceutical composition of matter
07/08/1981EP0031591A1 2,2-dimethyl-3-oxoandrosta-4,6-dien-17S-spiro-5'-(2'-oxo-3'-methyloxazolidin), process for its preparation and medicines containing this compound
07/08/1981EP0031584A2 2-Substituted-aminopropene- and propanenitrile compounds and antimicrobial and pharmaceutical, anti-inflammatory compositions
07/08/1981EP0031563A1 Nitrothiazolines, their preparation and pharmaceutical formulations containing them
07/08/1981EP0031509A1 Penem derivatives
07/08/1981EP0031473A1 Process for preparing 2-((alkoxycarbonyl)-amino)-5-(alkylthio)-1H-benzimidazoles
07/08/1981EP0031456A1 Substituted 4-amino-2,6-diaryl-tetrahydrothiopyranes, their acid-addition salts, processes for their preparation and pharmaceutical compositions
07/08/1981EP0031429A1 2-(N-(2-Fluoro-6-bromophenyl)-N-(thiemyl-2-methyl)-amino)-2-imidazoline, its addition salts, pharmaceutical compositions containing them and processes for their preparation
07/08/1981EP0031426A1 7-Oxo-PGI2 derivatives, process for their preparation and pharmaceutical compositions containing these compounds
07/08/1981EP0031407A1 Substituted 3,6 bis-(aminoalkoxy)acridines, and a process for their preparation
07/08/1981EP0031353A1 Use of perfluorocarbon as burn treatment.
07/07/1981US4277602 Eukalemic saluretic agents useful in treatment of edema and hypertension
07/07/1981US4277601 Alcoholysis of corresponding 3-n-protected carbamoyloxymethyl compound in anhydrous solvent in presence of basic catalyst
07/07/1981US4277501 Para-nitrophenylalkylamines and pharmaceutical compositions
07/07/1981US4277498 Derivatives of glycinamide as antidepressants
07/07/1981US4277497 And salts with amino acids
07/07/1981US4277495 Fluorene 9-aminoalkyl-9-carboxylic acids or esters
07/07/1981US4277492 Novel 4-bis((Phenylmethyl)amino)-benzenesulfonic acids possessing antiviral activity
07/07/1981US4277491 Hypotensive, vasodilatory, anti-aggregating, luteolytic, cytoprotective
07/07/1981US4277489 1(p-Chlorobenzoyl)-5-methoxy-2-methyl indole-3-acetic acid-3-oxo-isobenzofuranyl ester and pharmaceutical use thereof
07/07/1981US4277488 Water-soluble biotin-containing preparation
07/07/1981US4277487 Substituted 2-phenylamino-2-imidazolines as bradycardiacs
07/07/1981US4277486 1-[(Substituted-naphthyl)ethyl]-imidazole derivatives
07/07/1981US4277483 1.4-Dihydropyridine-derivatives with antihypertensive activity
07/07/1981US4277481 Organic compounds
07/07/1981US4277480 Tetrahydroindoloisoquinolines
07/07/1981US4277479 Tetrazolylalkoxycarbostyril derivatives and pharmaceutical compositions containing them
07/07/1981US4277478 Antibiotic and use thereof
07/07/1981US4277475 Contraceptive methods employing 1-substituted imidazole derivatives
07/07/1981US4277474 Dermatitis, rhinitis, asthma
07/07/1981US4277473 Viricides with fewer side effects on central nervous system
07/07/1981US4277472 3,6-Disubstituted-5,7-(lower alkano)-5,6,7,8-tetrahydropyrido(4,3-C)pyridazines; their intermediates, preparation, antihypertensive use and compositions
07/07/1981US4277470 Antidepressants
07/07/1981US4277468 Contraceptives, progestational activity
07/07/1981US4277467 Anthelmintics, larvicides
07/07/1981US4277461 Vaginal contraceptive
07/07/1981US4277401 Total synthesis of 1RS,4SR,5RS-4-(4,8-dimethyl)-5-hydroxy-7-nonen-1-yl)-4-methyl-3,8-dioxabicyclo[3.2.1]octane-1-acetic acid
07/07/1981US4276890 Tobacco smoking inhibitor
07/07/1981CA1104578A1 Compound, 4-carboxyphthalato(1,2-diaminocyclohexane)- platinum(ii) and alkali metal salts thereof and its use in alleviating murine leukemia
07/07/1981CA1104574A1 Antirhinovirus agents
07/07/1981CA1104572A1 2-benzylpyrrolidines, process for their preparation, and medicaments containing them
07/07/1981CA1104571A1 Mercaptoalkylsulfonyl proline derivatives and related compounds
07/07/1981CA1104567A1 Cycloalkyltriazoles and process for obtaining same
07/07/1981CA1104566A1 Process for the manufacture of azatetracyclic compounds
07/07/1981CA1104562A1 Cephalosporins, processes for their preparation and their use as medicaments
07/07/1981CA1104561A1 7-¬(sulfomethyl)phenyl| acetamidocephalosporin derivatives
07/07/1981CA1104560A1 Pyrrole cephalosporin derivatives
07/01/1981EP0031297A2 2,5 dioxo pyrrolidin compounds, process for their preparation and their use as microbicides
07/01/1981EP0031285A2 Immuno-stimulating preparations based on ribosomal RNA of Klebsiella pneumoniae and process for the preparation of these RNA
07/01/1981EP0031266A1 1-Amino-2-propanol derivatives, process for their preparation and their therapeutic use
07/01/1981EP0031234A1 Analgesic composition
07/01/1981EP0031219A1 Aniline derivatives
07/01/1981EP0031184A1 Process for the preparation of 4-(2-(dimethylamino)-ethoxy)-2-methyl-5-(1-methylethyl)-phenol esters and their salts
07/01/1981EP0031128A1 (E)-5-(2-halogenovinyl)-arabinofuranosyluracil, process for preparation thereof, and uses thereof
07/01/1981EP0031115A1 New pyrrolobenzotriazepines, their production and pharmaceutical compositions containing them
07/01/1981EP0031104A1 Thiazolidine compounds, processes for their preparation and pharmaceutical compositions containing them
07/01/1981EP0031088A1 Benzene-sulfonyl ureas, processes for their preparation, pharmaceutical compositions based on these compounds and their use
07/01/1981EP0031080A1 2-Acylaminomethyl-1,4-benzodiazepines and their salts, as well as a process for their preparation and pharmaceutical compositions containing these compounds
07/01/1981EP0031058A1 Sulfonyl ureas, processes for their preparation and pharmaceutical compositions containing these compounds
06/1981
06/30/1981US4276421 Histamine antagonists, antiulcer agents
06/30/1981US4276307 N-Phenethylaminopropiophenones as lipogenesis inhibitors
06/30/1981US4276304 Antidiabetic, anticoagulants
06/30/1981US4276299 1-(3-Bromo-isoxazol-5-yl)-2-tert.butylaminoethanol
06/30/1981US4276297 Pyridylaminotriazole therapeutic agents
06/30/1981US4276293 Cardiotonic agents
06/30/1981US4276289 Antitumor glycosides, their preparation and use
06/30/1981US4276285 Synergistic bactericides
06/30/1981US4276284 Corneal and stomach ulcers, rheumatoid arthritis
06/30/1981US4276280 Radiolabeled derivatives of folic acid
06/30/1981CA1104158A1 Antiarrhythmic n,n'-bis(phenylcarbamoyl- methyl)amidines
06/30/1981CA1104156A1 Analogues of bestatin
06/30/1981CA1104144A1 Dibenzothiophenes derivatives
06/30/1981CA1104142A1 Anthelmintic benzimidazol-carbamates
06/30/1981CA1104141A1 Lower alkyl 2-tri-(lower) alkylsilyl-acetylene-n- carbethoxyglycinates and process for using same
06/30/1981CA1104139A1 Antibacterial compounds
06/30/1981CA1104137A1 N-vinyl-3-hydroxy-pyrid-2-thione compounds
06/30/1981CA1104136A1 ¬1,2,3,4-tetrahydro-9h-pyrrolo¬3,4-b|quinoline- 9-one derivatives|
06/30/1981CA1104133A1 Nitroimidazoles and process for the preparation thereof
06/30/1981CA1104132A1 Process for the preparation of therapeutically useful 3,4,5-trimethoxy-benzene derivatives
06/30/1981CA1104131A1 4-desoxy-thiazolo-¬5,4-c|rifamycin derivatives, a process for preparing them and their use as antimicrobial agents
06/30/1981CA1104130A1 N-substituted carboxylic acid amides
06/30/1981CA1104126A1 Method for producing derivatives of penicillanic acid
06/30/1981CA1104124A1 Derivatives of 9-fluoroprednisolone
06/30/1981CA1104059A1 Carboxyalkanoyl derivatives of proline, pipecolic acid and azetidine-2-carboxylic acid
06/30/1981CA1104058A1 Endontic formula for treatment of root canal
06/25/1981WO1981001710A1 Mono and bis piperidinium androstanes derivatives
06/25/1981WO1981001653A1 Sedative drug
06/24/1981EP0030916A1 Azatetracyclic carbonitriles
06/24/1981EP0030861A2 Isoquinoline acetic acids and pharmaceutical compositions thereof
06/24/1981EP0030795A2 Quinoxaline derivatives, processes therefor, pharmaceutical compositions, and benzene derivatives
06/24/1981EP0030749A1 Carboximidamide derivatives, a process for preparing them and pharmaceutical preparations containing same
06/24/1981EP0030734A1 Tyrosine derivatives, a process for preparing the same and a pharmaceutical composition containing the same for treating hypertension
06/24/1981EP0030719A1 Antibiotic PA-39504-X1 and its salts, process for its production and pharmaceutical compositions
06/24/1981EP0030688A2 Piperidine derivatives of 3-hydroxy-thiophene-2-carboxylic acid esters, their preparation, and pharmaceutical preparations containing them