Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
05/2006
05/11/2006US20060100254 Thiazolyl-dihydro-indazole
05/11/2006US20060100253 Novel compounds for the treatment of neurological disorders
05/11/2006US20060100252 Beta 3 adrenergic receptor agonists; pollakiuria or urinary incontinence; antiulcer, overactive bladder, pancreatitis, obesity, diabetes, insulin resistance, hypertriglyceridemia, hypercholesterolemia, tocolytic agents; 4'-[2-(2-hydroxy-2-phenylethyl]amino]ethyl]-4-biphenylyl]acetic acid
05/11/2006US20060100251 Substituted phenylalkanoic acids
05/11/2006US20060100249 Pharmaceutical compositions comprising dihydropyridinone compounds and an immunoregulatory or an antiinflammatory agent and their uses
05/11/2006US20060100248 alleviating vision defects, multiple sclerosis, neurodegenerative diseases, stroke, spinal cord injury, Alzheimer's disease, Parkinson's disease or pain, comprising administering sodium channel modulators comprising pyrazole or indazole derivatives, such as 3-(5'-Hydroxymethyl-2'-furyl)-1-benzylindazole
05/11/2006US20060100247 Treatment of diabetes with thiazolidinedione and metformin
05/11/2006US20060100246 Synthesis of I kappa B kinase beta inhibitors that are 2-amino-4,6-disubstituted nicotinic acid ester analogs, by reacting an aryl ketone, an aldehyde and a cyanoacetate with an ammonium salt
05/11/2006US20060100245 Substituted biphenyl-4-carboxylic acid arylamide analogues
05/11/2006US20060100244 Such as (3-chloro-4-fluorophenyl)(4-fluoro-4-{[(5-hydoxypyridin-2-ylmethyl)amino]methyl}piperidin-1-yl)methanone; serotonin receptor agonists; for treating depression, pain, and substance abuse
05/11/2006US20060100243 Methylphenidate analogs and methods of use thereof
05/11/2006US20060100242 4-(2-Phenylsulfanyl-phenyl)-piperidine derivates as serotonin reuptake inhibitors
05/11/2006US20060100241 Method for enhancing mutant protein activity
05/11/2006US20060100240 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
05/11/2006US20060100239 Method for producing optically active amines
05/11/2006US20060100238 4',7-Dihydroxyisoflavanone (phenyl)hydrazone; 4,7-Dihydroxyisoflavanone(4,7-dihydroxyisoflavanone)hydrazone; anticarcinogenic and antiinflammatory agents; cyclooxygenase inhibitor
05/11/2006US20060100237 Excitatory amino acid receptor antagonists
05/11/2006US20060100236 5-HT4 receptor agonist compounds
05/11/2006US20060100235 Pharmaceutical use of substituted 1,2,4-triazoles
05/11/2006US20060100234 Gastric protection and gastric acid secretion-inhibitors; antiulcer agents; acid reflux, Zollinger-Ellison syndrome, heartburn and peptic ulcer bleeding; e.g. methyl 8-(2,3-dihydro-2-hydroxy-1-indenylamino)-2,3- dimethyl-imidazo(1,2a)pyridine-6-carboxylate
05/11/2006US20060100233 Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
05/11/2006US20060100232 Inhibitors of HIV-1 capsid formation: substituted aryl aminomethyl thiazole ureas and analogues thereof
05/11/2006US20060100231 Amorphous clopidogrel hydrogen sulfate
05/11/2006US20060100230 Indolin phenylsulfonamide derivatives
05/11/2006US20060100229 Pyrazolopyridines and analogs thereof
05/11/2006US20060100228 Sulfonamide-containing benzene derivatives; cancer and inflammatory, immunomodulatory or respiratory diseases
05/11/2006US20060100227 Pyrimidine derivaties
05/11/2006US20060100226 2-Thiopyrimidinones as therapeutic agents
05/11/2006US20060100225 Heteroaryl guanidines; inhibitors of viral replication
05/11/2006US20060100224 Piperidine ouracil used as a medicament for treating bacterial infections
05/11/2006US20060100223 Quinazoline derivatives and pharmaceutical compositions containing them
05/11/2006US20060100222 Selective phosphodiesterase 9a inhibitors as medicaments for improving cognitive processes
05/11/2006US20060100221 5-[[(2,3-Difluorophenyl)methyl]thio]-7-[[2-hydroxy-1-(hydroxymethyl) 1 methylethyl]amino]-thiazolo[4,5-d]pyrimidin-2(3H)-one; asthma and allergic diseases, autoimmune pathologies such as rheumatoid arthritis and atherosclerosis
05/11/2006US20060100219 Dihydroimidazoles and tetrahydropyrmidines containing amide and sulfonamide groups, e.g., 3-[(2,3-Dichlorobenzenesulphonyl)methylamino]-N-{2-[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]ethyl}-N-methylpropionamide; treating pain, skin disease, irritable bladder or colon, asthma, COPD, and stomach inflammation
05/11/2006US20060100218 Phosphodiesterase 4; asthma, chronic obstructive pulmonary disease, Alzheimer's disease, diffuse large-cell B cell lymphoma, and chronic lymphocytic leukemia; 8-[3-(3,4-dimethoxy-phenyl)-pyrrolo[2,3-b]pyridine-1-sulfonyl]-quinoline
05/11/2006US20060100216 Novel B1 bradykinin receptor antagonists
05/11/2006US20060100215 8A,9-dihydro-4aH-isothiazolo[5,4-b]quinoline-3,4-diones and related compounds as anti-infective agents
05/11/2006US20060100214 Fast dissolving and taste masked oral dosage form comprising sildenafil
05/11/2006US20060100213 Triazoles and methods of use
05/11/2006US20060100212 fewer side effects; 2-keto-oxadiazole derivatives; 7-phenyl-1-[5-(pyridin-2-yl)-1,3,4-oxadiazol-2-yl]-heptan-1-one;
05/11/2006US20060100211 2-(3,4-dichlorophenylamino)-4-thiocyanato-5-nitro-pyrimidine; 2-chloro-4-(2-acetylamino-ethylamino)-5-trifluoromethyl-pyrimidine; lung cancer
05/11/2006US20060100210 Methods for treatment of scleroderma
05/11/2006US20060100209 Formulations of 1-(4-benzoyl-piperazin-1-yl)-2-[4-methoxy-7-(3-methyl-[1,2,4]triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-ethane-1,2-dione
05/11/2006US20060100208 Pyrazole derivatives as cannabinoid receptor antagonists
05/11/2006US20060100207 Dihydropyridinone derivatives
05/11/2006US20060100206 Heterocyclic CB1 receptor antagonists
05/11/2006US20060100205 Compositions for affecting weight loss
05/11/2006US20060100204 Anti-cytokine heterocyclic compounds
05/11/2006US20060100202 Novel compounds
05/11/2006US20060100201 5-Cyano-furan-2-carboxylic acid (4-morpholin-4-yl-2-piperidin-1-yl-phenyl)-amide; selective and potent protein tyrosine kinase inhibitors providing inhibition of c-fms kinase; treating autoimmune diseases and diseases with an inflammatory component; treating metastasis from ovarian, breast cancer
05/11/2006US20060100200 Selective oxidation of the the N-atom of the quinoline group using a peroxomonosulfuric acid, peroxodisulfuric acid or their salts in the presence of a ketone; N-atoms of the 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one scaffold are not oxidized
05/11/2006US20060100199 Novel condensed imidazole derivatives
05/11/2006US20060100198 Polymorphic and amorphous forms of the phosphate salt of 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-ce]indol-6-one
05/11/2006US20060100197 7,8,9,10-Tetrahydropyrido[2,3-b]azocine derivatives; CCR5 chemokine receptor antagonists; prophylactic for lymphadenopathy associated and/or human T-cell leukemia/lymphoma virus infections in peripheral mononuclear blood cells; AIDS; quaternization, oxidation, condensation, deprotecting, amidation
05/11/2006US20060100196 Substituted amines for the treatment of alzheimer's disease
05/11/2006US20060100195 Remedies for urinary frequency
05/11/2006US20060100194 Lactam compounds useful as protein kinase inhibitors
05/11/2006US20060100193 Factor Xa inhibitors
05/11/2006US20060100192 Heteroaryl diazacycloalkanes, their preparation and use
05/11/2006US20060100191 Kinesin spindle protein (KSP) inhibitors, e.g., 4-(2,5-Difluorophenyl)-N-[(3S,4S)-3-fluoropiperidin-4-yl]-2-hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1N-pyrrole-1-carboxamide, and a carrier; antiproliferative and -carcinogenic agents; side effects reduction; used with an estrogen receptor modulator
05/11/2006US20060100190 Motexafin lutetium phototherapy with low fluences for treating vascular inflammation
05/11/2006US20060100189 Method of treating or preventing pathologic effects of acute increases in hyperglycemia and/or acute increases of free fatty acid flux
05/11/2006US20060100188 Treatment methods
05/11/2006US20060100187 Synergistic combinations of macrolide t-cell modulator or immunosuppressant and a retinoid
05/11/2006US20060100186 Trandsdermal compositions and methods for treatment of fibromyalgia and chronic fatigue syndrome
05/11/2006US20060100185 5-Androsten-3beta-ol steroid intermediates and processes for their preparation
05/11/2006US20060100184 5-beta-sapogenin and pseudosapogenin derivatives and their use in the treatment of dementia
05/11/2006US20060100183 Therapeutic agents targeting the NCCa-ATP channel and methods of use thereof
05/11/2006US20060100182 Pharmaceutical compositions for the treatment of urinary incontinence
05/11/2006US20060100181 Combinations for the treatment of inflammatory skin disorders
05/11/2006US20060100180 Composition containing an androgenous 11b-halogen steroid and a progestational hormone, and male contraceptive based on said composition
05/11/2006US20060100179 Compositions and methods for use in targeting vascular destruction
05/11/2006US20060100178 Dermal agent
05/11/2006US20060100177 Stabilized ascorbic acid derivatives
05/11/2006US20060100176 Carboxylic acid diesters, methods for the production thereof and methods for the production of pharmaceutical active substances coupled to free amino groups with polysaccharide or polysaccharide derivatives
05/11/2006US20060100175 Novel therapeutic use of low molecular weight heparins
05/11/2006US20060100174 Configuration of glycosaminoglycans
05/11/2006US20060100173 Ophthalmic solution
05/11/2006US20060100172 Use of prebiotics, preferably glucooligosaccharide, for the prevention of the onset of type II diabetes
05/11/2006US20060100171 Branched alpha-glucans for weight management
05/11/2006US20060100170 Isopycnic pharmaceutical formulation
05/11/2006US20060100169 Method to reduce an inflammatory response from arthritis
05/11/2006US20060100168 Method of treating cancer using adenosine and its analogs
05/11/2006US20060100167 Methods and compositions for the treatment of autoimmune disorders using clofarabine
05/11/2006US20060100166 Compounds for modulating the activity of exchange proteins directly activated by camp (epacs)
05/11/2006US20060100165 aqueous emulsion for the treatment of rosacea skin disorders, acne, dermatitis; Glycerol, Isopropyl palmitate, Cetyl alcohol, Stearyl monostearate, Oleyl alcohol, Ceteareth-20; good cosmetic properties and long shelf-life with minimum of 2 years
05/11/2006US20060100164 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal
05/11/2006US20060100163 Oligosaccharides linked by amide, imine,ether, ester, carbonate, carbamate, urea, thioester bond to active agent produce hydrophilicity; easily produced with homogeneity, predictable, desirable pharmacokinetic profile, enhanced biocompatibility
05/11/2006US20060100162 Methods of mimicking the metabolic effects of caloric restriction by administration of mannoheptulose
05/11/2006US20060100161 Mitotic kinesin inhibitors and methods of use thereof
05/11/2006US20060100159 Preventing desensitization of receptors
05/11/2006US20060100157 Novel use of peptide compounds for treating pain in painful diabetic neuropathy
05/11/2006US20060100155 Method for the therapeutic management of endometriosis
05/11/2006US20060100152 Methods and compositions in treating pain and painful disorders using 9949, 14230, 760, 62553, 12216, 17719, 41897, 47174, 33408, 10002, 16209, 314, 636, 27410, 33260, 619, 15985, 69112, 2158, 224, 615, 44373, 95431, 22245, 2387, 16658, 55054, 16314, 1613, 1675, 9569 or 13424 molecules
05/11/2006US20060100150 Pharmacokinetic and pharmacodynamic modeling of erythropoietin administration
05/11/2006US20060100148 Glutathione-S-transferase tag, hexahistidine tag, maltose binding protein tag, haemagglutinin tag, and cellulose binding protein; for treating and preventing Flaviviridae virus (e.g., hepatitis C virus) infections
05/11/2006US20060100146 AWAT-related methods and articles
05/11/2006US20060100140 Combination of a) n-{5-[4-(4-methyl-piperazino-methyl)-benzoylamido]2-methylphenyl}-4- (3-pyridyl)-2-pyrimidine-amine and b) a histone deacetylase inhibitor for the treatment of leukemia
05/11/2006US20060100139 Pharmaceutical used for treating HIV infection, the composition and uses thereof
05/11/2006US20060100136 Synergistic effects of combined administration of mirtazapine and a stimulant compound