Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
08/2006
08/10/2006WO2005079195A3 Pyrazolopyridines and analogs thereof
08/10/2006WO2005077048A3 Immune modulation by regulating expression of the “minor” gene in immune dendritic cells
08/10/2006WO2005062782A3 Non-animal product containing veterinary formulations
08/10/2006WO2005055956A3 Method for improving insulin sensitivity by administering an inhibitor of antitrypsin
08/10/2006WO2005041997A8 Methods and compositions comprising ilex
08/10/2006WO2005041856A3 Use of 2-thia-dibenzo[e, h]azulenes for the treatment and prevention of central nervous system diseases and disorders
08/10/2006WO2005027962A9 4’-thionucleosides and oligomeric compounds
08/10/2006WO2005023189A3 Method of cox-2 selective inhibitor and nitric oxide-donating agent
08/10/2006WO2005017101A3 Avian adenoassociated virus (aaav) and uses thereof
08/10/2006WO2004105694A3 Pharmaceutical compositions and dosage forms for administration of hydrophobic drugs
08/10/2006WO2004050894A3 Heart failure gene determination and therapeutic screening
08/10/2006US20060179496 Nucleic acid sequences differentially expressed in cancer tissue
08/10/2006US20060178518 3'-[(2z)-[1-(3,4-Dimethylphenyl)-1,5-dihydro-3-methyl-5-oxo-4h-pyrazol-4-ylidene]hy-drazino]-2'-hydroxy-[1,1'-biphenyl]-3-carboxylic acid bis-(monoethanolamine)
08/10/2006US20060178516 Substituted quinolone carboxylic acids, their derivatives, site of action, and uses thereof
08/10/2006US20060178514 Novel benzylamine derivatives as CETP inhibitors
08/10/2006US20060178439 Crystalline form of zoledronic acid
08/10/2006US20060178438 Muscarinic agonists
08/10/2006US20060178437 Such as systemic lupus erythematosus by administering suberoylanilide hydroxamic acid; histone deacetylase inhibitors
08/10/2006US20060178436 Use of docosahexanoic acid as active substance for the treatment of lipodystrophy
08/10/2006US20060178435 Apogossypolone and the uses thereof
08/10/2006US20060178434 Butenoic acid derivatives processes for the preparation thereof pharmaceutical compositions comprising them and use for the treatment of dyslipidaemia atherosclerosis and diabetes
08/10/2006US20060178433 3-Amino-3-arylpropionic acid n-alkyl esters, process for production thereof, and process for production of optically active 3-amino-3-arylpropionic acids and esters of the antipodes thereto
08/10/2006US20060178432 Dyslipidemias, diabetes; (2S)-2-ethoxy-3-[4-(2-{4-[(methylsulfonyl)oxy]phenoxy}ethyl)phenyl]propanoic acid
08/10/2006US20060178430 Synthetic analogs of naturally occurring and non-naturally occurring acyl-homoserine lactone (AHL) analogs; N-butanoyl-L-homoserine lactone
08/10/2006US20060178429 2-Phenyl-3-hydrogenated furanyl, pyranyl, thiophenyl or thiopyranyl-N-heteroaromatic propionamides, e.g., 2-(3,4-Dichloro-phenyl)-3-(tetrahydro-pyran-2-yl)-N-thiazol-2-yl-propionamide; compounds increase insulin secretion in the treatment of type II diabetes.
08/10/2006US20060178428 7-Carboxymethyloxy-3',4',5-trimethoxy flavone monohydrate, the preparation method and uses thereof
08/10/2006US20060178427 chemically linking the taxane to a cell binding agent such as monoclonal antibody for tumor antigen; taxane has extra ether bridge group, and chemical group for conjugation such as mercapto
08/10/2006US20060178426 Kappa agonists, especialy for the treatment and/or prophylaxis of irritable bowel syndrome
08/10/2006US20060178424 Preventing atrial fibrillation (af) with the use of stain drugs
08/10/2006US20060178423 Administer amino acid precursor L-dopa, tyrosine, D,L-Phenylalanine, and N-acetyl-L-tyrosine; serotonin precursor of 5-HTP and tryptophan; and cofactors of vitamin B6, Vitamin C, Calcium, Folate, Cysteine; minimal side effects at higher doses, one precursor balances the other
08/10/2006US20060178422 Process for making (2S, 3aS, 7aS)-1-[(2S)-2-[[(1S)-1-(ethoxycarbonyl) butyl] amino]-1-oxopropyl] octahydro-1H-indole-2-carboxylic acid
08/10/2006US20060178421 Hydrogenation catalysts
08/10/2006US20060178420 Indole derivatives as anti-inflammatory agents
08/10/2006US20060178419 3-Sulfonylamino-pyrrolindine -2- one derivatives as inhibitors of factor xa
08/10/2006US20060178418 For therapy of asthma, bronchial asthma, chronic obstructive pulmonary disease, allergic rhinitis, eosinophilic granuloma, nephritis, rheumatoid arthritis, cystic fibrosis, chronic bronchitis, multiple sclerosis, Crohns disease, psoraisis, uticaria, adult vernal conjunctivitis,
08/10/2006US20060178417 4-[6(2,2-dimethylpropanoyloxy)indan-1-ylmethyl]1H-imidazole, an alpha 2 adrenergic agonist, for the treatment of hypertension, glaucoma, headaches, diarrhea, ischemia, drug abuse and dependence, hypotension, shock, congestive heart failure, anxiety, as decongestants, analgesics or as sedatives
08/10/2006US20060178415 Azole derivatives as antifungal agents
08/10/2006US20060178414 Treating rheumatoid arthritis, psoriasis, reperfusion injury, cardiovascular , autoimmune, inflammatory disorders and bronchial asthma; e.g., 2-Methoxynaphthalene-1-carboxylic acid benzyl-indan-2-yl-amide
08/10/2006US20060178413 Diphenylurea derivatives and their use as chloride channel blockers
08/10/2006US20060178412 [3-(Benzo[b]thiophene-2-carbonyl)-5-(4-methyl phenyl)-1H-indol-1-yl]-acetic acid, for treating conditions resulting from fibrinolytic disorders, such as deep vein thrombosis, coronary heart disease, and pulmonary fibrosis; Alzheimer's disease
08/10/2006US20060178411 Sulfonimide containing compounds and their use in polymer electrolyte membranes for electrochemical cells
08/10/2006US20060178410 Preparation of N-{2-[4-(3-phenyl-4-methoxyphenyl)aminophenyl]ethyl}-2-hydroxy-2-(3-hydroxymethyl-4-hydroxyphenyl)ethylamine, for example; for the treatment of pulmonary diseases such as asthma and chronic obstructive pulmonary disease
08/10/2006US20060178409 Anthranilic acid amides and their use as VEGF receptor tyrosine kinase inhibitors
08/10/2006US20060178408 Phosphodiesterases (PDE); for treating respiratory, nervous system, cardiovascular, inflammatory and allergic diseases, disorders and conditions as well as wounds
08/10/2006US20060178407 Substituted pyridines and their uses
08/10/2006US20060178406 Process for production of sulfoxide derivatives or salts thereof in the amorphous state
08/10/2006US20060178405 Non-insulin dependent diabetes; 7-[2-(5-methyl-2-phenyl-4-oxazole)ethoxyl]-2-oxo-2H-1-benzopyran-3-carboxylic acid methyl ester; insulin-sensitizing activities
08/10/2006US20060178403 Antiobesity agent, antidepressants, anxiolytic agents;3-[4-OXO-4H-THIENO[3,2-D]PYRIMIDIN-3-YL]-PYRROLIDINE-1-CARBOXYLIC ACID [1-(PYRROLIDIN-3-YL]-METHYL-AMIDES
08/10/2006US20060178402 For reducing levels of tumor necrosis factor alpha in mammals; 3-(1-Oxo-4-aminoisoindolin-1-yl)-3-methylpiperidine-2,6 dione; 1,3-dioxo-2-(2,6-dioxopiperidin-3-yl)-5-aminoisoindoline
08/10/2006US20060178401 Aminophenoxyacetamide derivatives and pharmaceutical composition containing thereof
08/10/2006US20060178400 Novel acetyl-CoA carboxylase (ACC) inhibitors and their use in diabetes, obesity and metabolic syndrome
08/10/2006US20060178399 Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient
08/10/2006US20060178398 and atherosclerosis; LXR agonists which increase HDL levels; increases ABCA1 gene expression; reverse cholesterol transport; 1,2-benzisoxazole 6-yl compounds
08/10/2006US20060178397 1-(3-Methyl-isoquinolin-5-yl)-3-[1-(2-trifluoromethyl-benzyl)pyrrolidin-3-yl]urea; calcium level blocker; lower fluorescence; neuropathic, postrheumatoid, osteoarthritic, back, cancer pain, algesia, neuralgia, dental pain, headache, migraine, neuropathies, carpal tunnel syndrome, diabetic neuropathy
08/10/2006US20060178396 e.g. (3-endo)-3-(2-Hydroxy-2,2-di-2-thienylethyl)-8,8-dimethyl-8-azoniabicyclo[3.2.1]octane bromide; muscle relaxants, respiratory system disorders; asthma, emphysema, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis
08/10/2006US20060178395 3-(2-Benzyl-2-hydroxy-3-phenyl-propylidene)-8,8-dimethyl-8-azonia-bicyclo[3.2.1]octane iodide; muscle relaxants, respiratory system disorders; asthma, bronchitis, chronic obstructive lung disease, chronic bronchitis, chronic respiratory obstruction, pulmonary fibrosis, pulmonary fibrosis
08/10/2006US20060178394 Inhalable dose of a powder comprising apomorphine or pharmaceutically acceptable salts thereof for therapy of for sexual dysfunction
08/10/2006US20060178393 1H-imidazo[4,5-d]thieno[3,2-b]pyridine based tricyclic compounds and pharmaceutical compositions comprising same
08/10/2006US20060178392 CCI-779 polymorph and use thereof
08/10/2006US20060178391 Method of preparing enantiomers of indole-2,3-dione-3-oxime derivatives
08/10/2006US20060178390 1,3,8-Triazaspiro[4,5]decan-4-one derivatives useful for the treatment of ORL-1 receptor mediated disorders
08/10/2006US20060178389 Use of siramesine in the treatment of cancer
08/10/2006US20060178388 Phenyl-substituted pyrimidine compounds useful as kinase inhibitors
08/10/2006US20060178387 Combined treatment with capecitabine and an epidermal growth factor receptor kinase inhibitor
08/10/2006US20060178386 For therapy of obesity, diabetes, diabetic complications, atherosclerosis, impared glucose tolerance and dyslipidemia; central nervous system diseases which includes but is not limited to, anxiety, depression, obsessive compulsive disorder, panic disorder, psychosis, schizophrenia, sleep disorder
08/10/2006US20060178385 e.g. 1-Benzyl-7-phenyl-3-propyl-1H-pyrrolo[1,2-f]purine-2,4(3H,6H)-dione; antiinflammatory, anticarcinogenic agent; cerebral ischemia, asthma, neurodegeneration, glaucoma, ischemic heart pre-conditioning; diagnostic agents
08/10/2006US20060178384 2-(2,6-dimethoxy-phenylamino)-9-methoxy-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one; 3-bromo-N-[3-(9-methoxy-4-oxo-6,7-dihydro-4H-pyrimido[6,1-a]isoquinolin-2-ylamino)-phenyl]-benzamide; kinase inhibitor; neutropenia; cytopenia; anemias
08/10/2006US20060178383 Novel 2-amino-quinazoline derivatives useful as inhibitors of beta-secretase (BACE)
08/10/2006US20060178382 Chinazoline derivatives as aurora kinase inhibitors
08/10/2006US20060178381 GlyT-1 inhibitors; CNS disorders such as psychoses, dysfunction in memory and learning, schizophrenia, dementia, attention deficit disorders, or Alzheimer's disease; (2-isobutoxy-5-methanesulfonyl-phenyl)-(3-trifluoromethyl-5,7-dihydro-pyrrolo[3,4-b]pyridin-6-yl)-methanone and pyrrolo[3,4-c]pyridines
08/10/2006US20060178380 Methods for treating cancer and other pathological proliferating disorders by inhibiting mitosis using pyrrolo[2,3-d]pyrimidines
08/10/2006US20060178379 Methods of treating patients suffering from movement disorders
08/10/2006US20060178378 Novel kinase inhibitors
08/10/2006US20060178377 e.g. Ethyl 6-(azidomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidine-2-carboxylate; treating diabetes and micro- and macrovascular complications of diabetes, such as retinopathy, neuropathy, and nephropathy
08/10/2006US20060178376 Novel process for the preparation of hexacyclic compounds
08/10/2006US20060178375 2-(1-Cyclopentylpiperidin-4-yloxy)-5-(4-cyanophenyl)pyrimidine, for example; exhibits histamine receptor H3 antagonist or inverse agonist activity and is useful for the treatment and/or prevention of obesity, diabetes, hormonal secretion abnormality, sleep disorders
08/10/2006US20060178374 Aminoheteroaryl compounds as protein kinase inhibitors
08/10/2006US20060178373 Oxy substituted flavones as antihyperglycemic and antidyslipidemic agents
08/10/2006US20060178372 Therapeutic quinoline compounds
08/10/2006US20060178371 7-amino-pyrrazolo[1,5-a]pyrimidine derivatives, useful in the treatment and prevention of proliferative diseases, for example, cancer, inflammation and arthritis
08/10/2006US20060178370 Ketopiperazine derivatives as bradykinin antagonists
08/10/2006US20060178369 Cinnamic acid amides
08/10/2006US20060178368 Administering a combination of nicotinic acid or nicotinamide and riboflavin to treat urticaria, asthma, allergic rhinitis, and allergic oculorhinitis
08/10/2006US20060178367 Certain imidazo[1,2-a]pyrazin-8-ylamines, method of making, and method of use thereof
08/10/2006US20060178366 Compounds for the treatment of inflammatory disorders
08/10/2006US20060178365 Optionally oxidized 6-(2-(5-methylthio-2-pyrimidinyloxy)ethoxy)-2-phenylpyrimidin-4-yl-substituted sulfamides
08/10/2006US20060178364 Use of EGFR tyrosinkinase inhibitors for treatment of chronic rhinosinusitis
08/10/2006US20060178363 Tetrahydropyranyl cyclopentyl heterocyclic amide modulators of chemokine receptor activity
08/10/2006US20060178362 Substituted heterocyle fused gamma-carbolines
08/10/2006US20060178361 ATM inhibitors
08/10/2006US20060178360 N(2-hydroxyethyl)-4-methoxy-N,2,6-trimethylbenzene- sulphonamide; analgesic, antiinflammatory agent; hyperalgesia and major algesia connected with other pathological conditions such as cancer
08/10/2006US20060178359 Tricyclic compound, process for producing the same, and use
08/10/2006US20060178358 e.g. 2-(4-Fluorophenyl)-7-(1-methylpiperidin-4-yl)-3-(2-methylpyrimidin-4-yl)imidazo[1,2-a]-pyridine; protozoal diseases (toxoplasmosis, malaria, African typanosomiasis, Chagas disease, and opportunistic infections) in mammals and birds; controlling coccidiosis in poultry
08/10/2006US20060178357 Chphalosporin-derived mercaptans as inhibitors of serine and metallo-beta-lactamases
08/10/2006US20060178356 Treating oxidative stress-related conditions typically responsive to cellular enzyme modulation with a substituted phenolic compound having unsaturated groups, e.g. 1-((3-methyl-5-oxo-2-pyrazolin-1-yl), 4-(3-methoxy-4-hydroxy-phenyl)-vinyl-)benzene; skin disorders; antiischemic and cardiotonic agents
08/10/2006US20060178355 Analogs of leucascandrolide A
08/10/2006US20060178354 Methods and compositions for the treatment of chronic pain using dhea and derivatives thereof
08/10/2006US20060178353 Medicament for preventing and/or treating mammarycarcinoma, containing a steroidal aromatase inhibitor
08/10/2006US20060178352 Use of androgens to reduce the likelihood of acquiring or to treat skin aging
08/10/2006US20060178351 Treatment of immune-mediated disorders with active vitamin D compounds alone or in combination with other therapeutic agents