Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
11/2008
11/12/2008CN100431547C A triptolide composite preparation for treating osteoarthritis by joint intracavity injection
11/12/2008CN100431546C Progestational hormone composition, and its slow-release suppository device and preparation of said device
11/12/2008CN100431545C Use of compositions comprising an estrogenic component for the treatment and prevention of musculoskeletal pain
11/12/2008CN100431544C Formulations of glucocorticoids to treat pathologic ocular angiogenesis
11/12/2008CN100431543C Pharmaceutical composition
11/12/2008CN100431542C Application of yohimbine and berberine mixture in medicament preparation
11/12/2008CN100431541C Phentanyl-containing adhesive patch for application to oral-cavity mucosa
11/12/2008CN100431540C Treatment of diabetes with thiazolidinedione and metformin
11/12/2008CN100431539C Use of acetylchloinesterase inhibitor for preparing medicine for treating parkinson's disease
11/12/2008CN100431538C An anticancer pharmaceutical composition and preparation method thereof
11/12/2008CN100431537C Blood fluidity improving agent
11/12/2008CN100431536C Alpha 2b 0r 2b/2c adrenoceptor agonists for the treatment of neurodegeneration
11/12/2008CN100431535C Chlorhydric acid tranditerol aerosol
11/12/2008CN100431534C Methods of inhibiting vascular permeability and apoptosis
11/12/2008CN100431533C Medicinal composition containing backuchiol for treating female osteoporosis
11/12/2008CN100431532C Breviscapine and borneol constituted composite injection formulation and preparation method thereof
11/12/2008CN100431531C Transdermal pharmaceutical spray formulations comprising a vp/va copolymer and a non-aqueous vehicle
11/12/2008CN100431530C Soft polyene phosphatidylcholinecapsule and its prepn process
11/12/2008CN100431526C A rapidly disintegrating tablet of acid sensitive drug
11/12/2008CN100431516C Device for calculating elixir doses approprate for patient's weight
11/12/2008CN100431434C Soft drink replacer
11/11/2008US7449605 Drugs; therapy for kidney diseases; removal of bile acid; gastrointestinal disorders; core-shell polymer
11/11/2008US7449599 Phenyl carboxamide compounds useful as beta-secretase inhibitors for the treatment of alzheimer's disease
11/11/2008US7449595 Nitrosated and nitrosylated prostaglandins, compositions and methods of use
11/11/2008US7449594 Process for preparing 4-pentafluorosulfanylbenzoylguanidines
11/11/2008US7449589 passing a mobile phase comprising carbon dioxide through a stationary phase comprising a derivatised polysaccharide, and wherein the process is capable of providing at least 0.1 gram of the separated (-)- Delta 9-trans-tetrahydrocannabinol in less than a day
11/11/2008US7449585 1,2-dihydro-2-(4-trifluoromethylphenyl)-6-(3-trifluoromethyl-2-pyridinyl)-3H-indazol-3-one; capsaicin receptor ; analgesic, antiinflammatory, hypotensive agent; rheumatoid arthritis, osteoarthritis, headache, migraine, cancer and central nervous system pain, irritable bowel syndrome
11/11/2008US7449583 Process for the preparation of 4-(8-chloro-5 6-dihydro-11h-benzo-(5 6)-cyclohepta-(1 2b)-pyridin-11-ylidene-1-piperidiniecarboxylic acid ethyl ester (loratadine)
11/11/2008US7449582 particularly tyrosine kinase, serine-threonine kinases, and MAP kinases; cancer, nervous system disorders and autoimmune diseases; 6-phenyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidines, 3-phenyl-2-oxo-1,2-dihydro-[1,6]naphthyridines, and 3-phenyl-2-oxo-1,2-dihydroquinolines
11/11/2008US7449581 6-Substituted pyrido-pyrimidines
11/11/2008US7449575 preparing 4-[[4-amino-6-[(2,6-dichlorophenyl)methyl]-1,3,5-triazin-2-yl]amino]benzonitrile by reacting 2,6-dichlorobenzeneethanimidamide with phenyl N'-cyano-N-(4-cyanophenyl)-carbamimidate in a reaction-inert solvent; HIV (Human Immunodeficiency Virus) infection
11/11/2008US7449572 Reducing compound such as 3,3-ethylenedioxyestra-5(10), 9(11)-dien-17-ol, halogenating, epoxidation, alkylation, deprotecting, aromatization, saponification, neutralization to obtain compound such as 11-beta-(4-(2-(1-piperidinyl)ethoxy)phenyl)-17-alpha-fluoroestra-1,3,5(10)-trien-3-ol
11/11/2008US7449571 Halogenated aminoquinolines and oligonucleotides containing the same
11/11/2008US7449570 Use of nucleoside compounds for nonsense suppression and the treatment of genetic diseases
11/11/2008US7449565 Chimeric tumor suppressor gene and protein
11/11/2008US7449537 Antineoplastic polyalkoxyalkylsiloxanes and methods of use thereof
11/11/2008US7449495 e.g. 4-(3-(1-Adamantyl)-4-tert-butyldimethyl-silyloxyphenyl)benzaldehyde; antitumor, antiinflammatory agent; arthritic pathology, metastatisation, diabetic retinopathy, psoriasis, chronic inflammatory disease, and atherosclerosis; sarcoma, carcinoma, carcinoid, leukaemia
11/11/2008US7449494 made by the reaction of dimethyl ethanolamine, and tetra 2-hydroxyalkyl ethylene diamne with di-chloro glycerin in water
11/11/2008US7449493 N-[2-[[1-[[[(2,4-dimethylphenyl)methyl]amino]methyl]cyclohexyl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide; monocyte chemoattractant proteins receptor antagonists or partial agonists/antagonists; antiinflammatory agent, autoimmune diseases; rheumatoid arthritis, multiple sclerosis, atherosclerosis
11/11/2008US7449492 Therapeutic agents—I
11/11/2008US7449491 Natural vitamin E compositions with superior antioxidant potency
11/11/2008US7449490 Pharmaceutically active compounds and methods of use
11/11/2008US7449489 e.g. isopropyl [({2-[5-[2-(2-azabicyclo[2.2.2]oct-2-yl)- 1,1-dimethyl-2-oxoethyl]-2-(3,5-dimethylphenyl)-1H-indol-3-yl]propyl }amino)(3-pyridin-4-ylpyrrolidin-1-yl)methylene]carbamate; gonadotrophin releasing hormone antagonists; anticarcinogenic agent; breast, prostate, uretus cancer
11/11/2008US7449488 Pyrazolopyrimidines as protein kinase inhibitors
11/11/2008US7449487 In particular of avocado, soya bean and/or lupin oils, for preparation of a medicament intended to stimulate expression of TGF-62 or expression of the plasminogen activator inhibitor PAI-1
11/11/2008US7449486 Mitotic kinesin inhibitors and methods of use thereof
11/11/2008US7449485 N-sulfonylurea apoptosis promoters
11/11/2008US7449484 angiogenesis inhibitor; Tie2 receptor kinase inhibitors; 2-tert-Butyl-4-naphthalen-2-yl-5-pyridin-4-yl-imidazole;2-tert-Butyl-4-(6-Ethoxynaphthalen-2-yl)-5-pyridin-4-yl-imidazole;4-(2-tert-Butyl-5-(6-methoxy-naphthalen-2-yl)-3H-imidazol-4-yl)-pyridine; etc.
11/11/2008US7449483 e.g. 2-(Ethyl-{4-[2-methyl-3-(4-trifluoromethyl-phenyl)-benzo[b]thiophen-6-yl]-butyl}-amino)-ethanol; 2,3-oxidosqualene-lanosterol cyclase inhibitor; antidiabetic, antitumor, antiproliferative agent; hypercholesterolemia, hyperlipemia, arteriosclerosis, vascular diseases, mycoses, gallstones
11/11/2008US7449482 Piperidine compounds useful as malonyl-CoA decarboxylase inhibitors
11/11/2008US7449481 Thio-substituted biaryl-methanesulfinyl derivatives
11/11/2008US7449480 Small molecule inhibitors of HER2 expression
11/11/2008US7449479 Hepatitis C virus inhibitors
11/11/2008US7449478 Treatment of peroxisome proliferation activated receptor diseases such as diabetes, skin disorders or high blood pressure
11/11/2008US7449477 7-phenyl-isoquinoline-5-sulfonylamino derivatives as inhibitors of akt (protein kinase B)
11/11/2008US7449476 e.g. 2,3,4,5-tetrahydro-2-[2-[4-methoxy-7-(5-methyl-1H-1,2,4-triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-1,2-dioxoethyl]-5-phenyl-1H-pyrido[4,3-b]indole; inhibit HIV entry by attaching to exterior viral envelop protein gp120 and interrupting viral entry process by interfering with cellular receptor CD4
11/11/2008US7449475 e.g. 2-{[(2S)-3-(5-Chloro-1'H,3H-spiro[1-benzofuran-2,4'-piperidin]-1'-yl)-2-hydroxypropyl]oxy}-N-cyclopropylbenzamide; macrophage inflammatory protein (MIP)-1 alpha chemokine receptor modulator; antiinflammatory, antiproliferative agent, autoimmune diseases
11/11/2008US7449474 Tri-substituted ureas as cytokine inhibitors
11/11/2008US7449473 8-(1-methyl-1H-pyrrol-2-yl)-1,3-dipropyl-1H-pyrrolo[3,2-d]pyrimidine-2,6-dione; asthma, chronic obstructive pulmonary disorder, emphysema, diabetic disorders, inflammatory gastrointestinal tract disorders, immunological/inflammatory disorders, cardiovascular diseases, neurological disorders
11/11/2008US7449472 Methods of inhibiting p38 with substituted bicyclic pyrimidines
11/11/2008US7449471 5-phenylpyrimidines, their preparation, compositions comprising them and their use
11/11/2008US7449470 Antagonists to treat neurodegenerative diseases like Parkinson's disease; 2,4,6-trisubstituted pyrimidines; N-(2,6-diphenyl-pyrimidin-4-yl)-benzamide
11/11/2008US7449469 Improved pharmacological activity and tolerability; glaucoma; ocular hypertension
11/11/2008US7449468 Thiazole and oxazole derivatives as activators of human peroxisome proliferator activated receptors
11/11/2008US7449467 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
11/11/2008US7449466 Cyclic aminophenyl sulfamate derivative
11/11/2008US7449465 glycogen synthase kinase 3 alpha and 3 beta inhibitors; improved phanrmacological activity, potency, selectivity, solubility, permeability, metabolic stability; bipolar disorder; Alzheimer's disease; type II diabetes, neuropathic pain; depression; inflammatory diseases
11/11/2008US7449464 4-{3-[4-(6-Chlorobenzothiazol-2-yl)-1,4-diazepan-1-ylcarbonyl]benzyl}-1(2H)-phthalazinone; Cancer, BRCA deficient
11/11/2008US7449463 Morpholinyl containing benzimidazoles as inhibitors of respiratory syncytial virus replication
11/11/2008US7449462 2-{4-[4-(2-Ethyl-phenyl)-5-methyl-4H-[1,2,4]triazol-3-yl]-piperidin-1-yl}-pyrimidine; more potent, longer duration of action, broader range of activity, more stable, fewer side effects, selectivity; anxiety, cardiovascular disease, dysmenorrhoea, endometriosis, emesis, inflammation, sexual disorders
11/11/2008US7449461 Benzathiazol-acetamides
11/11/2008US7449460 3-Quinolinecarbonitrile protein kinase inhibitors
11/11/2008US7449459 Inhibitors of soluble adenylate cyclase
11/11/2008US7449458 Prodrugs of 2,4-pyrimidinediamine compounds and their uses
11/11/2008US7449457 Substituted heterocyclic carboxamides with antithrombotic activity
11/11/2008US7449456 signal transducer and activator of transcription-6 inhibitors; asthma, COPD, respiratory, inflammatory and allergic diseases; compounds have less suppressive effect on immunological functions; 4-[(2,5 -difluorobenzyl) amino]-2-[(4-morpholin-4-ylphenyl)amino]pyrimidine-5 -carboxamide
11/11/2008US7449455 1-[4-(2-azepan-1-yl-ethoxy)-benzyl]-2-(4-hydroxy-phenyl)-3-methyl-1H-indol-5-ol; contraception; melanoma; capable of inhibiting bone loss while showing little or no uterine stimulation, decrease the weight gain, decrease cholesterol levels, prevent bone loss
11/11/2008US7449454 Metallotexaphyrin derivatives
11/11/2008US7449453 Treatment of prostate cancer by administering an azetidinone-based cholesterol absorption inhibitor such as ezetimibe, the phenolic glucuronide of ezetimibe, SCH 48461 or SCH 58053, optionally with an anticancer agent
11/11/2008US7449451 Radiation resistance; prevent tissue damage; pretreatment with oxidation resistant
11/11/2008US7449450 Compounds, methods of screening, and in vitro and in vivo uses involving anti-apoptotic genes and anti-apoptotic gene products
11/11/2008US7449449 Providing microprojectiles carrying polynucleic acid sequences; accelerating the microprojectiles at the preselected-cells, with the microprojectiles contacting cells to penetrate vertebrate cells and deposit polynucleic acid
11/11/2008US7449448 Administering fructose of fructose containing oligosaccharide
11/11/2008US7449447 Peptidomimetic NS3-serine protease inhibitors of hepatitis C virus
11/11/2008US7449446 Synergistic mixture; anticoagulants
11/11/2008US7449444 Hydroxyethyl starch-containing polypeptide compositions
11/11/2008US7449442 EGFR inhibitors promote axon regeneration
11/11/2008US7449321 Controlling a flavivirus entry into a cell by administering to the cell an agent functionally interfering with a flavivirus receptor protein, the flavivirus receptor protein being an integrin
11/11/2008US7449315 Bifunctional energy-reversible acyl-compositions
11/11/2008US7449236 Porous polymeric particle comprising polyvinyl alcohol and having interior to surface porosity-gradient
11/11/2008US7449200 positively charged shell substrate, negatively charged core substrate with encapsulated bioactive agents; for projectile bombardment; composed of chitosan/poly-glutamic acid/insulin or chitosan/poly-glutamic acid/pDNA for transcutaneous delivery
11/11/2008US7449198 Stable salts of O-acetylsalicylic acid with basic amino acids
11/11/2008US7449197 Liposome formulation of 6,9-bis[(2-aminoethyl)-amino]benzo[g]isoquinoline-5, 10-dione dimaleate
11/11/2008US7449196 Anti tumor compositions and methods of use
11/11/2008US7449195 Fungicide mixtures
11/11/2008US7449175 Delivery of erectile dysfunction drugs through an inhalation route
11/11/2008US7449174 Delivery of analgesics through an inhalation route
11/11/2008US7449173 heating drugs used for the treatment of anxiety or insomnia, coated on solid supports to form vapors and condensing the vapor to form aerosols comprising microstructure particles of the drugs
11/11/2008US7449172 Delivery of antiemetics through an inhalation route
11/11/2008CA2588369A1 Methods of treatment and prevention of metabolic bone diseases and disorders