Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
07/2010
07/07/2010CN101229156B Medicine composition used for cardiovascular disorders
07/07/2010CN101229141B Aspirin sustained release tablet and preparing method thereof
07/07/2010CN101167743B Compound xylitol electrolyte injection and preparation method thereof
07/07/2010CN101138557B Chlorhexidine acetate partial film forming gel composition and uses thereof
07/07/2010CN101039939B Quinazolinylmethylene thiazolinones as CDK1 inhibitors
07/07/2010CN101023973B Extract of polysaccharide of lithospermum erthrorhizon and composition containing same and use thereof
07/07/2010CN101015545B Use of phenylpropionic acid and phenyl propyl compound with oxidation resistance function for protecting liver and brain damage
07/07/2010CN101015544B Use of phenyl propyl compound with oxidation resistance function for protecting liver and brain damage
07/07/2010CN101015543B Use of cinnamic acid and allyl benzoate compound with oxidation resistance function for protecting liver and brain damage
07/07/2010CN101002930B Medicine composition containing aniracetam and brain protein hydrolyte
07/06/2010USRE41425 Piperazine and piperidine compounds
07/06/2010US7750199 Kit systems for granulated decontamination formulations
07/06/2010US7750164 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
07/06/2010US7750161 N-Cyclopropyl-N-(1-{2-[3-(2,6-dimethyl-pyridin-4-yl)-ureido]-ethyl}-piperidin-4-yl)-2-fluoro-benzenesulfonamide; 2-(4-Chloro-phenyl)-N-(1-{2-[3-(2,6-dimethyl-pyridin-4-yl)-ureido]-ethyl}-piperidin-4-yl)-N-methyl-acetamide; neurohormonal antagonists
07/06/2010US7750160 inhibit p38, MAP kinase interacting serine/threonine kinase 2 (MKNK2 kinase) and serine-threonine kinases (STKs); treating proliferative diseases including cancer, leukemias; e.g. N-(isoxazolyl)urea compounds and thiourea compounds
07/06/2010US7750158 Sulfonamide-containing benzene derivatives; cancer and inflammatory, immunomodulatory or respiratory diseases
07/06/2010US7750154 Amide derivatives
07/06/2010US7750151 Inhibitors of Akt activity
07/06/2010US7750150 Process for producing acid adduct salt of polyacidic base compound
07/06/2010US7750148 chemical intermediates for making an oral antibiotics Sulbactam
07/06/2010US7750145 sodium glucose co-transporter 2 inhibitors; for prevention or treatment of diabetes, postprandial hyperglycemia, impaired glucose tolerance, diabetic complications, obesity
07/06/2010US7750140 Ghrelin binding nucleic acids
07/06/2010US7750121 A recombinant human telomerase reverse transcriptase (hTRT) protein; drug screening for antiproliferative agents that inhibit hTRT activity; cancer diagnosis and prognosis; anticarcinogenic agents
07/06/2010US7750053 Compositions and methods for alleviating hypertension or preventing a rise in blood pressure
07/06/2010US7750052 Separately protonation of alcohol and water; blending; food processing
07/06/2010US7750051 Amine oxidase inhibitors
07/06/2010US7750050 Enhancing activity of an acid sphingomyelinase (ASM) protein with an analogue of ceramide, sphingomyelin or phosphonucleotide; gene therapy
07/06/2010US7750049 vanilloid receptor antagonists such as 1-[4-(2-hydroxyethoxy)-2-bromo-5-methoxybenzyl]-3-[4-(trifluoromethyl)-benzyl]urea, useful for the treatment of neuropathic pain, urogenital disorders, hemorrhoids, inflammation, post-operative pain, respiratory and gastrointerstinal disorders
07/06/2010US7750048 GPR40 agonists
07/06/2010US7750047 benzoic acid derivatives, used as acetyltransferase enzyme inhibitors, used in the treatment of diseases due to defects in gene regulation predominantly cancer
07/06/2010US7750046 Treatment of symptoms associated with irritable bowel syndrome
07/06/2010US7750045 Compounds, compositions and methods for preventing neurodegeneration in acute and chronic injuries in the central nervous system
07/06/2010US7750044 Dimer poly-quaternary ester compounds
07/06/2010US7750043 Retinoic esters with pinacol; antiproliferative agents; disorders caused by abnormal cellular differentiation; psoriasis, cancers of skin, colon, lungs, breasts, prostate, or ovaries, leukemia, neuroblastomas, eczema, acne; improved wrinkle resistance, skin hydration, sebum secretions
07/06/2010US7750042 substituted bis[thio-hydrazide amide] compounds; synergistic effect with taxol or taxotere, anticancer agents, minimal toxic side-effects
07/06/2010US7750041 Using antihyperplastic agent; diffusion through capillaries; imaging veins, arteries; side effect reduction; antitumor agents
07/06/2010US7750040 G protein-coupled receptor S1P1/EDG1 agonists; low dosage, long lasting immunosuppressive effect; such as 1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalene-4-carboxylic acid 2,4-dimethoxy-benzylamide
07/06/2010US7750039 administering [7-(benzyloxy)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone to mammals as analgesics, antiinflammatory agents and as neuroprotectants
07/06/2010US7750038 1-methyl-5-[1-(methylsulfonyl)-2,3-dihydro-1H-indol-5-yl]-1H-pyrrole-2-carbonitrile; contraception; fibroids, uterine leiomyomata, endometriosis, dysfunctional bleeding, polycystic ovary syndrome, and hormone-dependent carcinomas; providing hormone replacement therapy; stimulating food intake
07/06/2010US7750037 Antidepressant
07/06/2010US7750036 Carvedilol salts, corresponding compositions, methods of delivery and/or treatment
07/06/2010US7750034 Aminocyclohexanes as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
07/06/2010US7750033 administering an enzyme inhibitor of c-Jun N-terminal Kinase (JNK), Anthra[1-9-cd]pyrazol-6(2H)-one for treating the vascular aneurysm
07/06/2010US7750032 Compounds and compositions as PPAR modulators
07/06/2010US7750031 Caffeic acid derivative and composition containing the same
07/06/2010US7750030 Acute pharmacologic augmentation of psychotherapy with enhancers of learning or conditioning
07/06/2010US7750029 administering (R)-2-(2-aminothiazol-4-yl)-4'-[2-[(2-hydroxy-2-phenylethyl)amino]ethyl]acetic acid anilide; treating urogenital disorders
07/06/2010US7750028 treating epilepsy comprising administering polymorphic rufinamide's that differ with respect to their thermodynamic stability, in their physical parameters, such as the absorption pattern of infrared and raman spectrum analysis
07/06/2010US7750027 Compounds having CRTH2 antagonist activity
07/06/2010US7750026 N-Cyclopropyl-3-[5-fluoro-3-(4-pyridinyl)-1H-indazol-6-yl]-4-methylbenzamide, useful in the treatment of conditions or disease states mediated by p38 mitogen-activated protein kinase activity or mediated by cytokines produced by the activity of p38 mitogen-activated protein kinases
07/06/2010US7750025 Derivatives of N-phenyl (piperidine-2-yl) methyl benzamide, preparation method thereof and applications of same in therapeutics
07/06/2010US7750024 [7-(1H-imidazol-1-yl)-6-nitro-2,3-dioxo-3,4-dihydroquinoxalin-1(2H)-yl]acetic acid, 2-[N-(4-chlorophenyl)-N-methylamino]-4H-pyrido[3,2-e]-1,3-thiazin-4-one, or 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(F)-quinoxaline; AMPA receptor antagonist; anticarcinogenic agents
07/06/2010US7750023 Quinuclidine derivatives and medicinal compositions containing the same
07/06/2010US7750022 modulators of nicotinic and/or of the monoamine receptors such as 3-(Dibenzofuran-2-yloxy)-1-azabicyclo[2.2.2]octane, useful for the treatment of nervous system disorders, neurodegenerative diseases and drug abuse and dependence
07/06/2010US7750021 3-{[2-(2-Trifluoromethyl-biphenyl-4-yl)-benzo[b]thiophen-5-ylmethyl]-amino}-propionic acid, useful in the treatment or prevention diseases associated with endothelial differentiation, G-protein-coupled (EDG) receptor mediated signal transduction, such as acute or chronic transplant rejection
07/06/2010US7750020 3-Cyclopentyl-2-(4-cyclopropylsulfamoyl-phenyl)-N-(5-methoxy-thiazolo[5,4-b]pyridin-2-yl)-propionamide; antidiabetic agent; insulin resistance, impaired glucose tolerance, obesity; with other hypolipidemic agent, anti-obesity and hypotensive agent
07/06/2010US7750019 Pyrimidine compound having benzyl(pyridylmethyl)amine structure and medicament comprising the same
07/06/2010US7750018 Use of carboxiamidotriazole (CAI) orotate in macular degeneration
07/06/2010US7750017 Anticancer agents; hyperproliferative diseases; 4-(phenylamino)benzothieno[2,3-d]pyrimidines; inhibit the tyrosine kinase activities of EGFR (erbB1) and HER2
07/06/2010US7750016 Hydroxyalkyl substituted pyrido-7-pyrimidin-7-ones
07/06/2010US7750015 Nitrogen-containing heterocyclic compounds and methods of use thereof
07/06/2010US7750014 Imidazo[1,2-C]pyrimidinylacetic acid derivatives
07/06/2010US7750013 N-oxides as prodrugs of piperazine and piperidine derivatives
07/06/2010US7750012 leukotriene A4 hydrolase inhibitors such as 4-{4-[4-(4-Iodo-phenoxy)-phenyl]-piperazin-1-yl]-butyric acid methyl ester, used for the treatment, prevention and/or prophylaxis of inflammatory diseases and disorders
07/06/2010US7750011 Diazabicyclic aryl derivatives and their medical use
07/06/2010US7750010 2-(2,5-Dioxo-5,6-dihydro-4H-imidazo[1,5,4-de]quinoxalin-1(2H)-yl)-N-(3-methyl-spiro[imidazolidine-4,2'-indane]-2,5-dione)acetamide, used as Calcitonin Gene-Related Peptide (CGRP), ligands useful in the treatment or prevention of headaches
07/06/2010US7750009 7-benzyloxy-6-chloro-2-piperazin-1-yl-4-pyrrolidin-1-yl-pteridine, uitable for treating respiratory system or gastrointestinal disorders, inflammatory diseases of the joints, skin or eyes, diseases of the peripheral or central nervous system and cancers
07/06/2010US7750008 poly(ADP-ribose) polymerase (PARP) inhibitors such as 9-[(Hydrozinooxy)carbonyl]-2,7-dihydro-6-methoxy 3H-pyrido-[4,3,2-de]phthalazin-3-one, used for treating neuron tissue damage resulting from ischemia and reperfusion injury, depression, inflammatory bowel disorders, arthritis, gout, pain and sepsis
07/06/2010US7750007 Imidazo[1,2-beta]pyridazine and pyrazolo[1,5-alpha]pyrimidine derivatives and their use as protein kinase inhibitors
07/06/2010US7750006 e.g. 4-[5-(Piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; multiple sclerosis
07/06/2010US7750005 Substituted hexahydropyrazino [1,2-A] pyrimidine-4,7-dione derivatives, process for their preparation and their use as medicaments
07/06/2010US7750004 Apoptosis promoters
07/06/2010US7750003 mammalian target of rapamysin (mTOR)/phosphatidylinositol (PI) kinase-related kinase (PIKK) family inhibitor; antiproliferative, anticarcinogenic, antiinflammation agent, immunostimulant;
07/06/2010US7750002 Anticancer agents; kinase inhibitors; viricides; antiinflammatory agents; immunotherapy; metabolism disorders
07/06/2010US7750001 2-(2-methylbenzimidazol-1-yl)-4,6-dimorpholino-1,3,5-triazine; phosphatidylinositol 3-kinase (PI3K) inhibitor; transplantation of organs or tissues, inflammatory bowel diseases, psoriasis or atopic dermatitis, chronic obstructive pulmonary disease, asthma, rheumatoid arthritis, scleroderma
07/06/2010US7750000 Substituted imidazo[1,2b]pyridazines as kinase inhibitors, their preparation and use as medicaments
07/06/2010US7749999 Alpha-ketoamides and derivatives thereof
07/06/2010US7749998 urotensin antagonists such as N-[1-(4-biphenyl)-1)-2-(1-pyrrolidinyl)ethyl]-2-(6,7-dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)-N-methylacetamide, used for treating congestive heart failure, stroke, ischemia, angina, overactive bladder or arrhythmia
07/06/2010US7749997 Pyrimido [4,5-B] -Oxazines for use as DGAT inhibitors
07/06/2010US7749996 Heterotricyclic metalloprotease inhibitors
07/06/2010US7749995 modulator of cholesteryl ester transfer protein (CETP), such as 1,1,1-Trifluoro-3-[3-[3-(1,1,2,2-tetrafluoro-ethoxy)-phenyl]-8-(3-trifluoromethoxy-phenyl)-2,3-dihydro-benzo[1,4]oxazin-4-yl]-propan-2-ol, used for treating cardiovascular disorders, dyslipidemia, and metabolic disorders
07/06/2010US7749994 serine/threonine kinase inhibitors, useful for therapy and/or prophylaxis of cancers in mammals
07/06/2010US7749993 Utillizing vasopressin antagonistic agent such as 5-dimethylamino-1-[4-(2-methylbenzoylamino)benzoyl]-2,3,4,5-tetrahydro-1H-benzazepine; safe with few side effects
07/06/2010US7749992 modulators of Cholesterol ester transfer protein activity, such as 5-[Acetyl-(3,5-bis-trifluoromethyl-benzyl)-amino]-7-trifluoromethyl-2,3,4,5-tetrahydro-benzo[b]azepine-1-carboxylic acid isopropyl ester, for treating or preventing cardiovascular disorders
07/06/2010US7749991 photosensitizers used in the photodynamic therapy of microbial infections, tumors, pre-cancerous and proliferative pathologies and/or in the diagnosis, as well as for blood and blood derivatives sterilization
07/06/2010US7749990 [3-(2,6-Dimethylbenzyloxy)-phenyl]-oxoacetic acid, useful for the treatment of insulin resistance syndrome, diabetes, hyperlipidemia, fatty liver disease, cachexia, obesity, atherosclerosis and arteriosclerosis
07/06/2010US7749989 Estrogenic compounds, methods of using and methods of administering the same
07/06/2010US7749988 Triterpenoid derivatives
07/06/2010US7749987 treating with a mixture comprising nomegestrol acetate and estradiol valerate or estradiol; side effect reduction
07/06/2010US7749986 Homogeneously formulating microdosed active principles
07/06/2010US7749985 3-{[1-Isobutanoyloxyethoxy]carbonylamino}propyl(n-butyl)phosphinic acid, used treating a disease chosen from mild cognitive impairment, cognitive impairment associated with Alzheimer's disease, depression, anxiety and epilepsy; intermediates for 3-aminopropylphosphinic acid and analogs
07/06/2010US7749984 drug design, a derivative of dextromethorphan having an imidazolidine group; calcium channel blockers
07/06/2010US7749983 viricides; anticarcinogenic agents; biological conjugated drug
07/06/2010US7749982 Complex containing mequitazine, a cyclodextrin and an interaction agent
07/06/2010US7749981 Drug-eluting stents coated with non-nucleotide P2Y12 receptor antagonist compound
07/06/2010US7749980 purinergic receptor antagonists such as 6-{2,2-Dimethyl-6-[6-(3-phenyl-ureido)-purin-9-yl]-tetrahydro-furo [3,4-d][1,3]dioxol-4-ylmethoxy}-5-fluoro-nicotinic acid, used as analgesics
07/06/2010US7749979 CpG DNA adjuvant in avian vaccines
07/06/2010US7749978 Compositions and methods for inhibiting expression of Huntingtin gene
07/06/2010US7749977 Therapeutic modulation of the Fas pathway
07/06/2010US7749976 increasing insulin production by PTPMT1 positive cells by contacting PTPMT1-positive cells with a siRNA molecule that recognizes and binds PTPMT1 thereby regulating insulin production