Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
08/2010
08/24/2010US7781435 (S)-2-[2-(3,5-Difluoro-phenyl)-acetylamino]-pentanoic acid {1-[2-(3-ethoxy-propylamino) -ethyl]-1H-imidazol-4-yl}-amide, having beta-amyloid peptide production inhibitory activity, used for the treatment of neurodegenerative disorders such as Alzheimer's disease
08/24/2010US7781434 7-Chloro-2-isopropyl-5-[3-(morpholine-4-carbonyl)-isoxazol-5-yl]-2,3-dihydro-isoindol-1-one; drug targets in the therapy of acute and chronic neurological and psychiatric disorders and chronic and acute pain disorders; schizophrenia or anxiety; Sandmeyer reaction of a 4-bromoaniline
08/24/2010US7781433 Pharmaceutical compounds
08/24/2010US7781432 analgesic. especially acute, chronic and/or neuropathic pain; epilepsy and other CNS-related disorders as well as for neuroprotection or cardioprotection; 9-benzyl-8-(cyclopentylamine)-6-(4-nitrobenzyl-mercaptopurine
08/24/2010US7781431 Thienopyrroles as antiviral agents
08/24/2010US7781430 Benzoxazole carboxamides for treating CINV and IBS-D
08/24/2010US7781429 solubilizing a nonsteroidal antiinflammatory drug (NSAID) such as diclofenac by combining with at least two of camphor, menthol and thymol
08/24/2010US7781428 Pyrazoline compounds
08/24/2010US7781427 cyclization of a 1,4-benzodiazepine with cyclopentene. in a diels-alders reaction to give a decahydrocyclopenta[c][1,4]diazepino[6,7,1-ij]quinoline, then resolving to form diastereomeric salts and dimer impurities; neuroleptic and dietetic agents
08/24/2010US7781426 cholesterol ester transfer protein (CETP) inhibitors such as (4S,5R)-5-[3,5-bis(trifluoromethyl)phenyl]-3-[2-(3,3-dimethylpiperidin-1-yl)-5-(trifluoromethyl)benzyl]-4-methyl-1,3-oxazolidin-2-one, useful for raising HDL-cholesterol, reducing LDL-cholesterol, and for treating or preventing atherosclerosis
08/24/2010US7781423 administering to a cancer patients, heterocyclic trialkyl ammonium-compounds such as [3-(3,4-dimethyl-9-oxo-9H-thioxanthen-2-yloxy)-2-hydroxypropyl]trimethylammonium chloride, to normalize blood cell and platelet counts and to reduce side effects of radiotherapy and chemotherapy
08/24/2010US7781422 Macrocyclic indole compounds, e.g., 16-cyclohexyl-3,6-dimethyl-17-phenyl-4,5,6,7,8,9-hexahydro-1H-13,15-(ethanediylidene)pyrrolo[2,1-f][1,2,7,10,13]thiatetraazacyclohexadecine-2,12(3H)-dione 10,10-dioxide; hepatitis C virus polymerase inhibitors
08/24/2010US7781421 such as (3 alpha ,5 alpha )-21-bromo-3-hydroxy-18,21-cyclopregn-18(21)-en-20-one used as anesthetics, anticonvulsants, anxiolytic agents or for prophylaxis of sleep disorders or drug abuse and dependence
08/24/2010US7781420 Use of clodronic acid for treatment podotrochlosis
08/24/2010US7781419 bisphosphonate is etidronate, tiludronate, risedronate, zoledronic acid; dosing schedule in a stepped-up dosage amount that is at least one and a half times the recommended dose for osteoporosis
08/24/2010US7781418 enantiomerically pure (1R,6S)-2-Azabicyclo-[4.3.0]nonane-8,8-diphosphonic acid; osteoporosis, osteolytic bone metastasis, rheumatoid arthritis and osteoarthritis; enhanced inhibitory effect on farnesyl pyrophosphate synthase
08/24/2010US7781417 Cyclodextrin dimers and derivatives thereof, methods for preparing them and their use, in particular, for the solubilizing pharmacologically active substances
08/24/2010US7781416 Inhibiting FGF growth factor with heparins; antitumor agents; angiogenesis inhibitor; antidiabetic agent treating diabetic retinopathy; antiinflammatory agent; treating retrolenticular fibroplasia, psoriasis, restenosis after angioplasty and after coronary by-pass; chemical intermediates; drug delivery
08/24/2010US7781414 Targets for tumor growth inhibition
08/24/2010US7781413 Comprises semaphorin polypeptide (SEMA3B) as tumor suppressor
08/24/2010US7781412 triclosan, hexachlorophene, or dichlorophen and anthracyclines (adriamycin, daunomycin, daunorubicin, doxorubicin, epirubicin, idarubicin); synergistic; reducing cardiotoxicity anticarcinogenic anthracycline drugs; inhibiting enzyme(s) that catalyze conversion to anthracycline metabolites
08/24/2010US7781411 Derivatives of avermectin, avermectin monosaccharide and avermectin aglycone
08/24/2010US7781410 treating acne or reducing the appearance of oil or pores on the skin, hair and scalp, comprising topical administration of 2'-hydroxy-2,3,5'-trimethoxychalcone, and optionally salicylic acid or benzoyl peroxide and a catechin
08/24/2010US7781409 Composition for external use
08/24/2010US7781408 Oral administration of gangliosides including 50% ganglioside GD3 as anticholesterol and antiinflammatory agents; decreased intestinal absorption of cholesterol; mediating inflammation of the intestine, retina or neural tissues; liquid or food suppliment for infants
08/24/2010US7781407 Reacting a gluconic acid with lactic acid in the presence of calcium hydroxide and water to obtain a calcium gluconolactate molecule having the formula HO-CH2-(CHOH)4-COO-Ca-OOC-CH(-OH)-CH3 with molecular weight of 324.2994; physical and chemical properties; nutraceuticals
08/24/2010US7781406 Modulating a transplantation-associated immune response for acute and chronic graft versus host disease (GVHD); kidney, heart and liver allogeneic transplantation; side effect reduction; biodrugs
08/24/2010US7781394 Methods for identifying anti-tumor and/or anti-angiogenesis drugs with deoxynucleoside 5′-monophosphate N-glycosidase as the target
08/24/2010US7781393 Methods for inhibiting tumor cell growth
08/24/2010US7781188 Nucleotide and protein sequences of Nogo genes and methods based thereon
08/24/2010US7781161 Detection cancer; controlling gene expression; detection hybrids
08/24/2010US7780988 Method for making homogeneous spray-dried solid amorphous drug dispersions using pressure nozzles
08/24/2010US7780987 Coating comprising aqueous dispersion of neutral ester copolymer without functional groups, polyglycol having melting point greater than 55 degrees C, pharmaceutically acceptable excipients, coated onto pharmaceutical oral dosage form, cured; FDA Orange book listed patent for metformin HCl
08/24/2010US7780986 Method of preparing sustained-release preparations of quinolone antibiotics
08/24/2010US7780984 Methods and compositions for treating proliferative diseases
08/24/2010US7780983 Amphoteric liposomes
08/24/2010US7780978 Oral pharmaceutical compositions and methods of using the same
08/24/2010US7780976 flat strip of supporting material, such as filter paper, having marked reference locations on each of one or more legs, for delivering controlled quantities of agents to the adnexa of the eye simultaneously upon dispensing liquid to strip at appropriate reference location
08/24/2010US7780959 Feline granulocyte macrophage colony stimulating factor nucleic acid molecules
08/24/2010US7780958 A biocompatible crosslinking polymer comprising acrylamide and methylene bis-acrylamide; medical procedure involves injection of polyacrylamide gel under the mucous membrane
08/24/2010US7780957 Polyethylene glycol/polycation block copolymers
08/24/2010US7780954 Glow and sunless tanning color enhancement by cationic copolymers
08/24/2010US7779715 Shifter with actuator incorporating magnetic unlock mechanism
08/24/2010CA2632585C Novel modifications to 2-amino-4-(4-fluorobenzylamino)-1-ethoxycarbonyl-aminobenzene and processes for preparing said compound
08/24/2010CA2621323C Histamine-3 receptor antagonists
08/24/2010CA2611638C Agent for the prevention and treatment of liver diseases containing pyrazolopyrimidinone derivative
08/24/2010CA2593621C Naphthalene derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2010CA2593618C Naphthalene derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2010CA2582049C Bilayer tablet comprising telmisartan and amlodipine
08/24/2010CA2572897C Pharmaceutical composition for the treatment of bone fracture
08/24/2010CA2570805C 2-(1h-indolylsulfanyl) -aryl amine derivatives for use in the treatment of affective disorders, pain, adhd and stress urinary incontinence
08/24/2010CA2557368C Polynucleotide participating in rheumatoid arthritis and utilization of the same
08/24/2010CA2551182C Novel kappa receptor selective opioid peptides
08/24/2010CA2541066C Derivatives of indanyl-piperazines, the process for preparing them and the pharmaceutical compounds that contain them
08/24/2010CA2536206C Pharmaceutical products comprising bisphosphonates
08/24/2010CA2524377C Thiadiazine derivatives and use thereof as positive ampa receptor modulators
08/24/2010CA2520897C Pyrrolo (2,1-c)(1,4) benzodiazepine dimers as antitumour agents and process thereof
08/24/2010CA2511219C Cyclopentenone derivatives for cancer therapy
08/24/2010CA2499314C Indole derivatives as beta-2 agonists
08/24/2010CA2490907C Amide derivative
08/24/2010CA2474031C Heterocyclic tripeptides as hepatitis c inhibitors
08/24/2010CA2467857C Piperidine-based mch antagonists for treatment of obesity and cns disorders
08/24/2010CA2467538C New amorphous ziprasidone hydrochloride (5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-2h-indol-2-one hydrochloride) and processes to produce the same
08/24/2010CA2464906C Improved endoprosthetic device
08/24/2010CA2463072C Thioester-terminated water soluble polymers and method of modifying the n-terminus of a polypeptide therewith
08/24/2010CA2462510C Wipe formulation
08/24/2010CA2460135C Use of pyridazinone compounds as phosphodiesterase iv inhibitors for treating cancer and other diseases
08/24/2010CA2458468C Use of non-feminizing estrogens as retinoprotective agents for the treatment of glaucoma
08/24/2010CA2445940C Prevention of epithelial cancer
08/24/2010CA2445386C Hypotensive lipid (prostaglandin derivatives) and timolol compositions and methods of using same
08/24/2010CA2436808C Liquid antimicrobial compositions
08/24/2010CA2430123C Agent for promoting excretion of accumulative chlorine-containing compound
08/24/2010CA2430122C Antiobesity agent and health food
08/24/2010CA2427520C Hydrophilic polymer blends used for dry cow therapy
08/24/2010CA2426883C Methylphenidate modified release formulations
08/24/2010CA2423103C N-acylsulfonamide apoptosis promoters
08/24/2010CA2414583C Neuroprotective 7-beta-hydroxysteroids
08/24/2010CA2391915C 3-phenyl-3,7-diazabicyclo[3.3.1]nonane compounds, process for their preparation and medicaments containing these compounds
08/24/2010CA2385655C Dna immunization against chlamydia infection
08/24/2010CA2362757C Effervescent pharmaceutical formulation containing metamizole
08/24/2010CA2345445C A composition for the prevention and/or treatment of atherosclerosis
08/24/2010CA2334858C Neuroprotective composition for the prevention and/or treatment of nervous and behavioural alterations due to anxiety states or depression
08/24/2010CA2302226C Camptothecin analogs and methods of preparation thereof
08/24/2010CA2274985C Synthetic antisense oligodeoxynucleotides targeted to human acetylcholinesterase
08/24/2010CA2273821C Detection and modulation of the iaps and naip for the diagnosis and treatment of proliferative disease
08/24/2010CA2257393C Compositions and methods for reducing respiratory depression
08/24/2010CA2256947C Depigmentation composition for lightening the skin and treating skin blotches.
08/24/2010CA2201396C Multifunctional molecular complexes for gene transfer to cells
08/24/2010CA2181924C Diagnosis and treatment of infections due to streptococci and enterococci
08/20/2010CA2655893A1 Use of voacamine and related compounds to enhance the activity of existing malaria treatments
08/20/2010CA2654839A1 Use of enoxaparin for reducing the risk of death in acutely ill medical patients
08/19/2010WO2010094040A1 Template-independent ligation of single-stranded dna
08/19/2010WO2010094009A2 Methods and compositions for the treatment of ras associated disorders
08/19/2010WO2010093992A1 Anti-fungal formulation
08/19/2010WO2010093930A1 Pharmaceutical compositions comprising (3-(1-(1h-imidazol-4-yl)ethyl)-2-methylphenyl)methanol
08/19/2010WO2010093910A1 4-(1-(3-(hydroxymethyl)-2-methylphenyl)ethyl)-1h-imidazole-2(3h)-thione
08/19/2010WO2010093890A2 Processes for producing phenyl-6-(1-(phenyl)ureido)nicotinamides)
08/19/2010WO2010093889A2 Solid forms of 2-(2, 4-difluorophenyl)-6-(1-(2,6-difluorophenyl)ureido)nicotinamide
08/19/2010WO2010093885A1 Inhibitors of akt activity
08/19/2010WO2010093873A2 Drug delivery through hydrogel plugs