Patents
Sitemap › A61 - Medical or veterinary science; Hygiene › A61K - Preparations for medical, dental, or toilet purposes › A61K 31 - Medicinal preparations containing organic active ingredients
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
12/2011
12/07/2011CN1946292B 减少共同滥用可能性的方法 Common method of reducing the likelihood of abuse
12/07/2011CN1926117B 用于改进感知、注意力、学习效率、和/或记忆力的6-氨基-5-氰基-嘧啶-4-酮类化合物 For improving perception, attention, learning efficiency, and / or memory of the 6-amino-5-cyano - pyrimidin-4-ones
12/07/2011CN1905886B 含有人参皂甙f1或化合物k的皮肤外用组合物 External composition for skin comprising ginsenoside f1 or the compound k
12/07/2011CN1875973B 一种含N<sub>3</sub>-邻甲苯甲酰基氟尿嘧啶的药物组合物及其脂质体制剂 Containing N <sub> 3 </ sub> - o-benzoyl-fluorouracil pharmaceutical compositions and liposomal formulations
12/07/2011CN1863791B {2-[1-(3,5-双-三氟甲基-苄基)-5-吡啶-4-基-1h-[1,2,3]三唑-4-基]-吡啶-3-基}-(2-氯苯基)-甲酮的新晶形 {2- [1- (3,5-bis - trifluoromethyl - benzyl) -5-pyridin-4-yl -1h- [1,2,3] triazol-4-yl] - pyridine - 3 - yl} - (2-chlorophenyl) - methanone new crystalline form of
12/07/2011CN1843504B 一种白蛋白毫微球组合药物及其制备和使用方法 One kind of albumin nanospheres combination of drugs and their preparation and use
12/07/2011CN1826324B 吲唑、苯并异*唑和苯并异噻唑激酶抑制剂 Indazole, benzoisoxazole * oxazole and benzisothiazole kinase inhibitors
12/07/2011CN1708307B 水可溶的美洛昔康颗粒 Water soluble meloxicam granules
12/07/2011CN1649598B 高剂量伊班膦酸制剂 High doses of ibandronate preparations
12/07/2011CN1494425B 用作治疗剂的羧酰胺衍生物 As therapeutic agents carboxamide derivatives
12/07/2011CN102272307A siNA介导的VEGF-C和RhoA的敲低对VEGF-A分泌、血管生成和/或新血管生成的抑制 siNA mediated knockdown of VEGF-C and VEGF-A on RhoA secretion, angiogenesis, and / or inhibiting neovascularization
12/07/2011CN102272136A 作为用于糖尿病的治疗或预防的二肽基肽酶-Ⅳ抑制剂的氨基四氢吡喃 For the treatment or prevention of dipeptidyl peptidase inhibitors for diabetes -Ⅳ aminotetrahydropyran
12/07/2011CN102272135A 唑并吡咯酮黑色素浓集激素受体-1拮抗剂 Razolo pyrrolone melanin concentrating hormone receptor-1 antagonist
12/07/2011CN102272134A Toll样受体调节剂 Toll-like receptor modulators
12/07/2011CN102272133A 淀粉样β的调节剂 A modulator of β-amyloid
12/07/2011CN102272132A 氟化苯并噻唑衍生物、其制备方法以及利用其用于诊断阿尔茨海默病的显像剂 Fluorinated benzothiazole derivatives, their preparation and the use thereof for diagnostic imaging agents for Alzheimer's disease
12/07/2011CN102272131A 哒嗪酮衍生物 Pyridazinones
12/07/2011CN102272130A [4-(6-氟-7-甲基氨基-2,4-二氧代-1,4-二氢-2h-喹唑啉-3-基)-苯基]-5-氯-噻吩-2-基-磺酰基脲盐、其相关的形式和方法 [4- (6-fluoro-7-methyl-amino-2,4-dioxo-1,4-dihydro--2h- quinazolin-3-yl) - phenyl] -5-chloro - thiophene - 2- group - sulfonylurea salt, and its related forms and methods
12/07/2011CN102272129A 硫酸化c-糖苷及其分离方法以及合成方法 C- glucoside sulfated and separation and synthesis method
12/07/2011CN102272128A Atp-结合盒转运蛋白的调节剂 Atp- binding cassette transporter protein modifier
12/07/2011CN102272127A Atp-结合盒转运蛋白调节剂 Atp- binding cassette transporter protein modifiers
12/07/2011CN102272125A 哒嗪酮衍生物 Pyridazinone derivatives
12/07/2011CN102272124A 舒尼替尼苹果酸盐的新晶形 The new crystalline form of sunitinib malate
12/07/2011CN102272121A 3-(1-{3-[5-(1-甲基-哌啶-4-基甲氧基)-嘧啶-2-基]-苄基}-6-氧代-1，6-二氢-哒嗪-3-基)-苄腈盐酸盐的新型多晶型物及其制备方法 3- (1- {3- [5- (1-methyl - piperidin-4-yl-methoxy) - pyrimidin-2-yl] - benzyl} -6-oxo-1,6-dihydro- - 3-yl) - benzonitrile hydrochloride novel polymorphs and its preparation method
12/07/2011CN102272120A 生物活性酰胺 Bioactive amides
12/07/2011CN102272119A 作为沉默调节蛋白调节剂的吡啶、双环吡啶和相关的类似物 As a sirtuin modulator of pyridine, pyridine and related bicyclic analogs
12/07/2011CN102272117A 作为hif羟化酶抑制剂的苯并噻喃衍生物 As benzothiopyrano derivative hif hydroxylase inhibitors
12/07/2011CN102272112A 苯并噻唑酮衍生物 Benzothiazole derivatives
12/07/2011CN102272111A 作为大麻素受体配体的1,2-噻唑基衍生物 1,2-thiazolyl derivatives as cannabinoid receptor ligands
12/07/2011CN102272109A 血管内造影剂 Intravascular contrast agent
12/07/2011CN102272108A 用于分析波生坦及相关物质的hplc方法以及这些物质作为参比标准和标记的用途 Hplc method for the analysis of bosentan and related substances, and these substances as a reference standard and labeling purposes
12/07/2011CN102272104A 用于治疗呼吸疾病的磺酰胺化合物 For the treatment of respiratory diseases sulfonamide compound
12/07/2011CN102272081A 四氢萘-2-醇衍生物 Tetrahydronaphthalene-2-ol derivative
12/07/2011CN102272077A 有机化合物的氟化 Fluorinated organic compounds
12/07/2011CN102271763A 抑制hdac2以促进记忆 Suppression hdac2 to promote memory
12/07/2011CN102271708A Cd37免疫治疗联合疗法及其用途 Cd37 immunotherapy and its use in combination therapy
12/07/2011CN102271688A 用于治疗hcv的环孢菌素衍生物和核苷的组合 Compositions for treating hcv cyclosporin derivatives and nucleosides
12/07/2011CN102271687A 包含轻泻剂、电解质和碳水化合物的能量营养型组合物 Energy nutritional composition comprises a laxative, electrolytes and carbohydrates
12/07/2011CN102271686A 通过反义寡核苷酸来调制Toll样受体4表达 By antisense oligonucleotides to modulate the expression of Toll-like receptor 4
12/07/2011CN102271685A 鉴定发展成器官功能衰竭的风险提高的危重患者的方法及用于其治疗的化合物 Identification develop into an increased risk of organ failure in critically ill patients for their treatment methods and compounds
12/07/2011CN102271684A 敏化多药耐受细胞的材料和方法 Materials and Methods sensitizing multidrug resistance cells
12/07/2011CN102271683A 恶性血液病的治疗 Treatment of hematologic malignancies
12/07/2011CN102271682A 用于治疗疼痛的P2X<sub>3</sub>受体拮抗剂 For the treatment of pain P2X <sub> 3 </ sub> receptor antagonist
12/07/2011CN102271681A Cxcr7调节剂 Cxcr7 moderator
12/07/2011CN102271680A 1-芳酰基-n-(2-氧代-3-哌啶基)-2-哌嗪甲酰胺类和相关化合物的化妆品应用 1-aryl acyl cosmetic applications -n- (2- oxo-3-piperidinyl) -2-piperazine carboxamides and related compounds
12/07/2011CN102271679A 包含磺酰胺的化合物及其用途 COMPOUNDS AND THEIR USE containing sulfonamide
12/07/2011CN102271678A 2-酰胺基丙醇型葡糖神经酰胺合成酶抑制剂 2-acylaminopropanol type glucosyl ceramide synthase inhibitors
12/07/2011CN102271677A 3.1.0双环G1yT1抑制剂及其制备和使用方法 3.1.0 bicyclic G1yT1 inhibitors and their preparation and use
12/07/2011CN102271676A 硫辛酸在治疗或预防陪伴动物的退行性关节病症、骨关节炎、软骨损伤，以及相关障碍中的应用 Lipoic acid treatment or prevention of degenerative joint disease in companion animals, osteoarthritis, cartilage injury, and related disorders of Application
12/07/2011CN102271675A 抗炎化合物及其组合物 Anti-inflammatory compounds, and combinations thereof
12/07/2011CN102271674A 用于治疗自身免疫病的包含dhodh抑制剂和氨甲喋呤的联合治疗 Combination therapy for the treatment of autoimmune diseases include dhodh inhibitor and methotrexate in
12/07/2011CN102271673A 尽管接受包括dpp-iv抑制剂的二甲双胍治疗但血糖控制仍不足的患者中的糖尿病的治疗 Including treatment of patients despite receiving metformin dpp-iv inhibitor but still insufficient glycemic control in diabetes
12/07/2011CN102271672A 用于治疗寄生物感染的包含单独的或与甲脒组合的1-芳基吡唑的组合物 For the treatment of parasitic infections comprising formamidine, alone or in combination with 1-aryl-pyrazole of the composition
12/07/2011CN102271671A 3，5-断-4-去甲-胆甾烷肟的新的衍生物、包含它们的药物组合物及其制备方法 3,5 breaking -4- norepinephrine - cholestane new oxime derivatives, pharmaceutical compositions containing them and preparation method
12/07/2011CN102271670A 生物油组合物，包含该生物油组合物的制剂，及其在预防或治疗心血管疾病中的应用 Bio-oil composition comprising the formulation of bio-oil composition, and its application in the prevention or treatment of cardiovascular diseases
12/07/2011CN102271669A 非大脑组织中β-淀粉样肽负载的改性 Non-brain tissues β- amyloid load modification
12/07/2011CN102271668A 表观遗传调控的小分子调节剂和其治疗应用 Epigenetic regulation of small molecule modulators and their therapeutic applications
12/07/2011CN102271667A 用于治疗椎管狭窄的5-ht2a和5-ht2b受体拮抗剂 For the treatment of spinal stenosis 5-ht2a receptor antagonist and 5-ht2b
12/07/2011CN102271665A 甾族组合物 Steroidal composition
12/07/2011CN102271663A 控制释放在低pH下水溶性差的可电离活性药物的固体组合物及其用法 Controlled release at low pH, the activity of a poorly water soluble ionizable solid pharmaceutical compositions and their use
12/07/2011CN102271657A 用于治疗阿尔茨海默病的组合物 For the treatment of Alzheimer's disease compositions
12/07/2011CN102271528A 用于抑制陪伴动物的组胺路径的含抗氧化剂的食品组合物 Companion animals for inhibiting histamine path food composition comprising an antioxidant
12/07/2011CN102271515A 吡唑并嘧啶jak抑制剂化合物和方法 Jak pyrazolopyrimidine inhibitor compounds and methods
12/07/2011CN102271514A 7-羟基-苯并咪唑-4-基-甲酮衍生物以及包含其的pbk抑制剂 7- hydroxy - benzimidazole-4-yl - methanone derivatives thereof and containing pbk inhibitor
12/07/2011CN102271509A 用于抗糖尿病药的新型环苯并咪唑衍生物 Novel ring benzimidazole derivatives for an antidiabetic drug
12/07/2011CN102271508A 含有刚性部分的吡啶并[4，3-b]吲哚类化合物 The rigid portion and containing pyridine [4,3-b] indoles
12/07/2011CN102271507A 分泌型磷脂酶A<sub>2</sub>(SPLA<sub>2</sub>)抑制剂和烟酸药物组合物以及治疗心血管疾病和血脂异常的方法 Secretory phospholipase A <sub> 2 </ sub> (SPLA <sub> 2 </ sub>) inhibitors and nicotinic acid pharmaceutical compositions and treatment of cardiovascular disease and dyslipidemia methods
12/07/2011CN102271505A (2-氨基)-四氢咔唑-丙酸的合成 (2-amino) - tetrahydro carbazole - propionic acid
12/07/2011CN102271504A 用于制备N-酰化-4-芳基β-氨基酸衍生物的方法和中间体 Method for the preparation of aryl-N- acylation -4- β- amino acid derivatives and intermediates
12/07/2011CN102271502A 增加内源性缩醛磷脂水平的方法 Increase the level of endogenous plasmalogen method
12/07/2011CN102271499A 用于向脑死亡的、心脏搏动的潜在器官供者施用的包含去甲肾上腺素和net抑制剂的组合物 For the death of the brain, the heart beat of the potential organ donor comprises administering norepinephrine and net inhibitor composition
12/07/2011CN102270281A 一种以cdk1为靶点的抗癌药物的筛选方法 Kind cdk1 targeting anticancer drug screening methods
12/07/2011CN102268467A 松乳菇菌丝多糖提取物及其应用 Mycelial Polysaccharide Extract and Its Applications
12/07/2011CN102268191A 七甲川吲哚花菁染料及其合成方法和应用 Heptamethine indocyanine dyes and synthetic method and application
12/07/2011CN102268099A 使君子提取物及其提取方法 Quisqualis extract and extraction method
12/07/2011CN102268098A 墨旱莲多糖铁络合物制备方法及其应用 Eclipta polysaccharide iron complex preparation method and its application
12/07/2011CN102268054A 一种β-胞嘧啶核苷-5'-三磷酸精氨酸衍生酯及其制备方法和应用 One kind of β- cytidine 5'-triphosphate ester derivatives of arginine and its preparation method and application
12/07/2011CN102268046A 基于9-咪蒽腙的类顺铂型配合物及其合成方法和应用 Cisplatin-based class type complexes and synthetic methods and application 9- anthracene microphone hydrazone
12/07/2011CN102268042A 一种米诺膦酸晶型ii及其制备方法 One kind of crystal ii minodronic acid and its preparation method
12/07/2011CN102268027A 具有抗肿瘤活性的酰胺类Au(III)配合物 Amides with anti-tumor activity of Au (III) complexes
12/07/2011CN102268024A 比阿培南新晶型及其合成方法 Biapenem new polymorphs and synthesis method
12/07/2011CN102268020A 头孢噻呋乙酰氧基乙基酯及其制备方法 Ceftiofur acetoxyethyl ester and its preparation method
12/07/2011CN102268014A 一类稠合杂芳基衍生物、制备方法及其应用 A class of fused heteroaryl derivatives, preparation method and application
12/07/2011CN102268013A 噻二唑衍生物、其制备方法和用途 Thiadiazole derivatives, their preparation and use
12/07/2011CN102268012A 噻唑衍生物、其制备方法和用途 Thiazole derivatives, their preparation and use
12/07/2011CN102268011A 哌嗪衍生物、其制备方法和用途 Piperazine derivatives, their preparation and use
12/07/2011CN102268005A 来源于色氨酸与脯氨酸的吲哚二酮哌嗪生物碱类化合物及其制备方法和用途 From tryptophan and proline diketopiperazine indole alkaloids and their preparation and use
12/07/2011CN102268000A 一类新型螺杂环化合物及其作为治疗剂的用途 A new class of spiro heterocyclic compounds and their use as therapeutic agents
12/07/2011CN102267998A 新型抗寄生虫吡嗪异喹啉衍生物 The new anti-parasitic pyrazine isoquinoline derivatives
12/07/2011CN102267996A 碳青霉烯类衍生物或其水合物的晶型及其制备方法 Crystal and its preparation method carbapenem derivative or hydrate
12/07/2011CN102267993A 一种多羟基去甲基托品烷类化合物及其制备方法与应用 A base plate to a polyhydroxy alkyl compounds product and its preparation method and application
12/07/2011CN102267990A 一种2,3-二氢苯并呋喃类衍生物及其制备与应用 One kind of 2,3-dihydrobenzofuran derivatives, preparation and application
12/07/2011CN102267989A 一种2-甲基苯并呋喃类化合物及其制备与应用 One kind of compounds and their preparation and application 2- methyl benzofuran
12/07/2011CN102267988A 2-氨基嘧啶衍生物及其医药用途 2-amino-pyrimidine derivatives and pharmaceutical use
12/07/2011CN102267987A 一种含氟的新抗菌化合物 A new antibacterial compounds containing fluorine
12/07/2011CN102267984A 4-羟基喹啉-3-酰胺衍生物及其制备方法和用途 4-hydroxy-quinoline-3-acid derivatives and their preparation and use
12/07/2011CN102267981A 4-甲基-n-[3-(4-甲基-咪唑-1-基)-5-三氟甲基-苯基]-3-(4-吡啶-3-基-嘧啶-2-基氨基)-苯甲酰胺的盐 4-Methyl -n- [3- (4- methyl - imidazol-1-yl) -5-trifluoromethyl - phenyl] -3- (4-pyridin-3-yl - pyrimidin-2-yl amino) - benzamide salt
12/07/2011CN102267978A 作为激酶活性调节剂的1,3-二芳基取代的脲 As the kinase activity of 1,3-diaryl-substituted urea modifier
12/07/2011CN102267977A 一种3-取代苯并[c]呋喃酮的硫代、硒代同系物、其制备方法及医药用途 One 3-substituted benzo [c] furan ketone thio, seleno homologues, their preparation and pharmaceutical use
12/07/2011CN102267971A 脂环并[c]苯并吡喃酮衍生物及其应用 Alicyclic and [c] benzopyran derivatives and their Applications
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