Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
05/2012
05/16/2012EP1919466B9 Formulations for treatment of lipoprotein abnormalities comprising a statin and a methylnicotinamide derivative
05/16/2012EP1909782B1 Compositions comprising arginine and r-alpha-lipoic acid and their use for improvement of sexual function
05/16/2012EP1909775B1 Formulation of radioprotective alpha, beta unsaturated aryl sulfones
05/16/2012EP1888615B1 17 -hsd1 and sts inhibitors
05/16/2012EP1874726B1 Organic compounds
05/16/2012EP1864665B1 Immunosuppressive agent comprising a heterocyclic compound as active ingredient
05/16/2012EP1860103B1 Anticancer compound, intermediate therefor, and processes for producing these
05/16/2012EP1836200B1 Benzisothiazole-1, 1-dioxide acting as antagonists to the vanilloid receptor subtype 1 (vr1) and uses thereof
05/16/2012EP1786428B1 Pde5 inhibitor compositions and methods for treating cardiac indications
05/16/2012EP1480993B2 Desaturase genes, enzymes encoded thereby, and uses thereof
05/16/2012EP0669809B2 Process for the heterotrophic production of microbial products with high concentrations of omega-3 highly unsaturated fatty acids
05/16/2012DE102010051404A1 Use of substituted salicylanilide compound or its salt or solvate for treating parasitosis in fish, which is an ornamental fish, preferably discus fishes, where the parasitosis is caused by parasitic Metazoa
05/16/2012DE102007037579B4 Neue Benzimidazol-2-yl-alkylamine und ihre Anwendung als mikrobizide Wirkstoffe New benzimidazol-2-yl-alkylamines and their application as microbicidal agents
05/16/2012CN1968697B Neuroprotective properties of dextrorotatory morphinans
05/16/2012CN1950397B Therapeutic use of a growth factor, NsG33
05/16/2012CN1946379B Prolonged-release compositions comprising torasemide and a matrix-forming polymer
05/16/2012CN102460163A 治疗剂和测定 Determination of the therapeutic agent and
05/16/2012CN102459611A Gene therapy for neurodegenerative disorders
05/16/2012CN102459599A Nucleic acid modulators of glycoprotein vi
05/16/2012CN102459598A Targeting micrornas for metabolic disorders
05/16/2012CN102459597A Treatment of dystrophin family related diseases by inhibition of natural antisense transcript to dmd family
05/16/2012CN102459596A Treatment of lipid transport and metabolism gene related diseases by inhibition of natural antisense transcript to a lipid transport and metabolism gene
05/16/2012CN102459594A Use of inhibitors of zdhhc2 activity for modulation of adipogenesis
05/16/2012CN102459588A Aptamer for chymase, and use thereof
05/16/2012CN102459587A Hepcidin binding nucleic acids
05/16/2012CN102459306A Novel amide derivatives of steroidal[3,2-c]pyrazole compounds with glucocorticoid activity
05/16/2012CN102459305A 具有糖皮质激素活性的甾类[3,2-c]吡唑化合物的新衍生物 The new derivatives of steroids having corticosteroid activity [3,2-c] pyrazole compounds
05/16/2012CN102459304A 用于女性保健的取代16,17-稠合的类固醇化合物 Health care for women replace 16,17 fused steroid compound
05/16/2012CN102459302A Nucleic acid delivery compositions and methods of use thereof
05/16/2012CN102459300A 用于治疗用途的新的7-脱氮嘌呤核苷 The new 7-deazapurine nucleosides for therapeutic use
05/16/2012CN102459299A N- [ (2 ' r) -2 ' -deoxy-2 ' -fluoro-2 ' -methyl-p-phenyl-5 ' -uridylyl] -l-alanine 1-methylethyl ester and process for its production
05/16/2012CN102459296A 具有抗微生物活性的酮内酯类化合物 Within one has antimicrobial activity Esters
05/16/2012CN102459291A 神经保护性化合物和它们的应用 Neuroprotective compounds and their applications
05/16/2012CN102459283A C-met 蛋白激酶的氨基吡唑三唑并噻二唑抑制剂 C-met protein kinase aminopyrazole triazolo thiadiazole inhibitor
05/16/2012CN102459282A 作为pi3-激酶抑制剂用于治疗癌症的硫杂-三氮杂-环戊二烯并薁 Sulfur as pi3- kinase inhibitors for the treatment of cancer hetero - triaza - cyclopenta azulene
05/16/2012CN102459281A 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors
05/16/2012CN102459280A 作为病毒复制抑制剂的噻吩并[2,3-b]吡啶衍生物 As inhibitors of viral replication thieno [2,3-b] pyridine derivatives
05/16/2012CN102459279A 治疗剂713 Therapeutic agent 713
05/16/2012CN102459278A 取代的-1,3,8-三氮杂螺[4.5]癸烷-2,4-二酮 Substituted triaza-spiro [4.5] decane-2,4-dione
05/16/2012CN102459272A 对P110δ具有选择性的为PI3K抑制剂的二环嘧啶化合物和使用方法 Selective for P110δ bicyclic pyrimidine compounds and methods of use for the PI3K inhibitor
05/16/2012CN102459269A 嘌呤衍生物以及使用所述嘌呤衍生物的抗肿瘤剂 Purine derivatives and purine derivative using the anti-tumor agent
05/16/2012CN102459268A Diazahomoadamantane derivatives and methods of use thereof
05/16/2012CN102459267A Dihydropyrrolonaphtyridinone compounds as inhibitors of jak
05/16/2012CN102459266A 3, 3'-螺二氢吲哚酮衍生物和它们用于癌症的用途 Uses 3, 3'-spiro-indolinone derivatives and their use for cancer
05/16/2012CN102459265A 激酶活性的嘧啶抑制剂 Pyrimidine inhibitors of kinase activity
05/16/2012CN102459264A 激酶活性的嘧啶抑制剂 Pyrimidine inhibitors of kinase activity
05/16/2012CN102459263A 取代的四氢β-咔啉的制备工艺 Preparation of substituted tetrahydro-β- carboline
05/16/2012CN102459262A 抑制raf蛋白激酶的吡咯并[2,3.b]吡啶 Inhibition of raf protein kinase pyrrolo [2,3.b] pyridine
05/16/2012CN102459261A 用于治疗变性和炎性疾病的新化合物 The new compounds for treating degenerative and inflammatory diseases for
05/16/2012CN102459260A 1H-吡唑并[4,3-c]异喹啉衍生物、其制备方法及其治疗用途 1H- pyrazolo [4,3-c] isoquinoline derivatives, their preparation and their therapeutic use
05/16/2012CN102459259A 吡唑并吡啶类 Pyrazolopyridines class
05/16/2012CN102459255A Azetidinyl diamides as monoacylglycerol lipase inhibitors
05/16/2012CN102459253A Oxazole substituted indazoles as pi3-kinase inhibitors
05/16/2012CN102459252A 用于治疗糖原合酶激酶3相关疾病诸如阿尔茨海默病的咪唑取代的嘧啶 For the treatment of glycogen synthase kinase 3-related diseases such as Alzheimer's disease pyrimidine substituted imidazole
05/16/2012CN102459251A 作为白三烯a4水解酶的调节剂的具有两个稠合双环杂芳基部分的化合物 Compound bicyclic heteroaryl moiety having two fused leukotriene a4 hydrolase as modulators of
05/16/2012CN102459250A 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors
05/16/2012CN102459249A 作为PI3K/mTOR抑制剂的苯并氧氮杂环庚三烯以及它们使用与制造方法 As the PI3K / mTOR inhibitor benzoxazepine cycloheptatriene and their use and manufacturing method
05/16/2012CN102459248A 作为PI3K/mTOR抑制剂的苯并氧杂环庚三烯以及它们使用与制造方法 As the PI3K / mTOR inhibitor benzoxepin-triene and their method of use and manufacture
05/16/2012CN102459247A 作为醛固酮合酶抑制剂的苯并噁唑酮衍生物 As aldosterone synthase inhibitors benzoxazole derivatives
05/16/2012CN102459246A 作为治疗剂的异噁唑-3(2h)-酮类似物 As therapeutic agents isoxazole -3 (2h) - one analogues
05/16/2012CN102459245A Thioxanthene derivatives for the treatment of infectious diseases
05/16/2012CN102459244A 喹唑啉二酮衍生物、其制备及其多种治疗用途 Quinazoline dione derivatives, their preparation and their therapeutic uses multiple
05/16/2012CN102459242A Phenoxymethyl heterocyclic compounds
05/16/2012CN102459240A Azetidinyl diamides as monoacylglycerol lipase inhibitors
05/16/2012CN102459238A 2,3-二氢-1h-茚化合物及其治疗癌症的用途 2,3-dihydro--1h- indene compounds and their use in the treatment of cancer
05/16/2012CN102459237A 6-(1h-咪唑-1-基)-2-苯基喹唑啉的晶型 6- (1h- imidazol-1-yl) -2-phenyl quinazoline crystalline form
05/16/2012CN102459236A 激酶活性的嘧啶抑制剂 Pyrimidine inhibitors of kinase activity
05/16/2012CN102459235A 吡嗪基吡唑 Pyrazinyl pyrazole
05/16/2012CN102459234A 作为p70s6激酶抑制剂的取代的苯并三嗪类和喹喔啉类 As the substituted benzo triazines and quinoxaline p70s6 kinase inhibitor
05/16/2012CN102459233A 二取代的酞嗪hedgehog途径拮抗剂 Disubstituted phthalazine hedgehog pathway antagonists
05/16/2012CN102459232A 7-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof, and therapeutic use thereof
05/16/2012CN102459231A 季铵盐化合物 Quaternary ammonium compounds
05/16/2012CN102459230A Azetidinyl diamides as monoacylglycerol lipase inhibitors
05/16/2012CN102459229A 用作食欲肽拮抗剂的3-氮杂二环[4.1.0]庚烷 Orexin antagonists used azabicyclo [4.1.0] heptane
05/16/2012CN102459228A Azetidinyl diamides as monoacylglycerol lipase inhibitors
05/16/2012CN102459227A Ccr2的4-氮杂环丁烷基-1-苯基-环己烷拮抗剂 Ccr2 4-azetidinyl-1-phenyl - cyclohexane antagonist
05/16/2012CN102459226A Ccr2的4-氮杂环丁烷基-1-杂原子连接的-环己烷拮抗剂 Ccr2 4-azetidinyl -1- heteroatom attached - cyclohexane antagonist
05/16/2012CN102459225A Ccr2的4-氮杂环丁烷基-1-杂芳基-环己烷拮抗剂 Ccr2 4-azetidinyl -1- heteroaryl - cyclohexane antagonist
05/16/2012CN102459224A 5-alkynyl-pyridines
05/16/2012CN102459223A 5-pyridin-3-yl-1,3-dihydro-indol-2-on derivatives and their use as modulators of aldosterone synthase and/or cyp11b1
05/16/2012CN102459222A 用作gpr119 调节剂的l-(哌啶-4-基)-吡唑衍生物 Used gpr119 modulators l- (piperidin-4-yl) - pyrazole derivatives
05/16/2012CN102459221A 噻吩衍生物 Thiophene derivative
05/16/2012CN102459220A 治疗心血管疾病的组合物及其方法 Composition for treatment of cardiovascular diseases and methods
05/16/2012CN102459218A 凝集素样氧化型ldl受体抑制用医药品以及动脉硬化预防医药品 Lectin-like oxidized ldl receptor inhibition with pharmaceuticals pharmaceuticals and atherosclerosis prevention
05/16/2012CN102459217A 影响血糖指数的化合物 Compounds on the glycemic index
05/16/2012CN102459216A Inhibitors of the renal outer medullary potassium channel
05/16/2012CN102459215A 3-(4-aminophenyl)-2-furancarboxylic acid derivative and pharmaceutically acceptable salt thereof
05/16/2012CN102459210A Arylsulfonamide ccr3 antagonists
05/16/2012CN102459207A 环戊二烯并[c]吡咯-2-甲酸酯衍生物、其制备及其治疗用途 Cyclopenta [c] pyrrole-2-carboxylic acid ester derivatives, their preparation and their therapeutic use
05/16/2012CN102459206A Oxadiazole derivatives
05/16/2012CN102459204A 溶血磷脂酸受体的多环拮抗剂 Lysophosphatidic acid receptor antagonists polycyclic
05/16/2012CN102459203A 用于调控视磺醇与视黄醇结合蛋白4(rbp4)结合的组合物和方法 Depending on the regulation of sulfur alcohol and retinol-binding protein 4 (rbp4) combination compositions and methods for
05/16/2012CN102459201A 杀真菌的1,2,4-三唑衍生物 Fungicidal 1,2,4-triazole derivatives
05/16/2012CN102459200A 适用于治疗响应于调节血清素5-ht6受体的疾病的苯磺酰基苯胺化合物 Applicable to the treatment response to serotonin 5-ht6 regulating receptor diseases Phenylsulfonylaniline compound
05/16/2012CN102459199A 适于治疗响应于5-羟色胺5-HT<sub>6</sub>受体调节的病症的苯磺酰苯胺化合物 Adapted to therapeutic response to serotonin 5-HT <sub> 6 </ sub> receptor modulated disorder benzenesulfonyl aniline compound
05/16/2012CN102459198A Crystals
05/16/2012CN102459197A 适用于治疗响应血清素5-HT<sub>6</sub>受体的调节的病症的N-苯基-(哌嗪基或高哌嗪基)-苯磺酰胺或苯磺酰基-苯基-(哌嗪或高哌嗪)化合物 Applicable to the treatment response serotonin 5-HT <sub> 6 </ sub> receptor modulated disorders of N- phenyl - (piperazinyl or homopiperazinyl) - benzenesulfonamide or benzenesulfonyl - phenyl - (piperazine or homopiperazine) compound
05/16/2012CN102459196A 用于制备罗苏伐他汀的新方法,可用于制备罗苏伐他汀的中间体化合物,以及用于制备所述中间体化合物的方法 A new method for the preparation of rosuvastatin, rosuvastatin preparing intermediate compounds, and methods for preparing the intermediate compounds may be used
05/16/2012CN102459195A 取代的1-烷基噌啉-4(1h)-酮衍生物、其制备以及其治疗用途 1-alkyl substituted cinnoline -4 (1h) - one derivatives, their preparation and their therapeutic use
05/16/2012CN102459193A 抗癌化合物和含有该化合物的药物组合物 Anti-cancer compounds and pharmaceutical compositions containing the compound